5327070
1
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53
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56
57
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61
62
63
64
65
66
67
68
69
70
71
72
73
8
8
8
8
8
8
8
8
8
8
8
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
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6
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6
6
6
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
2
2
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33
15
16
16
19
12
44
13
45
14
46
21
22
21
25
17
61
18
62
20
65
28
70
13
14
34
15
35
16
36
17
37
38
39
40
19
20
41
22
21
42
43
28
24
26
47
48
25
49
50
53
54
27
51
52
29
55
56
57
58
30
59
60
31
63
64
32
66
67
33
68
69
71
72
73
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
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1
2
1
1
1
1
1
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1
1
1
1
1
1
1
1
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1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
12
3
13
14
34
1
1
13
4
12
15
35
1
1
14
5
12
16
36
1
1
15
1
13
17
37
3
1
16
1
2
14
38
3
1
18
9
20
19
41
2
1
20
10
21
18
42
2
1
21
6
7
20
43
3
1
2
5
10
1
2
3
4
5
6
7
8
9
10
11
12
13
14
15
16
17
18
19
20
21
22
23
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32
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34
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43
44
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51
52
53
54
55
56
57
58
59
60
61
62
63
64
65
66
67
68
69
70
71
72
73
-0.9165
-2.9029
0.8296
0.2862
-1.8582
-3.3732
-1.8476
1.1405
-4.1065
-5.2838
-2.0163
0.1343
0.7786
-1.3379
0.4925
-1.505
1.0013
-3.2857
-3.1322
-3.8779
-3.2203
-3.1987
1.005
0.1558
-1.3117
2.4677
3.3088
-3.1195
4.7896
5.617
7.0702
7.8905
9.3265
0.209
1.8651
-1.9143
0.9638
-1.0201
0.3053
1.9871
-2.2942
-3.7348
-3.7394
1.7546
0.5134
-1.7382
0.6111
0.9418
0.2352
0.5447
2.8768
2.5301
-1.4085
-1.864
3.2226
2.9012
-4.0329
-3.0235
5.21
4.8709
1.4692
-4.1584
5.1763
5.5811
-5.6273
7.0985
7.518
7.8867
7.4366
-2.0096
9.8203
9.8952
9.3656
-1.7633
-1.5751
-2.9102
-4.4126
-3.3362
1.8658
2.8176
-0.396
-0.3372
1.7575
0.4558
-3.6848
-3.4471
-3.2632
-2.0196
-1.8489
-1.7898
0.4386
-0.2166
1.8429
2.58
0.4923
2.8339
4.0819
3.8624
3.0673
1.81
-0.0965
1.9965
0.7192
0.944
-0.3399
-0.1287
-4.7358
-3.5813
-3.9628
-1.2888
-1.1301
-2.1825
-2.2435
0.5068
2.3816
3.538
-3.21
-5.2927
-4.2492
1.9866
2.5612
4.3474
4.9246
3.8961
3.3586
3.6091
4.7902
1.5018
0.9896
0.1485
-1.1858
2.7849
2.3493
-0.2731
0.1313
-0.0794
0.387
2.6656
1.2979
1.7291
-0.6857
-1.1319
0.0612
0.6369
-1.0588
0.185
0.9675
-0.2441
-1.8821
1.3912
-2.2145
1.0041
-0.5311
2.5921
-2.3921
-1.161
3.0405
-0.9033
0.4648
-0.8902
0.9637
-0.3305
2.3822
-1.5239
-0.1792
-1.3959
-0.2311
0.968
0.18
-0.0791
0.2678
-0.2067
0.0246
2.3455
-0.3179
-0.1574
-0.5817
-0.4589
-0.9114
-1.2054
0.3985
-0.2718
0.2927
-1.006
3.1306
2.5243
-1.9874
-2.3399
-0.0986
-1.889
1.0459
-2.5267
-0.3942
1.2405
-1.1404
0.5039
0.3834
-1.2621
1.33
0.0779
1.074
-0.5794
2.8987
2.3357
0.3186
-1.3537
3.4989
-3.2426
-0.7666
0.8871
-1.1073
-1.6196
0.0396
0.5813
-1.0658
3.9292
-0.3045
-0.8138
-1.9595
