4852411
1
2
3
4
5
6
7
8
9
10
11
12
13
14
15
16
17
18
19
20
21
22
23
24
25
26
27
28
29
30
31
32
33
34
35
36
37
38
39
40
41
42
43
44
45
46
47
48
49
16
8
8
7
7
7
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
2
3
4
4
4
5
5
5
6
6
7
7
7
8
8
8
9
9
10
11
11
12
13
13
14
14
15
15
16
17
17
17
18
19
19
20
21
21
22
23
24
24
25
25
26
26
26
27
27
28
21
22
10
18
7
10
34
12
18
37
20
22
8
9
29
9
30
31
32
33
11
12
13
14
15
35
16
36
16
38
39
19
20
24
21
23
26
25
40
41
23
42
27
43
28
44
45
46
47
28
48
49
1
1
2
2
1
1
1
1
1
1
1
2
1
1
1
1
1
1
1
1
1
1
2
2
1
1
1
1
2
1
1
1
1
2
1
2
1
2
1
1
1
1
1
1
1
1
1
1
1
2
1
1
2
5
10
1
2
3
4
5
6
7
8
9
10
11
12
13
14
15
16
17
18
19
20
21
22
23
24
25
26
27
28
29
30
31
32
33
34
35
36
37
38
39
40
41
42
43
44
45
46
47
48
49
3.2157
-2.2333
1.3719
-3.1124
-0.2278
1.8069
-3.5255
-4.6235
-4.8395
-2.4828
-2.1409
-1.0522
-2.9399
-0.742
-2.6399
-1.541
2.5151
0.8917
3.7033
1.5818
1.5112
2.9662
3.9381
2.2473
0.4015
4.756
1.0587
0.135
-2.6956
-5.1372
-4.5248
-4.8855
-5.4969
-3.2444
-3.8227
0.0868
-0.4867
-3.2659
-1.3096
1.5253
0.9459
4.853
2.9477
-0.3282
4.3546
5.6125
5.1403
0.855
-0.7935
-1.7781
-0.383
-3.5997
1.0096
-1.9266
0.3022
2.0569
2.9945
1.9842
-0.1619
-1.1449
-1.9924
-1.2287
-2.922
-2.1591
-3.0057
1.782
-2.6998
1.05
1.3674
-2.334
-0.3772
-0.048
2.8986
2.0947
1.4084
3.6077
3.2049
2.4873
2.8373
4.0338
2.3434
1.1498
1.1851
-0.6112
-3.6124
-1.2228
-2.2297
-3.7305
-3.2313
-1.5672
-0.6262
3.2405
1.8059
1.3524
0.7262
2.4163
4.4705
3.7542
2.0876
1.6902
0.3516
0.0602
0.7527
1.1676
0.9527
0.5704
1.6587
0.4936
-0.5271
-0.3962
-1.6674
-1.3769
-2.6624
-2.5173
-0.5977
1.0362
-0.7263
0.3754
2.3681
1.0116
0.0886
-1.4076
0.5026
-1.7278
-1.2589
-0.3024
1.503
-0.3701
0.8589
2.6794
1.4469
-0.9317
-1.8065
-1.3477
1.4381
-3.5472
-3.2925
2.9949
2.9053
0.0025
-2.1649
1.255
-2.745
-1.6841
-1.5386
-1.8858
-0.1774
Conformer
ID
11
2.1
PubChem
ncbi.nlm.nih.gov
2009.12.11
004A0ABB00000002
Energy
MMFF94 NoEstat
7
1.7.2
Szybki
openeye.com
2012.11.26
85.7117
Feature
Self Overlap
7
2.1
PubChem
ncbi.nlm.nih.gov
2012.11.26
40.628
Fingerprint
Shape
2
2.1
PubChem
ncbi.nlm.nih.gov
2012.11.26
10165383 225 17096936973724949982
10369192 42 16082237223603597468
10675989 125 17691098841460813733
11513181 2 17269188359539536261
12156800 1 12602637754040912827
12422481 6 17691394218544632777
12553582 1 18115298973977281976
12633257 1 17530962441131868451
12788726 201 17984980646980193791
13965767 371 17768501938114038619
14790565 3 18115606949066440732
15274700 242 17894914075062001672
