4863108
1
2
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5
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9
10
11
12
13
14
15
16
17
18
19
20
21
22
23
24
25
26
27
28
29
30
31
32
33
34
35
36
37
8
8
8
7
7
7
6
6
6
6
6
6
6
6
6
6
6
6
6
6
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
2
2
3
4
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5
5
5
6
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9
9
11
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13
13
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15
15
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16
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17
17
18
19
19
19
20
20
20
12
19
14
20
10
6
7
16
8
10
21
11
8
13
11
10
12
15
22
14
23
24
25
17
18
26
27
28
29
18
30
31
32
33
34
35
36
37
1
1
1
1
2
1
1
1
1
1
1
2
2
1
1
1
2
1
1
1
1
1
1
2
2
1
1
1
1
1
1
1
1
1
1
1
1
1
2
5
10
1
2
3
4
5
6
7
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9
10
11
12
13
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17
18
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37
2.4023
4.7571
-0.0621
-4.6783
-1.185
-4.3544
-3.6025
-2.5402
1.211
-0.0448
-3.0211
2.3986
-3.7331
3.5901
1.215
-6.0698
3.594
2.4064
2.183
5.5339
-1.0721
-2.5023
-4.4416
-4.0867
-2.7788
0.3253
-6.1935
-6.3554
-6.6808
4.5186
2.4118
1.2225
2.9942
2.1675
5.8475
4.9666
6.4261
1.6916
0.2699
1.5294
0.1222
-0.3397
1.3424
-0.6855
0.0711
-0.3413
0.3813
1.2974
0.3346
-2.0658
-0.3773
-1.729
-0.2075
-1.765
-2.441
2.2069
0.7054
-1.2675
2.1778
-2.6405
-2.0641
-2.6004
-2.2957
-0.5921
-0.961
0.6901
-2.3259
-3.5206
1.8658
1.9058
3.2986
-0.1502
1.413
1.2099
-0.1849
-0.4587
0.8413
-0.0383
0.0119
0.4225
-0.2636
0.0754
0.2351
0.3843
0.4886
-0.0451
-0.7692
-0.1844
0.376
-0.2428
-0.0438
0.2364
-1.4957
0.6552
-0.3854
0.8373
-0.1635
-1.8053
-0.7452
0.635
-1.2581
0.4953
-0.1148
-0.1496
0.3552
-1.8948
-2.166
-1.4358
1.2617
1.268
0.2743
Conformer
ID
11
2.1
PubChem
ncbi.nlm.nih.gov
2009.12.11
004A348400000003
Energy
MMFF94 NoEstat
7
1.7.2
Szybki
openeye.com
2012.11.26
71.7086
Feature
Self Overlap
7
2.1
PubChem
ncbi.nlm.nih.gov
2012.11.26
35.535
Fingerprint
Shape
2
2.1
PubChem
ncbi.nlm.nih.gov
2012.11.26
10616163 171 18343021129398539439
11471102 20 18334859394286626066
11806522 49 18412825785471519176
12107183 9 17692535507577779059
12236239 1 18202003205057520489
13167823 11 18413107251827036471
13760787 19 18342458136299856895
13836976 161 18408326609423320886
14341114 176 18412269410944547759
14576447 43 18342170098396898631
15196674 1 18340769239036606187
15242433 33 18341612594820685159
17834072 33 18413386540580802543
18186145 218 17458344147824661763
18681886 176 18343298206449447546
200 152 18343863308049498393
20612939 158 18187372055408913900
20645477 70 18339643330424154718
21033648 29 14779814022854987597
21054139 6 18339070609499360374
21267235 1 18341058436470204875
21709351 56 18261387879528966237
221490 88 18337677541272845091
2255824 54 18260833691572832138
23402539 116 17458339745235328396
23402655 69 18410855430184833479
23557571 272 17489314048657574913
23559900 14 18271795878621099273
300161 21 18412256225384217583
3004659 81 18339361868463987295
3060560 45 18335143085751558206
34797466 226 17060341855139907776
3545911 37 18411136939758561899
4072396 5 18187634805013607050
4214541 1 18340486677913055081
42630746 31 18410573985742366294
46194498 28 17749390386134891589
474 4 18113903796426075212
5104073 3 18339081475708039059
5281201 14 17968096387288859677
58051976 100 18411701010862192471
58051976 378 18410857663536334911
602551 16 15913030062883877695
67856867 119 18338231694917173996
77779 3 18411702058744444155
9709674 26 18408892836405653483
9971528 1 18334860485519464820
9981440 41 17400079067922093241
Shape
Multipoles
8
1.8.3
OEShape
openeye.com
2012.11.26
379.04
11.85
2.19
0.85
7.16
0.44
-0.15
-0.12
-0.35
-1.06
-0.31
-0.21
-0.27
-0.97
Shape
Self Overlap
7
2.1
PubChem
ncbi.nlm.nih.gov
2012.11.26
805.886
Shape
Volume
7
1.8.3
OEShape
openeye.com
2012.11.26
213.5
Conformer
RMSD
7
2009.12.11
0.8
Diverse Conformer
ID List
6
2012.02.08
3
10
15
1
13
11
9
6
7
17
12
2
5
14
4
16
8
Charge
MMFF94 Partial
2
1.7.6
OEChem
openeye.com
2012.02.08
25
1 -0.36
10 0.54
11 0.14
12 0.08
13 0.18
14 0.08
15 -0.15
16 0.26
17 -0.15
18 -0.15
19 0.28
2 -0.36
20 0.28
21 0.37
22 0.15
26 0.15
3 -0.57
30 0.15
31 0.15
4 0.31
5 -0.49
6 -0.71
7 -0.33
8 0.06
9 0.09
Count
Effective Rotor
7
1.7.6
OEChem
ncbi.nlm.nih.gov
2012.01.18
5
Features
Pharmacophore
2
ImplicitMillsDean merged
1.8.1
OEShape
openeye.com
2012.02.08
7
1 1 acceptor
1 2 acceptor
1 3 acceptor
1 5 donor
1 6 acceptor
5 4 6 7 8 11 rings
6 9 12 14 15 17 18 rings
20
0
0
0
0
0
0
0
1
2