70634767 1 2 3 4 5 6 7 8 9 10 11 12 13 14 15 16 17 18 19 20 21 22 23 24 25 26 27 28 29 30 31 32 33 34 35 36 37 38 39 40 41 42 43 44 45 46 47 48 49 50 51 52 53 54 55 8 8 8 8 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 2 3 3 4 4 5 5 5 5 6 6 6 7 7 7 8 8 8 9 9 9 11 11 12 12 13 13 14 14 15 15 15 16 17 17 18 18 18 19 19 19 20 20 21 22 23 23 24 24 24 25 25 25 10 13 10 16 54 21 55 6 7 9 26 8 27 28 10 29 30 11 31 32 33 34 35 12 36 18 19 14 17 15 16 20 37 38 22 21 39 43 44 45 40 41 42 23 46 22 47 24 25 50 51 52 48 49 53 1 1 2 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 2 1 1 1 1 2 1 2 1 1 1 1 1 1 1 1 1 1 1 1 2 1 2 1 1 1 1 1 1 1 1 1 5 6 7 9 26 3 1 2 5 10 1 2 3 4 5 6 7 8 9 10 11 12 13 14 15 16 17 18 19 20 21 22 23 24 25 26 27 28 29 30 31 32 33 34 35 36 37 38 39 40 41 42 43 44 45 46 47 48 49 50 51 52 53 54 55 Conformer RMSD 7 2012.11.26 1.2 Diverse Conformer ID List 6 2012.11.26 6 37 112 109 82 136 139 114 2 113 25 4 48 115 27 67 121 143 64 106 92 8 117 34 79 80 73 146 86 155 132 28 56 36 95 35 111 72 137 94 59 101 53 77 7 39 85 147 99 145 144 119 65 148 151 45 18 74 11 135 157 128 102 118 110 47 98 41 57 40 108 22 60 104 152 51 122 58 134 156 127 142 83 21 153 138 107 89 149 70 26 62 71 125 15 84 141 61 29 13 38 24 54 126 5 44 63 158 120 105 16 50 76 20 69 14 133 1 66 30 49 33 154 116 159 129 123 87 97 103 31 12 17 78 81 90 19 100 3 23 93 131 55 52 96 9 75 91 130 32 88 10 124 43 150 68 140 42 46 Charge MMFF94 Partial 2 1.9.0 OEChem openeye.com 2012.11.26 28 1 -0.23 10 0.66 11 -0.29 12 -0.28 13 0.08 14 -0.14 15 0.28 16 0.08 17 -0.15 18 0.14 19 0.14 2 -0.57 20 -0.29 21 0.08 22 -0.15 23 -0.28 24 0.14 25 0.14 3 -0.53 36 0.15 39 0.15 4 -0.53 46 0.15 47 0.15 54 0.45 55 0.45 7 0.06 8 0.14 Count Effective Rotor 7 1.9.0 OEChem ncbi.nlm.nih.gov 2012.11.26 9 Features Pharmacophore 2 ImplicitMillsDean merged 1.8.3 OEShape openeye.com 2012.11.26 8 1 2 acceptor 1 3 donor 1 4 donor 1 9 hydrophobe 3 12 18 19 hydrophobe 3 23 24 25 hydrophobe 5 5 6 7 8 11 hydrophobe 6 13 14 16 17 21 22 rings 25 1 0 1 0 0 0 0 1 9