70029275 1 2 3 4 5 6 7 8 9 10 11 12 13 14 15 16 17 18 19 20 21 22 23 24 25 26 27 28 29 30 31 32 33 34 35 36 37 38 39 40 41 42 43 44 45 46 47 48 49 50 51 52 53 54 55 56 57 58 59 60 61 62 63 64 65 66 67 68 69 70 71 72 73 74 75 76 17 8 8 8 8 8 8 7 7 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 2 2 3 4 4 5 5 6 7 7 8 8 8 9 9 9 10 10 10 11 11 12 12 12 12 13 13 14 14 14 15 15 15 15 16 16 17 17 17 18 18 18 19 19 20 20 20 21 21 22 24 24 24 25 25 25 26 26 26 27 27 28 28 29 29 31 32 32 34 34 35 36 36 37 38 38 38 39 39 33 10 17 23 31 38 30 72 30 35 39 11 13 19 16 20 23 11 14 40 41 42 13 24 25 26 43 44 23 45 46 16 18 30 47 48 49 22 27 50 21 51 52 22 28 21 53 54 55 56 29 57 59 60 61 62 63 58 64 65 31 34 32 66 33 67 35 33 68 36 69 37 37 70 71 39 73 74 75 76 1 1 1 2 1 1 1 1 2 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 2 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 2 1 2 1 2 1 1 1 1 2 1 2 1 1 1 1 1 1 1 1 10 2 14 11 40 2 1 15 16 18 30 47 1 1 17 2 27 22 50 2 1 1 5 255 1 2 3 4 5 6 7 8 9 10 11 12 13 14 15 16 17 18 19 20 21 22 23 24 25 26 27 28 29 30 31 32 33 34 35 36 37 38 39 40 41 42 43 44 45 46 47 48 49 50 51 52 53 54 55 56 57 58 59 60 61 62 63 64 65 66 67 68 69 70 71 72 73 74 75 76 12.6647 8.2439 6.81 7.7178 2.31 3.81 8.1782 9.2188 5.31 7.81 8.2439 8.7083 9.4413 6.81 3.81 4.81 9.2188 3.31 10.0006 4.81 3.81 10.0006 6.31 7.9752 9.3884 8.0281 9.4413 10.8946 10.8946 3.31 8.7083 11.8007 11.8007 10.3969 8.9308 10.6194 9.8864 6.9488 7.1806 7.4801 7.6394 8.2439 9.7777 10.0126 6.9177 6.2274 3.19 5.3926 4.7023 8.6178 2.835 2.835 4.7023 5.3926 3.2274 3.9177 7.5535 8.4826 7.5207 8.3969 8.934 9.8102 9.843 7.6064 7.5736 10.8874 10.8874 12.3364 10.8514 11.2119 10.0243 2 6.3768 6.6151 7.1066 6.5614 0.5431 0.4199 -2.2131 1.9752 0.385 1.251 3.9927 -1.6045 -1.347 -0.481 -1.382 -3.2596 -2.5794 -0.481 -0.481 -0.481 0.6425 -1.347 -0.981 -2.2131 -2.2131 0.019 -1.347 -3.9398 -3.9927 -2.5266 1.6174 -1.5157 0.5536 0.385 2.2976 -1.0018 0.0398 1.9122 3.2725 2.8871 3.5672 2.6778 3.6933 0.0439 -1.52 -2.002 -3.1003 -2.3386 0.1296 -0.269 -0.481 -0.269 0.1296 1.2435 -0.9485 -1.7456 -2.8237 -2.4251 -2.4251 -2.8237 -3.4853 -2.1049 -4.3615 -4.3943 -4.4144 -4.4472 -3.571 -2.0721 -2.9483 -2.1356 1.1736 -1.3139 1.4904 3.0698 4.1717 0.9219 2.9172 2.1553 4.3089 3.7258 6 5 6 8 8 8 8 8 8 8 8 8 8 8 8 10 15 17 19 19 22 27 27 28 29 31 32 34 35 36 14 30 50 22 28 29 31 34 32 33 35 33 36 37 37 0 Compound Canonicalized 5 2012.11.26 1 Compound Complexity 7 E_COMPLEXITY 3.408 Cactvs xemistry.com 2012.11.26 867 Count Hydrogen Bond Acceptor 5 E_NHACCEPTORS 3.408 Cactvs xemistry.com 2012.11.26 7 Count Hydrogen Bond