70029123 1 2 3 4 5 6 7 8 9 10 11 12 13 14 15 16 17 18 19 20 21 22 23 24 25 26 27 28 29 30 31 32 33 34 35 36 37 38 39 40 41 42 43 44 45 46 47 48 49 50 51 52 53 54 55 56 57 58 59 60 61 62 63 64 65 66 67 68 69 70 71 72 73 74 75 76 77 17 8 8 8 8 8 8 8 7 7 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 2 2 3 4 5 5 6 7 7 8 8 9 9 9 10 10 10 11 11 11 11 12 12 13 13 13 14 14 14 15 15 16 16 16 16 17 17 17 18 18 19 19 19 22 22 22 23 23 24 25 25 25 26 26 26 27 27 27 29 29 30 30 31 31 32 32 34 35 35 36 37 37 38 39 39 39 40 40 40 33 17 22 20 21 28 69 28 34 39 36 40 12 15 20 18 21 23 12 13 28 41 42 43 14 44 45 15 46 47 48 49 18 25 26 27 19 21 50 51 52 20 53 54 24 29 55 24 30 31 56 57 58 59 60 61 62 63 64 34 35 32 65 33 66 33 67 36 37 68 38 38 70 71 72 73 74 75 76 77 1 1 1 2 2 1 1 2 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 2 1 1 1 1 1 1 1 1 1 1 1 2 1 2 1 2 1 1 1 1 2 1 2 1 1 1 1 1 1 1 1 1 11 12 13 28 41 3 1 17 2 19 21 50 1 1 22 2 29 24 55 2 1 1 5 255 1 2 3 4 5 6 7 8 9 10 11 12 13 14 15 16 17 18 19 20 21 22 23 24 25 26 27 28 29 30 31 32 33 34 35 36 37 38 39 40 41 42 43 44 45 46 47 48 49 50 51 52 53 54 55 56 57 58 59 60 61 62 63 64 65 66 67 68 69 70 71 72 73 74 75 76 77 12.6647 8.2439 6.81 7.6204 2.31 3.81 11.13 11.575 5.31 9.2188 3.81 4.81 3.31 3.81 4.81 9.1466 7.81 9.4413 6.81 6.31 8.2439 9.2188 10.0006 10.0006 8.8518 10.1022 8.191 3.31 9.4413 10.8946 10.8946 11.8007 11.8007 10.3969 8.7083 10.6194 8.9308 9.8864 12.0855 11.7975 4.12 5.3926 4.7023 2.835 2.835 3.2274 3.9177 4.7023 5.3926 7.4801 9.9355 8.8218 6.2274 6.9177 8.6178 8.2594 8.6691 9.4443 9.9195 10.6947 10.2849 8.3738 7.5986 8.0083 10.8874 10.8874 12.3364 8.1158 2 8.4763 10.0243 12.2683 12.678 11.9028 12.402 11.9355 11.1931 0.71 0.5869 1.4179 -1.9969 2.284 3.15 1.3989 3.3487 0.5519 -1.4376 1.4179 1.4179 0.5519 -0.3141 -0.3141 -3.3681 -0.3141 -2.4125 -0.3141 0.5519 -1.2151 0.8094 -0.8141 0.1859 -4.3237 -3.6628 -3.0734 2.284 1.7843 -1.3488 0.7206 -0.8349 0.2067 2.0791 2.4645 3.054 3.4394 3.7342 1.6936 4.3237 1.9549 1.63 2.0285 0.9504 0.1534 -0.5262 -0.9247 -0.9247 -0.5262 0.2109 -2.7869 -2.3893 -0.5262 -0.9247 1.4104 -4.1409 -4.9161 -4.5064 -4.2553 -3.8455 -3.0703 -2.4809 -2.8906 -3.6658 -1.9687 1.3405 -1.147 2.2817 2.8209 3.8611 4.3386 1.1012 1.8764 2.2861 4.1857 4.9281 4.4616 3 6 6 8 8 8 8 8 8 8 8 8 8 8 8 11 17 22 23 23 24 29 29 30 31 32 34 35 36 37 28 19 55 24 30 31 34 35 32 33 33 36 37 38 38 0 Compound Canonicalized 5 2012.11.26 1 Compound Complexity 7 E_COMPLEXITY 3.408 Cactvs xemistry.com 2012.11.26 911 Count Hydrogen Bond Acceptor 5 E_NHACCEPTORS 3.408 