70053351 1 2 3 4 5 6 7 8 9 10 11 12 13 14 15 16 17 18 19 20 21 22 16 8 8 8 7 6 6 6 6 6 6 1 1 1 1 1 1 1 1 1 1 1 1 1 2 2 3 3 4 5 5 5 6 6 7 7 7 8 8 9 9 9 10 10 6 8 10 21 11 22 11 6 7 14 9 12 8 11 13 15 16 10 17 18 19 20 1 1 1 1 1 1 2 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 6 1 5 9 12 3 1 7 5 8 11 13 3 1 2 5 10 1 2 3 4 5 6 7 8 9 10 11 12 13 14 15 16 17 18 19 20 21 22 Conformer RMSD 7 2012.05.21 0.6 Diverse Conformer ID List 6 2012.05.21 1 56 9 70 57 64 39 31 22 55 19 58 69 47 68 41 40 2 72 74 49 37 65 17 46 48 8 62 35 59 4 43 15 53 13 51 34 71 54 25 66 32 45 61 44 60 52 27 26 75 6 67 36 30 73 18 10 3 33 23 14 38 63 20 16 24 5 11 12 50 29 21 42 28 7 Charge MMFF94 Partial 2 1.7.6 OEChem openeye.com 2012.05.21 13 1 -0.46 10 0.28 11 0.66 14 0.36 2 -0.68 21 0.4 22 0.5 3 -0.65 4 -0.57 5 -0.9 6 0.5 7 0.33 8 0.23 Count Effective Rotor 7 1.7.6 OEChem ncbi.nlm.nih.gov 2012.05.21 4 Features Pharmacophore 2 ImplicitMillsDean merged 1.8.1 OEShape openeye.com 2012.05.21 8 1 2 acceptor 1 2 donor 1 3 acceptor 1 4 acceptor 1 5 cation 1 5 donor 3 3 4 11 anion 5 1 5 6 7 8 rings 11 2 0 2 0 0 0 0 1 1