5916053
1
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5
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53
54
55
8
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8
8
8
8
8
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6
6
6
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6
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6
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6
6
6
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
4
-1
6
-1
12
1
13
1
1
2
3
4
5
6
7
8
8
8
9
9
10
10
10
11
11
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34
34
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37
37
38
21
25
27
12
12
13
13
15
21
42
16
17
26
27
45
14
24
29
32
54
55
16
20
22
18
21
24
39
40
20
23
25
41
23
43
44
27
28
29
30
34
35
31
33
46
32
47
33
48
36
49
37
50
38
51
38
52
53
2
2
2
1
2
1
2
1
1
1
1
2
1
1
1
1
2
1
1
1
1
2
1
1
1
1
1
1
1
2
1
1
1
2
1
1
1
1
2
1
2
1
1
2
1
2
1
1
1
1
1
2
1
2
1
1
1
1
11
-1
14
24
27
18
2
1
2
5
10
1
2
3
4
5
6
7
8
9
10
11
12
13
14
15
16
17
18
19
20
21
22
23
24
25
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27
28
29
30
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34
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36
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38
39
40
41
42
43
44
45
46
47
48
49
50
51
52
53
54
55
-1.9311
5.1399
-4.6299
-1.2055
0.2376
-1.5421
-0.0581
0.1199
-1.2366
-2.8987
-5.0289
-0.7443
-1.0026
-5.5877
0.837
0.1484
-1.8951
-3.3788
2.9191
2.2159
-1.2386
0.866
2.2453
-4.1631
4.3553
-2.4066
-3.9218
4.9496
-1.3575
-2.9902
-0.8921
-1.4757
-2.5249
4.1186
6.3353
4.6733
6.8898
6.0588
-3.6342
-3.6891
2.738
0.6218
0.3543
2.7839
-2.4468
-3.8052
-0.0724
-3.0029
3.0364
7.0054
4.0264
7.9687
6.4907
-6.2498
-4.8795
-4.1453
-2.3142
-0.187
1.1301
0.3583
5.9567
5.7015
-3.3251
-2.1899
0.0444
-2.0772
1.0771
5.2642
-0.9257
-2.5877
-2.0298
-2.8738
-3.0573
-1.6822
-2.4194
-3.5154
-1.2923
-1.119
-1.9696
-1.5001
1.3539
-0.5732
-0.3488
1.8605
2.1428
3.1563
3.945
3.4383
0.6
-0.2231
1.6748
0.8517
1.8006
-3.0433
-4.0304
-2.8598
-3.73
-0.8461
-0.5417
-0.4905
1.823
3.5322
4.0251
0.5379
-0.9478
2.414
0.95
2.6374
-1.13
-0.3176
1.5111
-1.3042
-1.3582
2.9859
1.5227
-1.5372
0.0603
0.8255
-1.3579
0.2425
1.0148
1.8219
-0.6406
1.4259
-0.1224
-1.202
-0.4765
-0.6241
-0.9312
0.0196
0.7249
-2.1491
-2.0143
0.0561
-0.7946
0.0369
-0.4437
-0.0504
0.804
-0.9544
0.5797
-0.4118
-1.1788
0.5455
0.0492
1.2405
0.7443
1.34
-1.69
-0.2321
0.8659
1.6103
-2.9983
-2.7616
0.9801
-1.5882
1.189
-1.9592
0.4893
-0.4052
1.704
0.8221
1.881
2.1732
1.8375
Conformer
ID
11
2.1
PubChem
ncbi.nlm.nih.gov
2009.12.11
005A459500000002
Energy
MMFF94 NoEstat
7
1.7.2
Szybki
openeye.com
2012.11.26
135.6239
Feature
Self Overlap
7
2.1
PubChem
ncbi.nlm.nih.gov
2012.11.26
86.477
Fingerprint
Shape
2
2.1
PubChem
ncbi.nlm.nih.gov
2012.11.26
100830 39 18411132508064462452
10256941 240 17827351081866791164
10675989 125 15962585743722630936
11488393 25 17614014309997884915
12128747 34 18341055108625282502
12422481 6 18129104600525268218
12522641 126 16831203889241026711
12788726 201 18334847321065154578
13402501 40 18201718509056083938
13561361 72 18341319098525997000
14394314 77 18409451384560291851
14747282 140 16542119210451637824
15961568 22 18269554004487254630
