49878499
1
2
3
4
5
6
7
8
9
10
11
12
13
14
15
16
17
18
19
20
21
22
23
24
25
26
27
28
29
30
31
32
33
34
35
36
37
38
39
40
41
42
43
44
45
46
47
48
49
50
51
52
53
54
55
56
57
58
59
60
16
8
8
8
7
7
7
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
2
3
5
5
5
6
6
6
7
7
7
8
8
8
9
9
9
10
10
10
11
11
11
12
12
13
13
13
14
14
14
15
15
16
17
17
18
18
19
20
21
21
22
22
22
23
24
25
25
26
27
27
27
28
28
29
29
30
30
31
4
19
26
16
24
8
10
13
15
16
48
18
22
24
9
14
32
11
33
34
12
35
36
12
37
38
39
40
15
41
42
43
44
45
46
47
17
20
21
19
20
23
49
23
50
27
51
52
53
25
26
28
29
55
56
57
30
54
31
58
31
59
60
2
1
1
2
2
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
2
1
2
1
1
1
2
1
1
1
1
1
1
1
2
2
1
1
1
1
1
1
1
2
1
1
1
4
19
26
-1
3
1
8
5
9
14
32
3
1
2
5
10
1
2
3
4
5
6
7
8
9
10
11
12
13
14
15
16
17
18
19
20
21
22
23
24
25
26
27
28
29
30
31
32
33
34
35
36
37
38
39
40
41
42
43
44
45
46
47
48
49
50
51
52
53
54
55
56
57
58
59
60
4.158
-1.7864
5.4388
4.0528
-6.0583
-2.5284
3.2844
-6.8937
-8.3773
-6.2196
-8.5893
-7.6716
-4.6366
-6.7777
-3.9311
-1.5339
-0.1636
2.2344
2.481
0.8954
0.0919
3.0094
1.4056
4.5199
4.7352
4.6384
3.4909
5.12
4.9234
5.3925
5.2953
-6.5816
-8.7462
-8.9844
-5.8715
-5.6243
-9.6349
-8.3806
-7.7599
-7.9848
-4.1511
-4.4761
-6.8847
-7.563
-5.8281
-4.006
-4.3641
-2.277
0.6475
-0.696
3.549
1.9649
1.5723
5.2085
3.317
2.9623
4.562
4.8596
5.6859
5.5116
-0.7919
1.4189
2.0105
-2.0945
-0.1353
0.2848
1.6641
-1.3316
-0.931
0.8644
0.1283
1.3156
-0.4628
-2.3827
0.5944
0.7226
0.3481
0.7996
-0.3613
1.1461
-0.8046
3.1028
-1.1537
1.2461
-0.1766
-1.1945
3.7591
-0.4734
-2.5131
-1.7901
-2.8084
-1.8028
-0.5494
-1.811
0.4624
1.76
0.4552
-0.3016
2.0286
1.8414
-0.5877
-1.409
-1.9286
-3.1409
-2.9241
1.5916
0.6417
-0.2333
2.0026
-1.4721
3.5561
3.3642
-2.0517
0.3117
4.8391
3.3575
3.5928
-3.3284
-2.0209
-3.8342
-1.7223
0.7221
0.8765
-2.4577
-0.0218
-1.1595
0.0433
0.233
0.362
1.0488
1.4358
1.1896
-0.1631
-0.8802
-0.9996
-0.2771
-0.5886
-0.4211
-1.1839
-0.1536
-1.3178
0.043
-1.6216
0.5733
0.9124
-0.0399
-1.2343
2.2264
0.3353
2.5927
1.6479
1.1756
-0.5995
0.6073
2.01
0.8425
1.4407
2.423
2.0171
0.2788
0.8142
-0.687
-1.8716
-0.7791
-0.8452
-0.5561
-2.0053
-1.9944
0.4653
-1.6533
0.8842
0.2056
-2.2111
2.9733
-1.1986
-2.1053
-1.3893
-0.3804
3.6126
1.9318
Conformer
ID
11
2.1
PubChem
ncbi.nlm.nih.gov
2010.09.21
02F915E300000004
Energy
MMFF94 NoEstat
7
1.7.2
Szybki
openeye.com
2012.11.26
91.9659
Feature
Self Overlap
7
2.1
PubChem
ncbi.nlm.nih.gov
2012.11.26
45.692
Shape
Multipoles
8
1.8.3
OEShape
openeye.com
2012.11.26
609.26
23.5
3
1.95
56.02
1.28
-0.16
-8.08
-10.67
-5.12
-0.06
-2.47
-0.97
-2.1
Shape
Self Overlap
7
2.1
PubChem
ncbi.nlm.nih.gov
2012.11.26
1285.653
Shape
Volume
7
1.8.3
OEShape
openeye.com
2012.11.26
341.5
Conformer
RMSD
7
2010.09.21
1
Diverse Conformer
ID List
6
2012.02.08
4
151
45
104
71
124
30
40
90
18
157
128
137
91
94
84
139
121
152
153
127
173
78
68
130
95
44
156
171
52
170
70
14
163
72
176
92
131
67
28
57
140
76
41
99
166
26
77
183
36
43
119
1
134
51
111
96
168
88
161
46
143
165
39
155
162
106
150
115
33
174
66
7
69
25
129
172
98
37
120
180
116
123
31
16
9
136
60
109
55
59
75
169
8
54
27
101
21
138
63
5
48
147
133
122
126
145
34
81
117
160
24
50
181
113
159
35
144
178
53
97
2
149
177
112
47
175
23
32
65
58
182
79
15
3
87
146
12
132
38
85
74
13
93
10
105
107
110
73
56
64
82
22
135
29
61
125
89
49
20
167
184
142
100
11
19
102
164
17
118
108
86
154
141
179
148
80
6
103
42
83
158
62
114
Charge
MMFF94 Partial
2
1.7.6
OEChem
openeye.com
2012.02.08
34
1 0.37
10 0.27
13 0.27
15 0.3
16 0.54
17 0.09
18 0.12
19 0.06
2 -0.57
20 -0.15
21 -0.15
22 0.3
23 -0.15
24 0.54
25 0.09
26 0.06
28 -0.15
29 -0.15
3 -0.57
30 -0.15
31 -0.15
4 -0.5
48 0.37
49 0.15
5 -0.81
50 0.15
53 0.15
54 0.15
58 0.15
59 0.15
6 -0.73
60 0.15
7 -0.48
8 0.27
Count
Effective Rotor
7
1.7.6
OEChem
ncbi.nlm.nih.gov
2012.01.18
7.4
Features
Pharmacophore
2
ImplicitMillsDean merged
1.8.1
OEShape
openeye.com
2012.02.08
9
1 2 acceptor
1 3 acceptor
1 4 acceptor
1 5 cation
1 6 donor
6 17 18 19 20 21 23 rings
6 25 26 28 29 30 31 rings
6 5 8 9 10 11 12 rings
7 1 7 18 19 24 25 26 rings
31
2
0
2
0
0
0
0
1
2