Xenleta
- Lefamulin
- 1061337-51-6
- Lefamulin(BC-3781)
- BC-3781
- CHEMBL3291398
- Create:2009-03-16
- Modify:2025-01-18
- BC-3781
- lefamulin
- Xenleta
- Lefamulin
- 1061337-51-6
- Lefamulin(BC-3781)
- BC-3781
- CHEMBL3291398
- Xenleta
- 1061337-51-6 (free base)
- lefamulina
- lefamuline
- [(1S,2R,3S,4S,6R,7R,8R,14R)-4-ethenyl-3-hydroxy-2,4,7,14-tetramethyl-9-oxo-6-tricyclo[5.4.3.01,8]tetradecanyl] 2-[(1R,2R,4R)-4-amino-2-hydroxycyclohexyl]sulfanylacetate
- (3aR,4R,5R,7S,8S,9R,9aS,12R)-8-hydroxy-4,7,9,12-tetramethyl-3-oxo-7-vinyldecahydro-4,9a-propanocyclopenta[8]annulen-5-yl 2-(((1R,2R,4R)-4-amino-2-hydroxycyclohexyl)thio)acetate
- BC3781
- compound 7 [PMID: 24874438]
- Lefamulin (USAN/INN)
- Lefamulin(BC-3781)?
- SCHEMBL19766421
- GTPL10824
- DTXSID101027896
- Acetic acid, 2-[[(1R,2R,4R)-4-amino-2-hydroxycyclohexyl]thio]-, (3aS,4R,5S,6S,8R,9R,9aR,10R)-6-ethenyldecahydro-5-hydroxy-4,6,9,10-tetramethyl-1-oxo-3a,9-propano-3aH-cyclopentacycloocten-8-yl ester
- EX-A3600
- BDBM50019649
- AKOS040759180
- DA-64910
- HY-16908
- TS-09691
- CS-0012945
- NS00073375
- D11631
- G92093
- Q27253537
- (3aS,4R,5S,6S,8R,9R,9aR,10R)-6-ethenyl-5-hydroxy-4,6,9,10-tetramethyl-1-oxodecahydro-3a,9-propanocyclopenta[8]annulen-8-yl {[(1R,2R,4R)-4-amino-2-hydroxycyclohexyl]sulfanyl}acetate
- 62B
- Lefamulin; Acetic acid, 2-[[(1R,2R,4R)-4-amino-2-hydroxycyclohexyl]thio]-, (3aS,4R,5S,6S,8R,9R,9aR,10R)-6-ethenyldecahydro-5-hydroxy-4,6,9,10-tetramethyl-1-oxo-3a,9-propano-3aH-cyclopentacycloocten-8-yl ester; BC 3781; Lefamulin; (3aS,4R,5S,6S,8R,9R,9aR,10R)-6-Ethen
- Lefamulin (annotation moved to)
- BC-3781 intravenous (annotation moved to)
◉ Summary of Use during Lactation
No information is available on the use of lefamulin during breastfeeding. The manufacturer recommends that mothers should avoid breastfeeding during treatment and for 2 days after the final dose. An alternate drug may be preferred, especially while nursing a newborn or preterm infant.
◉ Effects in Breastfed Infants
Relevant published information was not found as of the revision date.
◉ Effects on Lactation and Breastmilk
Relevant published information was not found as of the revision date.
Patents are available for this chemical structure:
https://patentscope.wipo.int/search/en/result.jsf?inchikey=KPVIXBKIJXZQJX-FCEONZPQSA-N
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- PATENTSCOPE (WIPO)SID 393416351https://pubchem.ncbi.nlm.nih.gov/substance/393416351