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Inhibition of CK1

PubChem AID
463857
Primary Citation
Selectively nonselective kinase inhibition: striking the right balance [PMID: 20166671]
Source
External ID
BioAssay Type
Confirmatory
Tested Substances
Tested Compounds
Version
Status
Live
Dates
  • Deposit:
    2010-09-27
  • Modify:
    2022-08-30
Description
This bioassay record (AID 463857) reports results from the above primary citation. Additional data from the same publication are reported in a total of 44 BioAssay records in PubChem.

1 Description

Title: Selectively nonselective kinase inhibition: striking the right balance.

2 Comment

Compounds with activity <= 10uM or explicitly reported as active by ChEMBL are flagged as active in this PubChem assay presentation.

Journal: J Med Chem

Year: 2010

Volume: 53

Issue: 4

First Page: 1413

Last Page: 1437

DOI: 10.1021/jm901132v

Target ChEMBL ID: CHEMBL2793

ChEMBL Target Name: Casein kinase I alpha

ChEMBL Target Type: SINGLE PROTEIN - Target is a single protein chain

Relationship Type: H - Homologous protein target assigned

Confidence: Homologous single protein target assigned

3 Result Definitions

4 Data Table

5 Target

8 Identity

8.1 BioAssay Name

Inhibition of CK1

8.2 Source

8.3 External ID

8.4 Project Category

Literature, Extracted

8.5 BioAssay Type

Confirmatory

8.6 Deposit Date

2010-09-27

8.7 Modify Date

Version 1.1
Version 1.2
Version 1.3
Version 2.1
Version 2.2
Version 2.3
Version 3.1
Version 4.1
Version 4.2
Version 5.1
Version 5.2
Version 6.1
Version 6.2
Version 7.1
Version 7.2
2022-08-30 (currently shown)

8.8 Status

Live

9 Same-Publication BioAssays

10 BioAssay Annotations

Assay Type
Binding

11 Information Sources

  1. PubChem
  2. ChEMBL
    LICENSE
    Access to the web interface of ChEMBL is made under the EBI's Terms of Use (http://www.ebi.ac.uk/Information/termsofuse.html). The ChEMBL data is made available on a Creative Commons Attribution-Share Alike 3.0 Unported License (http://creativecommons.org/licenses/by-sa/3.0/).
    http://www.ebi.ac.uk/Information/termsofuse.html
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