744789
1
2
3
4
5
6
7
8
9
10
11
12
13
14
15
16
17
18
19
20
21
22
23
24
25
35
8
8
8
7
6
6
6
6
6
6
6
6
6
6
1
1
1
1
1
1
1
1
1
1
1
2
3
3
4
5
5
5
6
6
6
6
7
7
7
9
9
10
11
11
13
13
14
14
15
10
8
12
25
12
8
9
20
7
8
16
17
12
18
19
10
11
13
14
21
15
22
15
23
24
1
2
1
1
2
1
1
1
1
1
1
1
1
1
1
1
2
2
1
1
1
1
2
1
1
2
5
10
1
2
3
4
5
6
7
8
9
10
11
12
13
14
15
16
17
18
19
20
21
22
23
24
25
2.3791
-0.7072
-5.5905
-4.5975
0.4001
-2.0079
-3.2057
-0.7018
1.7672
2.7635
2.0753
-4.5127
4.1006
3.4125
4.4251
-2.0293
-2.0291
-3.1826
-3.1839
0.2225
1.3625
4.9038
3.6669
5.4661
-6.4339
2.8888
-1.6424
-0.6492
1.3949
0.431
0.362
-0.5796
-0.4148
0.0663
1.03
-1.2859
0.1739
0.6324
-1.6833
-0.7242
1.0053
1.0107
-1.2172
-1.2188
1.4332
-2.0956
1.365
-2.7393
-1.0338
-0.1482
0.0114
0.0103
0.0177
-0.0258
0.0017
0.002
-0.0009
-0.0011
0
0.0035
-0.0059
-0.0013
0.0013
-0.0082
-0.0047
0.8899
-0.882
-0.8921
0.8892
0.0027
-0.0108
0.004
-0.0132
-0.0066
0.0123
Conformer
ID
11
2.1
PubChem
ncbi.nlm.nih.gov
2009.12.11
000B5D5500000001
Energy
MMFF94 NoEstat
7
1.7.2
Szybki
openeye.com
2012.11.26
34.628
Feature
Self Overlap
7
2.1
PubChem
ncbi.nlm.nih.gov
2012.11.26
35.579
Fingerprint
Shape
2
2.1
PubChem
ncbi.nlm.nih.gov
2012.11.26
11471102 20 18410575089411694390
13081056 2 18335700559526607933
13167823 11 18342172293552584823
13675066 3 18114185258955681915
14123238 8 18187365428405978303
15196674 1 18410575063547282861
17834072 33 18341891930940456415
17844677 252 18411145736136680609
18186145 218 17894622669402840991
200 152 18131349700480011251
20606313 2 18410575089580557908
20645477 70 18340488876504274862
21267235 1 18340495478274891710
212847 35 18333453144716276420
22289505 5 18337104579861556620
23402539 116 18130780144903864069
23402655 69 18342457040966820644
23558518 356 17682958061383996634
23559900 14 18342174492585935122
3060560 45 18059864965349443166
351380 180 18409728456836938161
3545911 37 18412265064131416234
4047638 21 18411419531527054810
42 15 18334014969156027559
4214541 1 18410856547382680613
42788 4 18410575076273740807
5104073 3 18408886273563107587
522135 26 18408604751626670310
58051976 100 18340206392188968967
602551 16 15937269917788819657
69090 78 18411696599567035655
7364860 26 18341049718119078208
77779 3 18410293618693086223
8272917 22 18343306933390736326
9709674 26 18411143566619494631
9971528 1 18272368655580895792
Shape
Multipoles
8
1.8.3
OEShape
openeye.com
2012.11.26
292.05
10.65
2.12
0.6
13.21
1.33
0
-0.06
0.01
-2.15
0
-0.09
0.03
0.02
Shape
Self Overlap
7
2.1
PubChem
ncbi.nlm.nih.gov
2012.11.26
586.62
Shape
Volume
7
1.8.3
OEShape
openeye.com
2012.11.26
173.9
Conformer
RMSD
7
2009.12.11
0.6
Diverse Conformer
ID List
6
2012.02.08
1
35
41
9
18
23
46
20
13
42
34
24
15
16
45
3
27
50
26
10
44
12
2
29
47
17
22
38
11
48
6
25
5
36
7
14
39
30
28
43
21
8
19
31
49
37
4
40
32
33
Charge
MMFF94 Partial
2
1.7.6
OEChem
openeye.com
2012.02.08
21
1 -0.11
10 0.11
11 -0.15
12 0.66
13 -0.15
14 -0.15
15 -0.15
2 -0.57
20 0.37
21 0.15
22 0.15
23 0.15
24 0.15
25 0.5
3 -0.65
4 -0.57
5 -0.55
6 0.06
7 0.06
8 0.57
9 0.12
Count
Effective Rotor
7
1.7.6
OEChem
ncbi.nlm.nih.gov
2012.01.18
5
Features
Pharmacophore
2
ImplicitMillsDean merged
1.8.1
OEShape
openeye.com
2012.02.08
7
1 1 hydrophobe
1 2 acceptor
1 3 acceptor
1 4 acceptor
1 5 donor
3 3 4 12 anion
6 9 10 11 13 14 15 rings
15
0
0
0
0
0
0
0
1
2