70256963 1 2 3 4 5 6 7 8 9 10 11 12 13 14 15 16 17 18 19 20 21 22 23 24 25 26 27 28 29 30 31 32 33 34 35 36 37 38 39 40 9 8 8 8 8 8 8 8 7 6 6 6 6 6 6 6 6 6 6 6 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 2 2 3 3 4 4 5 5 6 6 7 7 8 9 9 9 10 10 10 11 11 12 12 13 13 14 15 15 16 16 17 17 17 18 18 19 20 20 20 13 11 14 12 31 14 32 15 35 16 36 18 40 19 10 19 27 11 12 21 15 22 13 23 14 24 17 16 25 18 26 28 29 30 33 34 20 37 38 39 1 1 1 1 1 1 1 1 1 1 1 1 1 2 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 10 9 11 12 21 1 1 11 2 15 10 22 2 1 12 3 13 10 23 2 1 13 1 12 14 24 3 1 14 2 4 13 17 1 1 15 5 11 16 25 1 1 16 6 15 18 26 1 1 2 5 10 1 2 3 4 5 6 7 8 9 10 11 12 13 14 15 16 17 18 19 20 21 22 23 24 25 26 27 28 29 30 31 32 33 34 35 36 37 38 39 40 Conformer RMSD 7 2012.05.21 0.8 Diverse Conformer ID List 6 2012.05.21 1 57 53 66 67 46 20 65 27 23 44 59 30 15 64 41 12 52 49 38 35 47 4 16 60 28 51 61 42 17 37 19 14 54 8 34 48 43 39 62 29 11 55 13 56 9 32 25 58 31 22 24 3 50 40 63 45 26 18 10 7 21 2 33 36 6 5 Charge MMFF94 Partial 2 1.7.6 OEChem openeye.com 2012.05.21 25 1 -0.34 10 0.3 11 0.28 12 0.28 13 0.34 14 0.56 15 0.28 16 0.28 18 0.28 19 0.57 2 -0.56 20 0.06 27 0.37 3 -0.68 31 0.4 32 0.4 35 0.4 36 0.4 4 -0.68 40 0.4 5 -0.68 6 -0.68 7 -0.68 8 -0.57 9 -0.73 Count Effective Rotor 7 1.7.6 OEChem ncbi.nlm.nih.gov 2012.05.21 6.2 Features Pharmacophore 2 ImplicitMillsDean merged 1.8.1 OEShape openeye.com 2012.05.21 14 1 2 acceptor 1 3 acceptor 1 3 donor 1 4 acceptor 1 4 donor 1 5 acceptor 1 5 donor 1 6 acceptor 1 6 donor 1 7 acceptor 1 7 donor 1 8 acceptor 1 9 donor 6 2 10 11 12 13 14 rings 20 7 6 1 0 0 0 0 1 2