Conformer
ID
11
2.1
PubChem
ncbi.nlm.nih.gov
2009.12.11
005148DE00000001
Energy
MMFF94 NoEstat
7
1.7.2
Szybki
openeye.com
2012.11.26
60.3062
Feature
Self Overlap
7
2.1
PubChem
ncbi.nlm.nih.gov
2012.11.26
106.713
Fingerprint
Shape
2
2.1
PubChem
ncbi.nlm.nih.gov
2012.11.26
107951 10 17312813884390480393
10864689 126 18339070494274078816
11513181 2 18127123074898960502
13761468 95 18115578254537012660
14279260 333 17894911811850873522
14659021 117 18049429637618613480
15183329 4 18409448082031036970
16719943 64 18408603656768615052
17627616 140 18191016816570069754
19311894 1 18339641260555418348
19930381 70 18338506436197353149
20775530 9 16752404111607864609
5265222 85 18261112997507494500
Shape
Multipoles
8
1.8.3
OEShape
openeye.com
2012.11.26
614.56
13.99
5.86
2.14
44.94
1.61
-0.97
-5.54
5.97
-2.08
0.71
-2.25
1.31
-0.26
Shape
Self Overlap
7
2.1
PubChem
ncbi.nlm.nih.gov
2012.11.26
1225.489
Shape
Volume
7
1.8.3
OEShape
openeye.com
2012.11.26
358
Conformer
RMSD
7
2009.12.11
1.2
Diverse Conformer
ID List
6
2012.02.08
1
106
76
73
365
4
145
299
197
319
83
7
234
84
114
67
254
126
343
111
133
324
311
216
174
134
361
140
54
51
349
267
326
47
118
154
138
208
280
246
308
24
59
105
151
135
269
167
221
356
33
262
34
6
64
95
98
122
30
353
20
223
102
63
345
312
320
272
115
228
43
120
191
350
39
36
220
329
159
91
250
110
201
16
300
5
149
195
292
177
49
146
72
341
85
61
100
87
104
2
328
11
335
198
330
116
288
169
69
70
50
137
66
354
180
22
12
321
271
336
38
275
46
127
3
230
351
233
327
144
89
204
26
263
298
264
241
227
82
213
125
305
291
214
18
217
75
346
161
136
290
239
28
357
229
52
245
265
301
340
237
331
232
274
225
10
215
306
194
107
266
178
53
322
74
150
9
231
206
257
338
199
32
171
90
68
93
253
157
176
251
212
309
158
35
363
160
183
238
302
313
27
168
268
130
323
339
284
56
166
222
139
19
259
121
256
86
304
360
45
163
283
242
153
21
79
337
293
211
60
203
202
13
261
48
189
196
249
358
42
205
77
92
310
235
276
80
162
210
185
99
112
317
244
143
147
124
297
270
348
344
252
131
156
94
226
318
175
25
17
224
148
141
186
296
108
364
282
219
71
184
325
209
155
129
192
277
142
187
286
285
97
352
182
23
200
367
289
170
315
273
41
333
172
303
295
314
101
279
260
236
278
14
132
366
165
31
181
355
179
294
258
15
243
188
359
316
103
342
287
255
8
65
207
62
109
164
281
55
44
117
96
88
218
173
347
57
58
40
128
248
362
119
29
334
307
81
247
332
113
37
152
123
190
193
78
240
Charge
MMFF94 Partial
2
1.7.6
OEChem
openeye.com
2012.02.08
31
1 -0.56
10 -0.68
11 -0.68
12 0.28
13 0.28
14 0.28
15 0.28
16 0.56
17 0.28
18 0.42
19 -0.06
2 -0.36
20 0.28
21 0.56
22 -0.06
25 0.28
28 0.42
3 -0.68
4 -0.68
44 0.4
45 0.4
46 0.4
5 -0.68
6 -0.36
61 0.4
62 0.4
65 0.4
7 -0.56
70 0.4
8 -0.68
9 -0.68
Count
Effective Rotor
7
1.7.6
OEChem
ncbi.nlm.nih.gov
2012.01.18
16
Features
Pharmacophore
2
ImplicitMillsDean merged
1.8.1
OEShape
openeye.com
2012.02.08
21
1 1 acceptor
1 10 acceptor
1 10 donor
1 11 acceptor
1 11 donor
1 2 acceptor
1 3 acceptor
1 3 donor
1 33 hydrophobe
1 4 acceptor
1 4 donor
1 5 acceptor
1 5 donor
1 6 acceptor
1 7 acceptor
1 8 acceptor
1 8 donor
1 9 acceptor
1 9 donor
6 1 12 13 14 15 16 rings
6 6 18 19 20 21 22 rings
33
8
5
3
0
0
0
0
1
1