9824345 1 2 3 4 5 6 7 8 9 10 11 12 13 14 15 16 17 18 19 20 21 22 23 24 25 26 27 28 29 30 31 32 33 34 35 36 37 38 39 40 41 42 43 44 45 46 47 48 49 50 51 52 53 54 55 16 8 8 8 7 7 7 7 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 2 2 3 4 5 5 5 6 6 6 7 7 8 9 9 9 10 10 10 11 11 11 12 12 12 13 13 13 14 14 15 15 15 16 17 17 18 18 19 19 19 20 21 21 21 22 22 22 23 23 28 28 29 29 30 30 31 16 18 8 26 25 24 9 10 15 19 24 25 26 27 27 11 34 35 12 32 33 13 36 37 14 38 39 14 42 43 40 41 16 44 45 17 20 46 20 26 21 47 48 49 27 50 51 23 24 29 25 28 30 52 31 53 31 54 55 1 1 1 1 2 2 1 1 1 1 1 1 2 1 2 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 2 1 1 2 1 1 1 1 1 1 1 1 1 1 2 1 2 1 1 1 1 2 1 1 1 5 255 1 2 3 4 5 6 7 8 9 10 11 12 13 14 15 16 17 18 19 20 21 22 23 24 25 26 27 28 29 30 31 32 33 34 35 36 37 38 39 40 41 42 43 44 45 46 47 48 49 50 51 52 53 54 55 11.0608 9.3007 4.9889 4.9889 13.1486 5.2619 8.3497 8.3497 12.5853 14.1458 12.88 14.826 13.8109 14.6769 12.6486 11.6486 11.0608 10.1097 6.2619 10.1097 6.7619 3.732 3.732 4.6783 4.6783 9.3007 7.7619 2.866 2.866 2 2 14.6827 13.963 12.1636 12.0483 12.2617 12.7876 15.4031 15.1752 14.8597 15.2952 13.4616 14.2326 13.2312 12.5409 11.2524 6.8445 6.1542 9.6082 6.1793 6.8695 2.866 2.866 1.4631 1.4631 0.2111 1.4898 0.1006 3.6111 -1.464 1.8559 0.1808 1.7989 -2.2902 -1.3892 -3.2458 -2.1223 -3.6111 -3.1111 -0.5979 -0.5979 -1.407 -0.0979 1.8559 -1.0979 0.9898 2.3559 1.3559 2.6606 1.0511 0.4898 0.9898 0.8559 2.8559 1.3559 2.3559 -1.0792 -0.7968 -1.8357 -2.6002 -3.2921 -3.8588 -2.3488 -1.61 -3.7036 -3.0648 -4.1234 -4.0656 -0.3859 0.0126 -1.9966 2.0679 2.4664 -1.4624 0.7778 0.3793 0.2359 3.4759 1.0459 2.6659 8 8 8 8 8 8 8 8 8 8 8 8 8 8 8 8 1 1 2 2 7 7 8 16 17 18 22 22 23 28 29 30 16 18 8 26 26 27 27 17 20 20 23 29 28 30 31 31 0 Compound Canonicalized 5 2010.07.16 1 Compound Complexity 7 E_COMPLEXITY 3.402 Cactvs xemistry.com 2012.05.21 633 Count Hydrogen Bond Acceptor 5 E_NHACCEPTORS 3.402 Cactvs xemistry.com 2012.05.21 7 Count Hydrogen Bond Donor 5 E_NHDONORS 3.402 Cactvs xemistry.com 2012.05.21 0 Count Rotatable Bond 5 E_NROTBONDS 3.402 Cactvs xemistry.com 2012.05.21 6 Fingerprint SubStructure Keys 16 extended 2 E_SCREEN 3.402 Cactvs xemistry.com 2012.05.21 00000371E07BB000400000000000000000000000000162C4800030000000058000005801F000001E04040000000C00C1DB04311187181008AD02237236008380892408B0698839380CD8882EB2A0DD1184310864C723A889879DC8808E80000000001000000000000000200000000000000000 IUPAC Name Allowed 1 2.1.0 LexiChem openeye.com 2012.05.21 2-[2-[5-[5-(azepan-1-ylmethyl)-2-thienyl]-1,2,4-oxadiazol-3-yl]ethyl]isoindoline-1,3-dione IUPAC Name CAS-like Style 1 2.1.0 LexiChem openeye.com 2012.05.21 2-[2-[5-[5-(1-azepanylmethyl)-2-thiophenyl]-1,2,4-oxadiazol-3-yl]ethyl]isoindole-1,3-dione IUPAC Name Preferred 1 2.1.0 LexiChem openeye.com 2012.05.21 2-[2-[5-[5-(azepan-1-ylmethyl)thiophen-2-yl]-1,2,4-oxadiazol-3-yl]ethyl]isoindole-1,3-dione IUPAC Name Systematic 1 2.1.0 LexiChem openeye.com 2012.05.21 2-[2-[5-[5-(azepan-1-ylmethyl)thiophen-2-yl]-1,2,4-oxadiazol-3-yl]ethyl]isoindole-1,3-dione IUPAC Name Traditional 1 2.1.0 LexiChem openeye.com 2012.05.21 2-[2-[5-[5-(azepan-1-ylmethyl)-2-thienyl]-1,2,4-oxadiazol-3-yl]ethyl]isoindoline-1,3-quinone InChI Standard 1 1.0.4 InChI iupac.org 2012.05.21 InChI=1S/C23H24N4O3S/c28-22-17-7-3-4-8-18(17)23(29)27(22)14-11-20-24-21(30-25-20)19-10-9-16(31-19)15-26-12-5-1-2-6-13-26/h3-4,7-10H,1-2,5-6,11-15H2 InChIKey Standard 1 1.0.4 InChI iupac.org 2012.05.21 QUKKMGJVXHURCY-UHFFFAOYSA-N Log P XLogP3-AA 7 3.0 sioc-ccbg.ac.cn 2012.05.21 3.6 Mass Exact 7 2.1 PubChem ncbi.nlm.nih.gov 2012.05.21 436.156912 Molecular Formula 1 2.1 PubChem ncbi.nlm.nih.gov 2012.05.21 C23H24N4O3S Molecular Weight 7 2.1 PubChem ncbi.nlm.nih.gov 2012.05.21 436.52666 SMILES Canonical 1 1.7.6 OEChem openeye.com 2012.05.21 C1CCCN(CC1)CC2=CC=C(S2)C3=NC(=NO3)CCN4C(=O)C5=CC=CC=C5C4=O SMILES Isomeric 1 1.7.6 OEChem openeye.com 2012.05.21 C1CCCN(CC1)CC2=CC=C(S2)C3=NC(=NO3)CCN4C(=O)C5=CC=CC=C5C4=O Topological Polar Surface Area 7 E_TPSA 3.402 Cactvs xemistry.com 2012.05.21 108 Weight MonoIsotopic 7 2.1 PubChem ncbi.nlm.nih.gov 2012.05.21 436.156912 31 0 0 0 0 0 0 0 1 1