Donor 5 E_NHDONORS 3.408 Cactvs xemistry.com 2012.11.26 1 Count Rotatable Bond 5 E_NROTBONDS 3.408 Cactvs xemistry.com 2012.11.26 6 Fingerprint SubStructure Keys 16 extended 2 E_SCREEN 3.408 Cactvs xemistry.com 2012.11.26 00000371F07B38000400000000000000000000000000000000003C6881000580000000914000001E02000800000F1EE1982632CE83000600880225D258008208002127000888010EEE880F273EC5B39B87782AE7E611DAE807DCD1F30E00004120000A40000000824000148000000000000000 IUPAC Name Allowed 1 2.2.0 LexiChem openeye.com 2012.11.26 (3R)-1-[2-[(3S,5R)-7-chloro-5-(2,3-dihydro-1,4-benzodioxin-5-yl)-1-(2,2-dimethylpropyl)-3,5-dihydro-2H-4,1-benzoxazepin-3-yl]acetyl]piperidine-3-carboxylic acid IUPAC Name CAS-like Style 1 2.2.0 LexiChem openeye.com 2012.11.26 (3R)-1-[2-[(3S,5R)-7-chloro-5-(2,3-dihydro-1,4-benzodioxin-5-yl)-1-(2,2-dimethylpropyl)-3,5-dihydro-2H-4,1-benzoxazepin-3-yl]-1-oxoethyl]-3-piperidinecarboxylic acid IUPAC Name Preferred 1 2.2.0 LexiChem openeye.com 2012.11.26 (3R)-1-[2-[(3S,5R)-7-chloro-5-(2,3-dihydro-1,4-benzodioxin-5-yl)-1-(2,2-dimethylpropyl)-3,5-dihydro-2H-4,1-benzoxazepin-3-yl]acetyl]piperidine-3-carboxylic acid IUPAC Name Systematic 1 2.2.0 LexiChem openeye.com 2012.11.26 (3R)-1-[2-[(3S,5R)-7-chloranyl-5-(2,3-dihydro-1,4-benzodioxin-5-yl)-1-(2,2-dimethylpropyl)-3,5-dihydro-2H-4,1-benzoxazepin-3-yl]ethanoyl]piperidine-3-carboxylic acid IUPAC Name Traditional 1 2.2.0 LexiChem openeye.com 2012.11.26 (3R)-1-[2-[(3S,5R)-7-chloro-5-(2,3-dihydro-1,4-benzodioxin-5-yl)-1-neopentyl-3,5-dihydro-2H-4,1-benzoxazepin-3-yl]acetyl]nipecotic acid InChI Standard 1 1.0.4 InChI iupac.org 2012.11.26 InChI=1S/C30H37ClN2O6/c1-30(2,3)18-33-17-21(15-26(34)32-11-5-6-19(16-32)29(35)36)39-27(23-14-20(31)9-10-24(23)33)22-7-4-8-25-28(22)38-13-12-37-25/h4,7-10,14,19,21,27H,5-6,11-13,15-18H2,1-3H3,(H,35,36)/t19-,21+,27+/m1/s1 InChIKey Standard 1 1.0.4 InChI iupac.org 2012.11.26 AHAHFDPYRBUSFQ-NUANOYTQSA-N Log P XLogP3-AA 7 3.0 sioc-ccbg.ac.cn 2012.11.26 4.8 Mass Exact 7 2.1 PubChem ncbi.nlm.nih.gov 2012.11.26 556.234015 Molecular Formula 1 2.1 PubChem ncbi.nlm.nih.gov 2012.11.26 C30H37ClN2O6 Molecular Weight 7 2.1 PubChem ncbi.nlm.nih.gov 2012.11.26 557.07758 SMILES Canonical 1 1.9.0 OEChem openeye.com 2012.11.26 CC(C)(C)CN1CC(OC(C2=C1C=CC(=C2)Cl)C3=C4C(=CC=C3)OCCO4)CC(=O)N5CCCC(C5)C(=O)O SMILES Isomeric 1 1.9.0 OEChem openeye.com 2012.11.26 CC(C)(C)CN1C[C@@H](O[C@H](C2=C1C=CC(=C2)Cl)C3=C4C(=CC=C3)OCCO4)CC(=O)N5CCC[C@H](C5)C(=O)O Topological Polar Surface Area 7 E_TPSA 3.408 Cactvs xemistry.com 2012.11.26 88.5 Weight MonoIsotopic 7 2.1 PubChem ncbi.nlm.nih.gov 2012.11.26 556.234015 39 3 3 0 0 0 0 0 1 1