53348004 1 2 3 4 5 6 7 8 9 10 11 12 13 14 15 16 17 18 19 20 21 22 23 24 25 26 27 28 29 30 31 32 33 34 35 36 37 38 39 40 41 42 43 44 45 46 47 48 49 50 51 52 53 54 55 56 57 58 59 60 61 62 63 64 65 66 67 68 69 70 71 72 73 74 75 76 77 8 8 8 8 7 7 7 7 7 7 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 2 3 3 4 4 5 5 5 6 6 6 7 7 7 8 9 10 11 11 11 12 12 12 13 13 13 14 14 14 15 15 15 16 16 16 17 17 17 18 18 19 19 19 20 20 20 21 21 21 22 22 22 23 23 25 26 26 26 27 27 27 28 28 29 30 30 31 31 32 32 33 34 34 36 36 36 37 37 37 24 25 33 36 35 37 11 14 25 17 24 60 8 9 28 29 10 29 12 13 38 15 41 42 16 39 40 19 24 43 18 44 45 18 46 47 20 21 48 49 50 26 27 51 22 54 55 23 52 53 23 58 59 56 57 28 64 65 66 61 62 63 67 68 30 31 32 33 69 34 70 35 35 71 72 73 74 75 76 77 2 2 1 1 1 1 1 1 1 1 1 1 1 1 1 2 2 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 2 1 1 1 2 1 2 1 1 1 1 1 1 1 1 14 5 19 24 43 3 1 2 5 10 1 2 3 4 5 6 7 8 9 10 11 12 13 14 15 16 17 18 19 20 21 22 23 24 25 26 27 28 29 30 31 32 33 34 35 36 37 38 39 40 41 42 43 44 45 46 47 48 49 50 51 52 53 54 55 56 57 58 59 60 61 62 63 64 65 66 67 68 69 70 71 72 73 74 75 76 77 5.1703 0.7455 -5.6983 -7.9034 2.7595 3.1314 -0.7981 -1.699 -1.2795 -2.587 3.4837 2.9479 3.423 3.5412 3.6641 4.1372 3.3895 3.6041 4.6846 2.8945 2.596 1.402 1.2172 4.053 1.3748 4.1976 5.4835 0.6723 -2.8052 -4.112 -4.2773 -5.2189 -5.5493 -6.4909 -6.6561 -4.5167 -8.9809 4.5404 2.4022 3.9138 3.0785 1.8766 2.9113 3.2143 4.7123 5.2129 4.0184 4.4657 4.1837 2.5663 5.3986 2.5349 3.0637 3.3839 3.0863 0.811 0.5109 0.8289 1.0448 2.2142 6.2631 5.9845 4.8366 3.4787 5.044 3.7002 0.709 1.0965 -3.3946 -5.1207 -7.304 -4.8217 -4.0507 -3.8169 -9.8968 -8.8757 -9.1091 -1.2151 1.7106 -1.7855 -0.3017 0.8841 -2.1076 1.0375 0.3367 2.0559 2.0389 1.2886 0.5657 2.8082 0.246 1.0194 3.2594 -3.4679 2.5349 1.1347 -3.7385 -4.4681 -4.0134 -4.5219 -1.0831 1.1511 2.4883 0.4092 0.6995 1.0011 0.6641 -0.4084 1.4089 -0.7361 1.0813 0.0088 -2.4952 0.5095 1.0143 3.1979 3.3133 -0.5165 0.7213 0.0076 0.5324 0.6979 3.0672 4.3414 -3.6552 2.8312 2.8404 1.3522 -4.2002 -5.458 -4.637 -2.918 -5.5384 -3.8775 -3.0893 -4.7361 -1.892 1.0643 -0.486 0.1095 2.9853 3.1665 2.3607 -0.3871 1.1981 -0.9647 2.25 1.7033 -3.2948 -2.9798 -1.8582 0.1215 1.5483 0.428 0.1037 -0.7249 -1.5691 -0.7573 0.1221 0.7615 1.4729 0.77 2.1991 1.9708 -1.0586 -2.2972 -1.2308 1.1508 -3.5665 -2.5022 0.3583 -3.7351 1.6847 -1.0567 1.1907 -0.8951 0.535 0.5991 0.1773 2.2131 2.7717 1.4492 1.1141 0.6325 -0.2441 1.0397 -0.7133 0.5701 -0.3063 -1.9359 -0.2929 -0.9778 -1.2664 -0.3965 -2.1818 -2.4521 2.0129 -4.4392 -3.5282 -2.4043 -2.6298 0.4386 -4.6166 -3.9167 0.8815 2.2503 1.1209 -1.4527 -1.7542 0.5541 1.071 -1.0358 -1.6355 1.1382 3.1764 2.3935 3.6035 1.5633 2.3662 3.1818 1.5584 2.3259 -0.5393 1.7218 0.9284 -2.6192 -1.071 -2.4877 -0.751 -0.6238 0.7918 Conformer ID 11 2.1 PubChem ncbi.nlm.nih.gov 2012.05.21 032E06A400000005 Energy MMFF94 NoEstat 7 1.7.2 Szybki openeye.com 2012.11.26 100.6471 Feature Self Overlap 7 2.1 PubChem ncbi.nlm.nih.gov 2012.11.26 55.826 Fingerprint Shape 2 2.1 PubChem ncbi.nlm.nih.gov 2012.11.26 11135609 149 17607785236934513234 11796584 16 17561083592677418633 12539747 167 17393615005530165874 12728209 76 17749102284656625581 12758862 65 16343410795538077306 12788726 201 17616822467080518314 13533116 47 18270963440538333371 1361 2 18410290294098730106 14092694 8 17822557409106922055 15001296 14 18272642438076624083 15183329 4 16950561056835940033 15250474 111 18343864407745995695 15264996 154 18200323121717288407 15448158 6 17695907731521900938 15799311 1 18202571670461379523 16114785 44 16050368029902728944 18365409 1 18269271425957786366 19315092 285 17986101916786146338 21223535 225 16879047682483458565 21304303 282 17322969201792029636 25222932 49 17560220535593542053 3044373 193 17240486914192601993 4073 2 18200020893557595699 4093350 32 17821732745316057269 44317340 157 16732988665076150953 46194498 28 17821731606775001895 463206 1 18272081721553669803 474144 1 18341620265600894255 513532 50 17846786178738546782 5223283 242 17317034746378212405 54076057 255 9583232898749448346 Shape Multipoles 8 1.8.3 OEShape openeye.com 2012.11.26 708.08 18.18 4.95 3 44.63 7.03 -1.73 -3.41 -1.93 -7.6 -1.33 -4.76 -2.51 -3.95 Shape Self Overlap 7 2.1 PubChem ncbi.nlm.nih.gov 2012.11.26 1481.204 Shape Volume 7 1.8.3 OEShape openeye.com 2012.11.26 400.4 Conformer RMSD 7 2012.05.21 1.2 Diverse Conformer ID List 6 2012.05.21 5 35 93 114 127 85 59 98 16 29 131 65 20 45 7 14 125 95 68 41 79 51 58 43 15 117 21 31 134 75 53 111 25 135 89 47 17 106 109 86 42 33 18 119 3 52 110 77 132 67 87 32 61 103 48 122 56 28 24 120 88 76 113 19 55 84 12 4 104 126 121 38 94 8 63 23 102 123 40 116 46 57 112 96 11 36 13 49 54 37 129 97 50 73 118 60 72 6 108 69 22 100 30 107 64 78 124 115 44 82 133 10 90 92 66 27 62 70 101 80 71 99 2 9 26 105 81 130 39 91 128 1 34 74 83 Charge MMFF94 Partial 2 1.7.6 OEChem openeye.com 2012.05.21 29 1 -0.57 10 -0.23 11 0.3 14 0.36 17 0.3 2 -0.57 24 0.57 25 0.57 28 0.32 29 0.46 3 -0.36 30 0.05 31 -0.15 32 -0.15 33 0.08 34 -0.15 35 0.08 36 0.28 37 0.28 4 -0.36 5 -0.66 6 -0.73 60 0.37 69 0.15 7 0.58 70 0.15 71 0.15 8 -0.71 9 -0.42 Count Effective Rotor 7 1.7.6 OEChem ncbi.nlm.nih.gov 2012.05.21 14.2 Features Pharmacophore 2 ImplicitMillsDean merged 1.8.1 OEShape openeye.com 2012.05.21 11 1 1 acceptor 1 2 acceptor 1 3 acceptor 1 4 acceptor 1 6 donor 3 19 26 27 hydrophobe 3 8 10 29 cation 5 17 20 21 22 23 rings 5 7 8 9 10 29 rings 6 11 12 13 15 16 18 rings 6 30 31 32 33 34 35 rings 37 1 0 1 0 0 0 0 1 2