5324287 1 2 3 4 5 6 7 8 9 10 11 12 13 14 15 16 17 18 19 20 21 22 23 24 25 26 27 28 29 30 31 32 33 34 35 36 37 38 39 40 8 8 8 7 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 2 2 3 3 4 4 4 5 5 5 5 6 6 6 7 7 8 8 9 9 9 10 10 11 11 11 12 12 13 14 14 15 15 16 17 18 18 18 19 19 20 21 8 16 14 39 20 40 7 12 18 6 8 9 10 7 15 22 11 23 14 24 12 25 26 13 16 13 27 28 29 30 19 17 31 17 32 20 33 34 35 36 21 37 21 38 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 2 1 1 1 1 1 1 1 1 1 2 1 2 1 1 1 1 2 1 1 1 5 6 8 9 10 1 1 6 5 15 7 22 2 1 7 4 6 11 23 1 1 8 1 14 5 24 2 1 14 2 8 17 31 1 1 2 5 10 1 2 3 4 5 6 7 8 9 10 11 12 13 14 15 16 17 18 19 20 21 22 23 24 25 26 27 28 29 30 31 32 33 34 35 36 37 38 39 40 1.7914 0.7093 4.0401 -2.9059 -0.4945 -1.5772 -2.2287 0.5348 -1.1779 0.4672 -1.2022 -2.0437 0.1786 0.8498 -1.0624 1.7379 0.0112 -4.1647 1.23 2.7869 2.52 -2.3431 -2.9909 0.236 -1.8102 -0.4395 -1.1075 -1.5907 -1.3889 -2.6392 1.9005 -1.6225 0.3039 -4.0253 -4.7144 -4.817 1.0684 3.3243 -0.2204 4.0199 0.9209 3.8894 -0.8587 -1.1905 0.4957 0.7773 -0.5983 1.6078 -0.0492 -0.517 -1.6253 -1.2894 -1.5472 2.536 1.5463 -0.2544 2.3438 -0.5146 -2.4002 -1.0911 -2.1813 1.4317 -0.4538 2.2005 0.7374 -0.3102 -1.4194 -2.6472 -2.1604 -1.5305 2.4244 1.4987 2.9023 0.5055 -1.0768 -0.4766 -3.2293 -2.8592 4.0264 -0.0573 1.2404 0.1041 0.6851 0.3771 0.5841 -0.46 -0.8076 0.8687 1.8567 0.0636 -1.4038 1.5656 -0.8105 -0.3363 -1.6433 0.5302 -1.5693 0.6924 -1.146 0.2248 -0.6159 -0.0221 -1.5858 1.7421 2.2888 2.6259 -2.4783 -1.3105 1.4393 2.4557 -0.6288 -2.5727 -2.455 1.0633 1.4559 -0.1871 -1.8296 -0.8929 0.3557 1.2368 Conformer ID 11 2.1 PubChem ncbi.nlm.nih.gov 2009.12.11 00513DFF00000001 Energy MMFF94 NoEstat 7 1.6.0 Szybki openeye.com 2012.01.18 72.9812 Feature Self Overlap 7 2.1 PubChem ncbi.nlm.nih.gov 2012.01.18 52.925 Fingerprint Shape 2 2.1 PubChem ncbi.nlm.nih.gov 2012.11.26 10863032 1 17557706867634788107 10948715 1 16680922030260241036 12035758 1 18264764372891529249 12403814 3 18339068337714393914 12423570 1 11142607001003850881 12592029 89 17829345922249970173 13140716 1 18057314192229643938 13172582 1 18272929448970448898 13299463 15 17626360352134994668 13681431 1 18117022002881156845 141345 1 16456032341388552863 14142880 1 18129377090625704432 14181834 199 18267591393126713479 144361 1 17472653333819129837 14817 1 10862617623532031379 14955137 171 18127152954886198458 15881359 60 18127101178638889083 16945 1 18201991162074899423 17357779 13 18339348670271814055 19868273 325 18335704884110067694 20600515 1 17895773819317058343 21330990 113 17836382449239583269 22907989 373 17977965483495508718 23419403 2 18057298653164171505 23557571 272 18190468168915883558 23559900 14 17898272932665647434 2748010 2 18197190647221644644 576247 118 18189074047831926675 6442390 28 17112707986135533761 7364860 26 18265623267223524729 81228 2 17828506685650771064 84936 31 18195256739148550821 9981440 41 17407077026210467522 Shape Multipoles 8 1.8.1 OEShape openeye.com 2012.01.18 409.58 4.31 3.11 1.59 0.2 2.61 0.01 -2.78 -1.21 -1.04 0.94 0.47 0.02 0.66 Shape Self Overlap 7 2.1 PubChem ncbi.nlm.nih.gov 2012.01.18 930.238 Shape Volume 7 1.8.1 OEShape openeye.com 2012.01.18 211.2 Conformer RMSD 7 2009.12.11 0.6 Diverse Conformer ID List 6 2010.05.05 1 Charge MMFF94 Partial 2 1.7.6 OEChem openeye.com 2012.05.21 26 1 -0.36 10 -0.14 11 0.14 12 0.27 13 -0.14 14 0.42 15 -0.29 16 0.08 17 -0.29 18 0.27 19 -0.15 2 -0.68 20 0.08 21 -0.15 3 -0.53 32 0.15 33 0.15 37 0.15 38 0.15 39 0.4 4 -0.81 40 0.45 5 0.14 6 0.14 7 0.27 8 0.28 Count Effective Rotor 7 1.7.6 OEChem ncbi.nlm.nih.gov 2012.01.18 1.2 Features Pharmacophore 2 ImplicitMillsDean merged 1.8.1 OEShape openeye.com 2012.05.21 10 1 1 acceptor 1 2 acceptor 1 2 donor 1 3 donor 1 4 cation 5 1 5 8 10 16 rings 6 10 13 16 19 20 21 rings 6 4 5 6 7 9 12 rings 6 5 6 7 10 11 13 rings 6 5 6 8 14 15 17 rings 21 5 5 0 0 0 0 0 1 3