70611433 1 2 3 4 5 6 7 8 9 10 11 12 13 14 15 16 17 18 19 20 21 22 23 24 25 26 27 28 29 30 31 32 33 34 35 36 37 38 39 40 41 42 8 8 8 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 2 3 4 4 4 4 5 5 5 6 6 6 7 7 7 8 8 8 9 9 10 10 11 11 12 12 13 13 13 14 15 16 16 16 17 17 17 19 20 20 20 18 42 18 19 5 6 10 21 8 24 25 7 22 23 9 28 29 9 26 27 30 31 11 12 14 32 15 33 14 15 16 35 36 17 18 34 19 37 38 20 39 40 41 1 1 2 2 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 2 1 1 1 2 1 2 1 1 1 1 1 1 1 1 1 1 1 1 1 1 16 13 17 18 34 3 1 2 5 10 1 2 3 4 5 6 7 8 9 10 11 12 13 14 15 16 17 18 19 20 21 22 23 24 25 26 27 28 29 30 31 32 33 34 35 36 37 38 39 40 41 42 Conformer RMSD 7 2012.11.26 0.8 Diverse Conformer ID List 6 2012.11.26 1 75 91 66 21 72 29 73 22 3 65 64 11 51 45 31 82 53 58 23 61 26 87 67 25 41 93 77 30 48 12 80 83 55 49 40 2 88 60 85 28 94 17 38 32 10 39 90 89 81 24 63 19 7 15 47 57 79 42 35 9 68 84 6 18 92 76 95 54 52 44 70 20 59 13 71 27 16 33 78 43 8 14 50 37 56 4 34 46 36 69 62 5 86 74 Charge MMFF94 Partial 2 1.9.0 OEChem openeye.com 2012.11.26 20 1 -0.65 10 -0.14 11 -0.15 12 -0.15 13 -0.14 14 -0.15 15 -0.15 16 0.2 17 0.06 18 0.66 19 0.45 2 -0.57 20 0.06 3 -0.57 32 0.15 33 0.15 35 0.15 36 0.15 4 0.14 42 0.5 Count Effective Rotor 7 1.9.0 OEChem ncbi.nlm.nih.gov 2012.11.26 6.2 Features Pharmacophore 2 ImplicitMillsDean merged 1.8.3 OEShape openeye.com 2012.11.26 6 1 1 acceptor 1 2 acceptor 1 3 acceptor 3 1 2 18 anion 6 10 11 12 13 14 15 rings 6 4 5 6 7 8 9 rings 20 1 0 1 0 0 0 0 1 3