68632730
1
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43
9
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6
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6
6
6
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6
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6
1
1
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1
1
1
1
1
1
1
1
1
2
2
3
3
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19
19
19
20
21
21
22
22
23
23
25
25
25
26
26
26
20
17
25
18
26
5
9
19
11
12
15
24
42
43
9
10
11
15
12
14
13
16
20
21
17
27
28
18
29
18
30
31
32
22
23
33
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34
24
35
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37
38
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40
41
1
1
1
1
1
1
1
1
2
1
2
1
1
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2
1
1
1
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2
1
2
2
1
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1
1
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2
1
1
1
1
2
1
2
1
1
1
1
1
1
1
1
1
2
5
10
1
2
3
4
5
6
7
8
9
10
11
12
13
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15
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17
18
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20
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32
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36
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43
2.1955
-1.9161
-4.4648
0.9188
1.9509
-2.642
4.5932
-0.0566
-0.3083
-1.1543
1.3554
-2.4428
2.1837
-0.9754
-1.5921
-3.53
-2.0873
-3.3634
1.1847
2.5777
2.5903
3.3783
3.3906
3.7847
-0.574
-4.9966
0.0297
-1.8199
-4.5395
0.8325
2.2589
0.6534
2.2908
3.6781
3.7001
-0.0458
-0.0323
-0.6265
-5.8642
-4.2544
-5.3206
4.8886
4.8798
0.0542
-3.0574
-1.955
3.3832
2.5243
2.437
-3.2893
1.4165
2.7812
0.5254
1.3299
1.104
0.1503
-0.8725
3.2946
0.2364
-1.7071
-1.1527
4.8028
-0.4523
-0.3891
-1.5943
-1.5312
-2.1339
-3.5412
-2.3639
-1.2638
4.352
0.6457
5.2394
4.9723
5.235
0.0678
-2.0547
-1.9426
-3.2714
-3.2291
-4.6347
-3.003
-2.9372
-1.4941
-3.6804
-3.7263
-2.2575
0.2236
0.215
0.0542
0.0664
0.102
0.1965
0.1066
0.077
0.1352
0.0983
0.1313
0.1188
0.166
0.0745
0.1591
0.1931
0.1896
0.0202
-1.076
1.3393
-1.0502
1.365
0.1703
0.225
-1.0434
0.1676
0.0521
0.1577
0.958
-0.0906
-0.8313
2.2796
-1.988
2.3224
-0.6961
1.1245
0.2507
-0.8575
-1.608
-1.6237
1.0811
-0.6693
Conformer
ID
11
2.1
PubChem
ncbi.nlm.nih.gov
2012.05.21
0417409A00000001
Energy
MMFF94 NoEstat
7
1.7.2
Szybki
openeye.com
2012.11.26
101.2717
Feature
Self Overlap
7
2.1
PubChem
ncbi.nlm.nih.gov
2012.11.26
50.874
Fingerprint
Shape
2
2.1
PubChem
ncbi.nlm.nih.gov
2012.11.26
10319926 262 17907552768145009586
10411042 1 18410572877298438851
10616163 171 18048599214139084290
10967382 1 18050287260924489489
1100329 8 18339082584448261449
11578080 2 17531787105202996604
11582403 64 15896087422551382160
12363563 72 18411702079876545207
12553582 1 18338529611049604403
12788726 201 18120677746215991460
12839892 36 17907842252476039104
13140716 1 18269556052659712289
138480 1 14735917726165227754
14790565 3 17907315251088272024
14863182 85 17615134712115096821
14866123 147 18195809557833465803
15042514 8 18121786032219392561
15230672 131 16823905834453492662
16728300 4 17107580336555179264
16752209 62 18263360283293563987
17492 89 18339921636284777975
19591789 44 17763474919949983921
19930381 70 18266175230967438859
20028762 73 18201438022628512213
20600515 1 18127692634723147456
20645477 70 18051692445506506199
20905425 154 18268718392466419692
21197605 99 14734247340903438538
21421861 104 18191587651756607369
23184049 29 18410291415037526160
23419403 2 17559368341109965224
23559900 14 18196085762383864787
335352 9 18338516323201473613
34934 24 17835798977995686217
59755656 215 18193837278380488292
7364860 26 18124598840566666960
9709674 26 18266742561692088779
Shape
Multipoles
8
1.8.3
OEShape
openeye.com
2012.11.26
496.13
7.55
5.38
1.03
1.67
3.74
0.28
-8.02
0.5
-0.21
-0.13
-0.81
-0.34
-0.5
Shape
Self Overlap
7
2.1
PubChem
ncbi.nlm.nih.gov
2012.11.26
1112.524
Shape
Volume
7
1.8.3
OEShape
openeye.com
2012.11.26
267.1
Conformer
RMSD
7
2012.05.21
0.6
Diverse Conformer
ID List
6
2012.05.21
1
4
2
5
6
3
Charge
MMFF94 Partial
2
1.7.6
OEChem
openeye.com
2012.05.21
32
1 -0.19
11 0.23
12 0.31
13 0.05
14 -0.15
15 0.16
16 -0.15
17 0.08
18 0.08
19 0.26
2 -0.36
20 0.19
21 -0.15
22 -0.15
23 -0.15
24 0.1
25 0.28
26 0.28
27 0.15
28 0.15
29 0.15
3 -0.36
33 0.15
34 0.15
35 0.15
4 0.31
42 0.4
43 0.4
5 -0.71
6 -0.62
7 -0.9
9 -0.15
Count
Effective Rotor
7
1.7.6
OEChem
ncbi.nlm.nih.gov
2012.05.21
3
Features
Pharmacophore
2
ImplicitMillsDean merged
1.8.1
OEShape
openeye.com
2012.05.21
10
1 2 acceptor
1 3 acceptor
1 5 acceptor
1 6 acceptor
1 7 cation
1 7 donor
5 4 5 8 9 11 rings
6 10 12 14 16 17 18 rings
6 13 20 21 22 23 24 rings
6 6 8 9 10 12 15 rings
26
0
0
0
0
0
0
0
1
2