Cactvs xemistry.com 2012.11.26 7 Count Hydrogen Bond Donor 5 E_NHDONORS 3.408 Cactvs xemistry.com 2012.11.26 1 Count Rotatable Bond 5 E_NROTBONDS 3.408 Cactvs xemistry.com 2012.11.26 8 Fingerprint SubStructure Keys 16 extended 2 E_SCREEN 3.408 Cactvs xemistry.com 2012.11.26 00000371F07B38000400000000000000000000000000000000003C6080000580000000014000001E02000800000F1EE1982632CE83000600880225D258028208002127000888014EEE880F273EC5B39F87702A67E611DAE807DDD1F30E00004120000A40000000824000148000000000000000 IUPAC Name Allowed 1 2.2.0 LexiChem openeye.com 2012.11.26 1-[2-[(3S,5R)-7-chloro-5-(2,3-dimethoxyphenyl)-1-(2,2-dimethylpropyl)-2-oxo-5H-4,1-benzoxazepin-3-yl]acetyl]piperidine-3-carboxylic acid IUPAC Name CAS-like Style 1 2.2.0 LexiChem openeye.com 2012.11.26 1-[2-[(3S,5R)-7-chloro-5-(2,3-dimethoxyphenyl)-1-(2,2-dimethylpropyl)-2-oxo-5H-4,1-benzoxazepin-3-yl]-1-oxoethyl]-3-piperidinecarboxylic acid IUPAC Name Preferred 1 2.2.0 LexiChem openeye.com 2012.11.26 1-[2-[(3S,5R)-7-chloro-5-(2,3-dimethoxyphenyl)-1-(2,2-dimethylpropyl)-2-oxo-5H-4,1-benzoxazepin-3-yl]acetyl]piperidine-3-carboxylic acid IUPAC Name Systematic 1 2.2.0 LexiChem openeye.com 2012.11.26 1-[2-[(3S,5R)-7-chloranyl-5-(2,3-dimethoxyphenyl)-1-(2,2-dimethylpropyl)-2-oxidanylidene-5H-4,1-benzoxazepin-3-yl]ethanoyl]piperidine-3-carboxylic acid IUPAC Name Traditional 1 2.2.0 LexiChem openeye.com 2012.11.26 1-[2-[(3S,5R)-7-chloro-5-(2,3-dimethoxyphenyl)-2-keto-1-neopentyl-5H-4,1-benzoxazepin-3-yl]acetyl]nipecotic acid InChI Standard 1 1.0.4 InChI iupac.org 2012.11.26 InChI=1S/C30H37ClN2O7/c1-30(2,3)17-33-22-12-11-19(31)14-21(22)26(20-9-6-10-23(38-4)27(20)39-5)40-24(28(33)35)15-25(34)32-13-7-8-18(16-32)29(36)37/h6,9-12,14,18,24,26H,7-8,13,15-17H2,1-5H3,(H,36,37)/t18?,24-,26-/m0/s1 InChIKey Standard 1 1.0.4 InChI iupac.org 2012.11.26 JRSHGFNBFYKGIE-FVKAUKPSSA-N Log P XLogP3-AA 7 3.0 sioc-ccbg.ac.cn 2012.11.26 4.2 Mass Exact 7 2.1 PubChem ncbi.nlm.nih.gov 2012.11.26 572.228929 Molecular Formula 1 2.1 PubChem ncbi.nlm.nih.gov 2012.11.26 C30H37ClN2O7 Molecular Weight 7 2.1 PubChem ncbi.nlm.nih.gov 2012.11.26 573.07698 SMILES Canonical 1 1.9.0 OEChem openeye.com 2012.11.26 CC(C)(C)CN1C2=C(C=C(C=C2)Cl)C(OC(C1=O)CC(=O)N3CCCC(C3)C(=O)O)C4=C(C(=CC=C4)OC)OC SMILES Isomeric 1 1.9.0 OEChem openeye.com 2012.11.26 CC(C)(C)CN1C2=C(C=C(C=C2)Cl)[C@@H](O[C@H](C1=O)CC(=O)N3CCCC(C3)C(=O)O)C4=C(C(=CC=C4)OC)OC Topological Polar Surface Area 7 E_TPSA 3.408 Cactvs xemistry.com 2012.11.26 106 Weight MonoIsotopic 7 2.1 PubChem ncbi.nlm.nih.gov 2012.11.26 572.228929 40 3 2 1 0 0 0 0 1 2