60620005 1 2 3 4 5 6 7 8 9 10 11 12 13 14 15 16 17 18 19 20 21 22 23 24 25 26 27 28 29 30 31 32 33 34 35 36 37 38 39 40 41 42 43 44 45 46 47 48 49 50 51 52 53 54 55 56 57 58 59 16 8 8 8 7 7 7 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 2 3 3 4 4 5 5 5 6 6 6 7 7 8 8 8 9 9 9 10 10 10 11 11 11 12 12 13 13 14 14 14 15 15 16 17 17 18 18 19 19 19 20 20 21 21 22 23 24 25 26 26 27 27 28 29 29 30 31 32 32 24 25 16 28 32 30 32 8 11 14 13 16 46 23 25 9 13 33 10 34 35 12 36 37 12 38 39 40 41 42 43 15 44 45 17 18 19 20 47 21 48 23 49 50 22 51 22 52 53 24 54 26 27 29 28 55 30 31 56 31 57 58 59 1 1 2 1 1 1 1 1 1 1 1 1 1 1 2 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 2 1 1 1 1 2 1 1 1 1 2 1 1 1 1 2 1 1 2 1 1 1 2 2 1 1 1 1 1 8 5 9 13 33 3 1 1 5 255 1 2 3 4 5 6 7 8 9 10 11 12 13 14 15 16 17 18 19 20 21 22 23 24 25 26 27 28 29 30 31 32 33 34 35 36 37 38 39 40 41 42 43 44 45 46 47 48 49 50 51 52 53 54 55 56 57 58 59 9.9443 7.7861 14.4021 14.4021 5.5714 7.9671 10.7533 6.5659 7.1537 6.7469 5.1646 5.7524 6.9726 4.9836 3.989 8.3739 3.4013 3.5823 9.3684 2.4067 2.5878 2 9.7751 9.2751 10.8578 11.7238 12.5899 13.4559 11.7238 13.4559 12.5899 14.9857 6.2014 7.5844 7.6677 7.3485 6.7037 4.7339 4.6506 5.9233 5.1952 6.371 7.0159 4.8127 5.5408 8.3316 3.6534 3.9467 9.97 9.3251 2.0423 2.3356 1.3834 8.6585 12.5899 11.1869 12.5899 15.4466 15.4466 -2.3964 -0.5781 -2.1849 -3.7943 2.267 1.1444 -0.9951 2.1625 2.9715 3.8851 3.1806 3.9896 1.249 1.458 1.5626 0.2309 0.7535 2.4761 0.1264 0.8581 2.5806 1.7716 -0.7872 -1.6532 -1.9896 -2.4896 -1.9896 -2.4896 -3.4896 -3.4896 -3.9896 -2.9896 1.6609 2.5255 3.3182 4.0351 4.5036 3.6266 2.8339 4.5856 4.2614 1.099 0.6305 0.862 1.1862 1.646 0.1871 2.9777 0.2764 0.7449 0.3565 3.147 1.8364 -1.718 -1.3696 -3.7996 -4.6096 -3.4043 -2.5749 8 8 8 8 3 8 8 8 8 8 8 8 8 8 8 8 8 8 1 1 7 7 8 15 15 17 18 20 21 23 26 26 27 28 29 30 24 25 23 25 13 17 18 20 21 22 22 24 27 29 28 30 31 31 0 Compound Canonicalized 5 2012.05.21 1 Compound Complexity 7 E_COMPLEXITY 3.402 Cactvs xemistry.com 2012.05.21 617 Count Hydrogen Bond Acceptor 5 E_NHACCEPTORS 3.402 Cactvs xemistry.com 2012.05.21 6 Count Hydrogen Bond Donor 5 E_NHDONORS 3.402 Cactvs xemistry.com 2012.05.21 1 Count Rotatable Bond 5 E_NROTBONDS 3.402 Cactvs xemistry.com 2012.05.21 7 Fingerprint SubStructure Keys 16 extended 2 E_SCREEN 3.402 Cactvs xemistry.com 2012.05.21 00000371E07B30004000000000000000000000000001624000003C608000000000004801D000001E04100000000C2CC5DE07B08F93C81408AC032572540082F8A0612A380888B53EAC981D66BAA4F51BB4302A64D611AEA807B0D0120E20000100000040004000020000008000000000000000 IUPAC Name Allowed 1 2.1.0 LexiChem openeye.com 2012.05.21 2-[2-(1,3-benzodioxol-5-yl)thiazol-4-yl]-N-[(1-benzyl-2-piperidyl)methyl]acetamide IUPAC Name CAS-like Style 1 2.1.0 LexiChem openeye.com 2012.05.21 2-[2-(1,3-benzodioxol-5-yl)-4-thiazolyl]-N-[[1-(phenylmethyl)-2-piperidinyl]methyl]acetamide IUPAC Name Preferred 1 2.1.0 LexiChem openeye.com 2012.05.21 2-[2-(1,3-benzodioxol-5-yl)-1,3-thiazol-4-yl]-N-[(1-benzylpiperidin-2-yl)methyl]acetamide IUPAC Name Systematic 1 2.1.0 LexiChem openeye.com 2012.05.21 2-[2-(1,3-benzodioxol-5-yl)-1,3-thiazol-4-yl]-N-[[1-(phenylmethyl)piperidin-2-yl]methyl]ethanamide IUPAC Name Traditional 1 2.1.0 LexiChem openeye.com 2012.05.21 2-[2-(1,3-benzodioxol-5-yl)thiazol-4-yl]-N-[(1-benzyl-2-piperidyl)methyl]acetamide InChI Standard 1 1.0.4 InChI iupac.org 2012.05.21 InChI=1S/C25H27N3O3S/c29-24(26-14-21-8-4-5-11-28(21)15-18-6-2-1-3-7-18)13-20-16-32-25(27-20)19-9-10-22-23(12-19)31-17-30-22/h1-3,6-7,9-10,12,16,21H,4-5,8,11,13-15,17H2,(H,26,29) InChIKey Standard 1 1.0.4 InChI iupac.org 2012.05.21 SJSIPQZIKKUVCD-UHFFFAOYSA-N Log P XLogP3-AA 7 3.0 sioc-ccbg.ac.cn 2012.05.21 4.1 Mass Exact 7 2.1 PubChem ncbi.nlm.nih.gov 2012.05.21 449.177313 Molecular Formula 1 2.1 PubChem ncbi.nlm.nih.gov 2012.05.21 C25H27N3O3S Molecular Weight 7 2.1 PubChem ncbi.nlm.nih.gov 2012.05.21 449.56518 SMILES Canonical 1 1.7.6 OEChem openeye.com 2012.05.21 C1CCN(C(C1)CNC(=O)CC2=CSC(=N2)C3=CC4=C(C=C3)OCO4)CC5=CC=CC=C5 SMILES Isomeric 1 1.7.6 OEChem openeye.com 2012.05.21 C1CCN(C(C1)CNC(=O)CC2=CSC(=N2)C3=CC4=C(C=C3)OCO4)CC5=CC=CC=C5 Topological Polar Surface Area 7 E_TPSA 3.402 Cactvs xemistry.com 2012.05.21 91.9 Weight MonoIsotopic 7 2.1 PubChem ncbi.nlm.nih.gov 2012.05.21 449.177313 32 1 0 1 0 0 0 0 1 2