54649888
1
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67
68
35
16
8
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1
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1
1
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1
1
1
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1
1
1
1
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32
3
6
19
24
66
25
9
11
13
25
52
21
23
10
14
35
12
21
12
36
37
22
15
16
38
24
39
40
18
41
42
17
43
44
20
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46
20
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48
26
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29
23
51
25
53
54
55
57
63
60
61
62
56
58
59
30
31
32
64
33
65
34
34
67
68
1
2
1
1
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2
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2
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1
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2
1
1
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2
1
2
1
1
1
2
3
6
19
-1
1
1
9
6
10
14
35
1
1
2
5
10
1
2
3
4
5
6
7
8
9
10
11
12
13
14
15
16
17
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68
-2.0666
4.592
5.1303
2.3801
-2.5046
3.3533
-3.6449
-1.3064
2.4691
1.0824
2.5568
1.134
-4.978
2.7254
-5.9584
-5.4577
-5.7756
-6.2753
5.7505
-6.7613
-0.1464
-0.0195
-1.2122
2.1209
-2.4786
5.6433
5.3875
7.1665
-0.3179
-0.9902
0.1878
-1.1567
0.0211
-0.6509
2.6875
2.6986
2.7656
-4.927
2.1459
3.6966
-5.5575
-6.8934
-6.3639
-4.7075
-4.8505
-6.1922
-7.0443
-5.3878
-7.7356
-6.9132
0.0255
-3.5469
1.0355
2.5257
6.4098
7.9102
4.6827
7.2897
7.4214
6.2342
5.2427
4.5557
5.7976
-1.3833
0.7055
1.9794
0.4128
-0.7723
-5.0133
0.6574
-0.7336
-2.2864
3.5767
0.789
1.5707
0.2815
-0.3599
0.201
2.0317
1.5821
2.1263
-1.494
1.3186
2.2211
0.8522
-0.0489
1.5978
0.0723
-0.412
2.3352
1.6314
-1.1892
2.3411
3.0849
1.3703
1.0856
-1.8285
-2.5986
-2.4282
-3.9684
-3.7979
-4.5681
-0.69
2.6639
2.6081
3.1432
-2.3563
-1.9826
1.1837
1.8844
2.8393
2.7245
0.2739
0.9818
-0.5446
-0.6916
0.5762
-0.9269
3.4122
0.5616
-1.0803
-0.2985
3.6593
1.6657
3.5295
0.0369
1.1652
1.6968
0.3126
1.9632
3.2547
-2.1334
-1.8455
-2.0756
-4.2644
-5.634
-1.3138
-0.9273
-1.071
-2.7161
0.0862
0.1795
0.3167
0.4385
0.4995
0.4276
0.254
0.2851
0.2449
-0.4942
1.1021
-1.2074
-1.8089
0.4967
0.0965
-0.9443
0.5063
0.2176
0.296
-1.8515
0.2317
-0.2542
1.5671
-0.184
0.7168
-0.2323
1.8703
-0.028
2.0746
1.1254
1.5216
-0.6299
1.1589
0.6532
-0.1336
-0.4779
2.1139
1.2031
-1.2427
-1.8288
-1.9217
-2.8143
1.1004
0.5321
-0.9586
-1.3677
0.1118
0.3818
-1.827
-2.3341
0.2799
0.3748
0.0133
0.1106
-1.2475
2.1881
1.8208
1.9501
-1.3263
-1.1344
2.6284
-3.5767
2.9738
1.3001
Conformer
ID
11
2.1
PubChem
ncbi.nlm.nih.gov
2011.09.13
0341E42000000001
Energy
MMFF94 NoEstat
7
1.7.2
Szybki
openeye.com
2012.11.26
111.3771
Feature
Self Overlap
7
2.1
PubChem
ncbi.nlm.nih.gov
2012.11.26
55.902
Fingerprint
Shape
2
2.1
PubChem
ncbi.nlm.nih.gov
2012.11.26
102385 1 17760932139986135609
10319688 67 18268686442637202976
10906281 52 18341905133474810324
11007060 377 18343585174505090585
11135926 11 18335133147593003829
11136131 41 18042675126908728051
11421498 54 17559679443404060609
11488393 25 17842573846529484383
11991303 11 18115308998061490751
12440605 4 17614580549606994769
12597179 24 18343586243909456678
12788726 201 18191859235445072186
13692114 37 18129085883031301098
13911987 19 18334564742725363269
140371 6 17182210856157848441
14040221 310 17628909321258311844
14068700 686 18263643961916402869
14190465 44 18267293417540701984
14790565 3 18408885105448339249
14955137 171 17759232999521302890
15131766 46 15215017283024168652
15849732 13 17385724707719503236
15927050 60 18410571790682535522
16993438 75 18198620132460149598
18681886 176 18261386789045999665
19311894 1 18271236248952113727
20028762 73 18198898111243777487
20775438 99 18131063801503007038
21133410 62 18189032297631794919
21344244 181 18129956584640506894
21521721 280 18411708664357037033
22393880 68 18122065299973595621
23516275 137 16844474673156163567
23569917 315 18336546032176222042
249057 3 18260832601458377380
3178227 256 18334869329021106369
354706 35 18189594100802125991
4258327 124 17823998899122091868
5171179 24 17625818640542151649
59755656 520 18335413590980517356
6036956 94 16964924290710183804
6669772 16 18412264995618200734
Shape
Multipoles
8
1.8.3
OEShape
openeye.com
2012.11.26
676.94
14.88
5.67
1.63
1.33
7.55
-0.38
-14.48
-3.16
3.78
0.25
0.07
1.4
0.53
Shape
Self Overlap
7
2.1
PubChem
ncbi.nlm.nih.gov
2012.11.26
1418.272
Shape
Volume
7
1.8.3
OEShape
openeye.com
2012.11.26
389.2
Conformer
RMSD
7
2011.09.13
1
Diverse Conformer
ID List
6
2012.02.08
1
30
42
40
32
22
11
36
8
26
25
12
18
21
19
38
2
17
31
28
6
13
7
16
33
20
24
27
41
5
3
29
10
35
34
23
9
37
39
4
15
14
Charge
MMFF94 Partial
2
1.7.6
OEChem
openeye.com
2012.02.08
31
1 -0.11
10 -0.14
11 0.41
12 -0.14
13 0.3
19 0.19
2 0.37
21 0.31
22 -0.15
23 0.4
24 0.28
25 0.54
3 -0.5
30 -0.15
31 -0.15
32 0.11
33 -0.15
34 -0.15
4 -0.68
5 -0.57
51 0.15
52 0.37
6 -0.6
64 0.15
65 0.15
66 0.4
67 0.15
68 0.15
7 -0.73
8 -0.62
9 0.41
Count
Effective Rotor
7
1.7.6
OEChem
ncbi.nlm.nih.gov
2012.01.18
9.8
Features
Pharmacophore
2
ImplicitMillsDean merged
1.8.1
OEShape
openeye.com
2012.02.08
11
1 1 hydrophobe
1 4 acceptor
1 4 donor
1 5 acceptor
1 7 donor
1 8 acceptor
4 19 26 27 28 hydrophobe
5 6 9 10 11 12 rings
6 13 15 16 17 18 20 rings
6 29 30 31 32 33 34 rings
6 8 10 12 21 22 23 rings
34
2
2
0
0
0
0
0
1
2