16067690 210 18189599687916112410
16992787 43 18267293241642027005
21033648 144 18201159850370765412
21792965 270 18192153917999501635
22393880 68 18052821343310973788
25019877 29 16772963664792825647
392239 28 18411140263720857826
469060 322 18192740919685800459
50150288 127 16127828326524187321
508706 21 18411706457128377062
57527585 21 16773230661207504904
Shape
Multipoles
8
1.8.3
OEShape
openeye.com
2012.11.26
706.07
12.01
6.91
1.79
17.04
9.55
0.27
-1.53
2.32
-5.77
-1.4
-0.24
0.06
2.84
Shape
Self Overlap
7
2.1
PubChem
ncbi.nlm.nih.gov
2012.11.26
1555.063
Shape
Volume
7
1.8.3
OEShape
openeye.com
2012.11.26
373.8
Conformer
RMSD
7
2009.12.11
1
Diverse Conformer
ID List
6
2012.02.08
2
97
157
399
126
231
30
416
61
300
230
74
64
104
34
368
386
19
158
127
404
140
314
274
335
154
178
279
260
229
217
320
190
67
145
184
233
100
53
54
96
327
141
156
385
411
313
1
323
255
247
87
210
357
253
63
267
150
250
188
360
7
109
241
28
421
422
418
280
119
316
251
44
206
256
4
98
232
277
131
289
339
62
312
80
331
208
407
221
378
120
342
307
406
161
376
220
333
153
286
72
66
75
324
58
159
5
303
39
396
84
420
48
348
201
202
41
79
21
392
325
130
194
223
165
134
35
135
155
346
116
90
379
209
414
359
29
152
287
167
108
240
33
137
257
290
213
36
189
132
375
121
138
244
398
270
336
102
49
365
363
20
219
423
203
94
245
299
410
388
24
304
14
81
11
114
305
3
111
107
395
263
105
183
243
122
55
146
193
310
52
215
309
258
268
234
65
391
60
9
293
284
271
106
344
83
10
403
142
301
384
82
93
358
362
417
242
144
383
139
367
173
185
147
332
133
89
377
69
246
177
374
401
45
370
166
302
355
207
424
59
322
294
168
389
148
170
103
118
295
380
101
292
99
394
259
88
285
187
199
216
326
262
204
197
15
27
180
387
31
218
330
275
70
77
272
186
6
162
95
112
195
334
17
222
353
85
32
382
402
361
124
366
337
16
235
163
296
113
171
136
264
86
397
356
347
117
172
91
40
151
364
92
71
288
249
343
393
12
160
128
338
236
282
110
78
42
56
149
179
212
408
311
283
409
169
298
308
321
23
22
164
239
390
319
123
345
328
248
192
176
18
369
38
214
351
273
352
8
13
371
211
175
115
51
381
174
46
405
278
349
143
47
237
318
252
350
340
297
73
125
265
266
254
315
228
226
57
191
196
415
200
238
413
205
291
198
76
372
317
329
224
269
68
227
400
276
182
26
37
261
354
129
306
25
281
341
43
225
419
50
181
412
373
Charge
MMFF94 Partial
2
1.7.6
OEChem
openeye.com
2012.02.08
53
1 -0.57
10 -0.55
11 -0.5
12 0.91
13 0.91
14 -0.67
15 0.12
16 0.18
17 0.39
18 0.12
19 0.09
2 -0.57
20 -0.15
21 0.63
22 -0.15
23 -0.15
24 0.39
25 0.4
26 0.12
27 0.63
28 0.09
29 0.13
3 -0.57
30 -0.15
31 -0.15
32 0.13
33 -0.15
34 -0.15
35 -0.15
36 -0.15
37 -0.15
38 -0.15
4 -0.52
41 0.15
42 0.37
43 0.15
44 0.15
45 0.37
46 0.15
47 0.15
48 0.15
49 0.15
5 -0.52
50 0.15
51 0.15
52 0.15
53 0.15
54 0.36
55 0.36
6 -0.52
7 -0.52
8 -0.55
9 -0.63
Count
Effective Rotor
7
1.7.6
OEChem
ncbi.nlm.nih.gov
2012.01.18
9
Features
Pharmacophore
2
ImplicitMillsDean merged
1.8.1
OEShape
openeye.com
2012.02.08
17
1 1 acceptor
1 10 donor
1 11 acceptor
1 2 acceptor
1 3 acceptor
1 4 acceptor
1 4 anion
1 5 acceptor
1 6 acceptor
1 6 anion
1 7 acceptor
1 8 donor
1 9 acceptor
6 15 16 19 20 22 23 rings
6 26 29 30 31 32 33 rings
6 28 34 35 36 37 38 rings
6 8 9 15 16 17 21 rings
38
0
0
0
1
1
0
0
1
83