70679366 1 2 3 4 5 6 7 8 9 10 11 12 13 14 15 16 17 18 19 20 21 22 23 24 25 26 27 28 29 30 31 32 33 34 35 36 37 38 39 40 41 42 43 44 45 46 47 48 49 8 8 8 8 8 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 2 2 3 4 4 5 6 6 6 6 7 7 7 8 8 8 9 9 9 10 10 10 11 11 11 12 12 13 13 13 14 14 15 15 15 16 16 16 16 17 17 18 18 20 21 22 22 12 14 22 48 19 23 49 23 7 8 24 25 9 26 27 10 28 29 11 30 31 12 32 33 13 34 35 36 37 38 39 40 17 18 19 20 21 19 22 41 42 20 43 21 44 45 46 23 47 1 1 1 1 2 1 1 2 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 2 1 1 2 1 1 1 1 1 1 1 2 1 1 1 1 1 22 2 16 23 47 3 1 2 5 10 1 2 3 4 5 6 7 8 9 10 11 12 13 14 15 16 17 18 19 20 21 22 23 24 25 26 27 28 29 30 31 32 33 34 35 36 37 38 39 40 41 42 43 44 45 46 47 48 49 Conformer RMSD 7 2012.11.26 1.2 Diverse Conformer ID List 6 2012.11.26 7 69 56 85 78 45 43 74 1 25 51 9 16 65 23 55 21 3 39 47 29 52 37 11 77 10 28 35 26 12 87 24 57 4 59 19 27 40 80 22 70 49 82 58 53 5 33 63 72 2 20 81 15 76 30 8 62 64 60 17 14 44 84 41 71 73 54 38 18 66 6 13 79 83 31 50 67 48 34 86 36 46 75 68 42 32 61 Charge MMFF94 Partial 2 1.9.0 OEChem openeye.com 2012.11.26 22 1 -0.36 12 0.28 14 0.08 15 0.09 16 0.06 17 -0.15 18 -0.15 19 0.42 2 -0.68 20 -0.15 21 -0.15 22 0.34 23 0.66 3 -0.57 4 -0.65 43 0.15 44 0.15 45 0.15 46 0.15 48 0.4 49 0.5 5 -0.57 Count Effective Rotor 7 1.9.0 OEChem ncbi.nlm.nih.gov 2012.11.26 12 Features Pharmacophore 2 ImplicitMillsDean merged 1.8.3 OEShape openeye.com 2012.11.26 11 1 1 acceptor 1 13 hydrophobe 1 2 acceptor 1 2 donor 1 3 acceptor 1 4 acceptor 1 5 acceptor 3 4 5 23 anion 3 6 8 10 hydrophobe 3 7 9 11 hydrophobe 6 14 15 17 18 20 21 rings 23 1 0 1 0 0 0 0 1 2