754726
1
2
3
4
5
6
7
8
9
10
11
12
13
14
15
16
17
18
19
20
21
22
23
24
25
26
27
28
29
30
31
32
33
34
9
9
9
7
7
7
7
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
1
1
1
1
1
1
1
1
1
1
1
1
2
3
4
4
4
5
5
6
7
8
9
9
10
10
11
12
12
13
13
14
16
16
17
17
18
18
18
19
19
19
20
21
23
23
23
15
15
15
6
8
9
8
10
14
22
12
11
15
11
13
24
14
22
16
17
18
20
25
21
26
27
28
29
20
21
23
30
31
32
33
34
1
1
1
1
1
1
1
2
2
3
2
2
1
1
1
1
1
1
2
1
1
1
1
2
1
1
1
1
2
1
1
1
1
1
1
1
2
5
10
1
2
3
4
5
6
7
8
9
10
11
12
13
14
15
16
17
18
19
20
21
22
23
24
25
26
27
28
29
30
31
32
33
34
-0.9414
-2.6041
-2.5951
-1.8534
0.1169
-3.2099
-1.9531
-1.2373
-1.0969
0.8177
0.2434
-2.2474
2.3015
-3.4297
-1.8158
3.0637
2.9234
-4.8181
5.0813
4.4555
4.3152
-2.0858
6.5696
0.8715
2.6184
2.3475
-5.0019
-5.5452
-5.0125
5.0418
4.7913
6.9983
6.8967
6.9769
3.8214
2.8773
2.9618
0.3023
-1.0805
0.1792
-4.4563
-0.9488
1.4816
0.0168
1.3988
-1.8829
-0.0815
-1.1337
2.7963
0.9359
-1.1912
-1.6294
-0.2665
0.8435
-1.2838
-3.2954
-0.3649
2.2759
1.7983
-1.9921
-2.2211
-0.8104
-2.2635
1.6393
-2.1518
0.1369
-1.4095
0.0972
-0.1293
-1.1766
1.0017
0.0001
0.0249
0.0108
0.1185
0.0276
-0.0396
0.0022
-0.0432
0.0563
0.0032
0.0447
-0.0859
0.5722
-0.5646
0.0649
0.0056
0.5733
-0.5635
0.0904
0.0062
-0.1131
1.0585
-1.0205
0.9676
0.0497
-0.8063
1.0252
-1.0121
0.8804
0.0444
-0.8986
Conformer
ID
11
2.1
PubChem
ncbi.nlm.nih.gov
2009.12.11
000B842600000001
Energy
MMFF94 NoEstat
7
1.7.2
Szybki
openeye.com
2012.11.26
48.0332
Feature
Self Overlap
7
2.1
PubChem
ncbi.nlm.nih.gov
2012.11.26
30.574
Fingerprint
Shape
2
2.1
PubChem
ncbi.nlm.nih.gov
2012.11.26
10319926 262 18268692958624713194
10411042 1 18122063379638359035
10493431 412 18125449609564707881
10616163 171 18411420622575900702
1100329 8 18192715764067641691
11056379 131 18411146814104634094
12107183 9 17685768031153099066
12173636 292 18193555558395333268
12236239 1 17530682109175704626
12403259 226 18199181966154064088
12403259 415 17989198258016117976
12553582 1 18337094778630252915
12788726 201 18260823800094254162
13140716 1 18195532721015187827
138480 1 16176789313263769513
14508225 48 18339911731936849389
14790565 3 18339086973910495793
14863182 85 15739103056183650391
15042514 8 18337676433229655643
15230672 131 17976549313184668870
15927050 60 17981889636506002381
15961568 22 18191021412608031364
16087824 20 18337671920215955741
17844677 252 18410580591803072148
1813 80 17676484007716873668
19141452 34 18200316649016449231
19591789 44 17978798908893172955
20510252 161 18341892957200224505
20600515 1 18127992960410832371
20693207 138 17844272665098130430
21065198 57 18411699855900948962
21236236 1 18341894060790671361
21267235 1 18337398239328208834
22122407 14 15841283660664828930
22182313 1 17846227609873222838
2297311 6 18411427228055727822
23366157 5 17321822401951715413
23402539 116 18343297094037301623
23557571 272 18272658935187848404
23559900 14 18340480183891154048
23845131 108 17619927062858371897
266924 87 18266449902926579311
283562 15 18339922619979455795
3178227 256 18263096564783281211
335352 9 18338234977158327359
350125 39 18413393159378912128
4214541 1 18411700946574806768
4409770 3 18261663814625573359
5104073 3 18270675364972342498
559249 180 18117835509112332466
59755656 215 18411136926995661742
7364860 26 17474389553121660121
81228 2 18335428975558873777
9709674 26 18343025463125815302
Shape
Multipoles
8
1.8.3
OEShape
openeye.com
2012.11.26
431.58
10.31
4.03
0.72
13.95
0.57
-0.02
-3.94
0.24
-5.65
-0.07
0.07
0.19
0.63
Shape
Self Overlap
7
2.1
PubChem
ncbi.nlm.nih.gov
2012.11.26
951.224
Shape
Volume
7
1.8.3
OEShape
openeye.com
2012.11.26
234.5
Conformer
RMSD
7
2009.12.11
0.6
Diverse Conformer
ID List
6
2010.05.05
1
Charge
MMFF94 Partial
2
1.7.6
OEChem
openeye.com
2012.05.21
28
1 -0.34
10 0.35
11 -0.14
12 0.02
13 0.09
14 0.11
15 1.16
16 -0.15
17 -0.15
18 0.18
19 -0.14
2 -0.34
20 -0.15
21 -0.15
22 0.54
23 0.14
24 0.15
25 0.15
26 0.15
3 -0.34
30 0.15
31 0.15
4 0.6
5 -0.58
6 -0.71
7 -0.56
8 -0.03
9 -0.17
Count
Effective Rotor
7
1.7.6
OEChem
ncbi.nlm.nih.gov
2012.01.18
2
Features
Pharmacophore
2
ImplicitMillsDean merged
1.8.1
OEShape
openeye.com
2012.05.21
6
1 5 acceptor
1 6 acceptor
1 7 acceptor
5 4 6 8 12 14 rings
6 13 16 17 19 20 21 rings
6 4 5 8 9 10 11 rings
23
0
0
0
0
0
0
0
1
1