59459452
1
2
3
4
5
6
7
8
9
10
11
12
13
14
15
16
17
18
19
20
21
22
23
24
25
26
27
28
29
16
8
8
7
6
6
6
6
6
6
6
6
6
6
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
2
2
3
4
4
5
5
5
5
7
7
7
8
8
8
9
9
9
10
10
11
11
11
12
13
13
13
6
10
14
29
14
6
12
6
7
8
9
15
22
23
16
17
18
19
20
21
11
12
13
24
25
26
14
27
28
1
1
1
1
2
2
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
2
1
1
1
1
1
1
1
2
5
10
1
2
3
4
5
6
7
8
9
10
11
12
13
14
15
16
17
18
19
20
21
22
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27
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29
-0.5672
4.9438
4.6769
-1.5958
-3.285
-1.879
-3.3862
-4.2923
-3.7125
0.4793
1.9199
-0.2434
2.7376
4.204
-4.4142
-5.3094
-4.3154
-4.0332
-4.7524
-3.0971
-3.6393
-3.0649
-2.7535
2.062
2.3332
0.1688
2.6342
2.3786
5.8913
-0.666
-1.1187
0.32
1.383
-0.4148
0.2071
-1.7649
0.5491
-0.6686
0.6252
0.5578
1.6211
-0.3148
-0.3155
-2.1452
0.1412
1.5169
0.737
-1.0124
-1.4322
0.2481
-1.6583
-2.5329
0.1934
1.5757
2.5502
0.065
-1.3496
-1.1184
0.6518
-0.8734
0.8642
-0.5426
-0.0003
-0.0277
-0.746
-0.6638
1.4616
0.2283
0.5408
-0.3946
-0.4289
-0.0695
-0.7478
-0.6406
-0.149
-1.7125
1.5126
1.9501
2.0587
-1.7887
-0.2876
1.5673
0.5357
-0.7652
-1.4516
-0.3993
-0.6194
Conformer
ID
11
2.1
PubChem
ncbi.nlm.nih.gov
2012.05.21
038B477C00000001
Energy
MMFF94 NoEstat
7
1.7.2
Szybki
openeye.com
2012.11.26
20.1164
Feature
Self Overlap
7
2.1
PubChem
ncbi.nlm.nih.gov
2012.11.26
30.505
Fingerprint
Shape
2
2.1
PubChem
ncbi.nlm.nih.gov
2012.11.26
10680689 15 18410014325274912401
11046707 91 18341328972207189831
11132069 177 18341891909064706190
11401426 45 18335132103066215537
11543360 7 14418137356547020282
12032990 46 18261397779586851649
12251169 10 12175615187669981104
13760787 19 16225760818351614825
14252887 29 17988649584122362558
14911166 2 18040146327879591101
14993402 34 16660364783504380702
17834074 16 18343864407324015662
18186145 218 16370721577813417405
19141452 34 18202003248440028599
200 152 17632852027762561853
20279233 1 18273496767005428063
20281407 28 18413106164735755608
20281475 54 18272938253653048532
20325693 3 16805323297489513419
20374829 77 18409443678835126614
20432913 95 17989489619305910570
20645476 183 16153708751725840755
20645477 70 18341607144158715398
20871999 31 17894629227575543125
21119208 17 16443063898160269598
22485316 2 18342735217429850758
23402539 116 18040990744003530126
23557571 272 18262803939200707300
23559900 14 18260547840567616424
26918003 58 17346878940392837122
42 15 16343989095899065200
Shape
Multipoles
8
1.8.3
OEShape
openeye.com
2012.11.26
275.24
9.74
1.39
1.02
8.25
0.07
0.17
-2.97
-0.72
-0.71
-0.29
-0.39
-0.2
0.55
Shape
Self Overlap
7
2.1
PubChem
ncbi.nlm.nih.gov
2012.11.26
539.826
Shape
Volume
7
1.8.3
OEShape
openeye.com
2012.11.26
167.9
Conformer
RMSD
7
2012.05.21
0.6
Diverse Conformer
ID List
6
2012.05.21
1
5
17
23
7
6
25
16
14
29
3
24
11
15
22
26
2
18
9
19
27
20
28
21
10
8
13
12
4
Charge
MMFF94 Partial
2
1.7.6
OEChem
openeye.com
2012.05.21
13
1 -0.08
10 -0.14
11 0.18
12 0.08
13 0.06
14 0.66
2 -0.65
26 0.15
29 0.5
3 -0.57
4 -0.57
5 0.18
6 0.2
Count
Effective Rotor
7
1.7.6
OEChem
ncbi.nlm.nih.gov
2012.05.21
4
Features
Pharmacophore
2
ImplicitMillsDean merged
1.8.1
OEShape
openeye.com
2012.05.21
6
1 2 acceptor
1 3 acceptor
1 4 acceptor
3 2 3 14 anion
4 5 7 8 9 hydrophobe
5 1 4 6 10 12 rings
14
0
0
0
0
0
0
0
1
1