15297060 5 17560523885187039723
15403338 16 17460593611524538529
15420108 30 18057318384581584637
15664445 248 16690175013666916599
16752209 62 17988633134334516807
1979834 28 17840869569352109905
21133410 90 17338661199446669493
21315764 21 17315882633737251894
21756936 100 18263938781334694994
21860390 5 18117285752817883387
22149856 69 17488189189630919609
23558518 356 18121785198858807784
238 59 17681244948884296806
445580 8 18339077069129543400
513202 73 17037232027695792410
57100710 29 18342443846806435347
70251023 43 17552926534659336414
Shape
Multipoles
8
1.8.3
OEShape
openeye.com
2012.11.26
553.39
7.8
5.07
2.36
2.01
0.26
0.45
4.91
-0.66
1.12
1.17
0.36
-1.6
-4.72
Shape
Self Overlap
7
2.1
PubChem
ncbi.nlm.nih.gov
2012.11.26
1188.839
Shape
Volume
7
1.8.3
OEShape
openeye.com
2012.11.26
306.4
Conformer
RMSD
7
2009.12.11
1
Diverse Conformer
ID List
6
2012.02.08
2
168
175
145
80
375
322
324
137
124
307
189
290
178
44
250
50
242
269
97
300
188
82
347
90
143
144
224
264
112
136
222
45
135
357
117
326
345
293
321
208
47
192
329
176
210
5
284
313
184
294
198
185
373
29
105
39
18
283
118
32
359
343
238
103
288
87
261
296
230
36
330
3
8
173
17
335
6
295
48
204
206
201
353
102
193
1
212
195
225
43
54
21
57
227
356
235
33
126
362
79
122
107
249
234
120
183
245
319
374
113
292
132
114
203
25
364
360
31
268
200
239
312
276
301
28
180
226
323
4
260
139
7
156
367
56
15
243
92
219
190
221
327
63
164
369
246
304
53
42
197
110
275
202
55
263
361
354
352
236
74
181
34
303
94
131
241
157
240
127
244
207
171
169
342
149
13
211
334
231
121
213
377
259
11
167
370
291
194
88
141
311
70
256
58
138
328
12
115
20
170
129
340
27
187
305
116
237
38
267
262
147
270
160
281
346
318
60
358
146
196
232
297
109
166
152
123
325
298
62
338
35
376
71
229
91
10
155
75
217
314
365
125
77
30
162
255
182
69
215
46
140
289
351
142
86
159
252
177
341
220
78
279
309
366
266
223
165
37
61
85
331
22
172
64
100
320
153
344
355
233
59
251
306
41
111
199
339
119
133
209
24
65
128
265
274
148
106
84
299
40
248
277
214
337
99
163
378
186
253
332
310
16
315
179
286
317
280
98
130
350
271
89
348
258
247
14
108
174
254
333
67
23
26
73
205
68
372
287
272
371
49
363
19
273
52
158
216
154
218
134
257
285
101
151
93
95
278
228
66
316
9
96
302
191
336
150
81
51
368
282
349
76
308
104
72
161
83
Charge
MMFF94 Partial
2
1.7.6
OEChem
openeye.com
2012.02.08
43
1 -0.33
10 0.54
11 0.09
12 0.12
13 -0.15
14 -0.15
15 -0.15
16 -0.15
18 0.57
19 -0.14
2 -0.57
20 0.31
21 0.29
22 0.41
23 -0.15
24 -0.15
25 -0.15
26 0.14
27 -0.15
28 -0.15
29 0.1
3 -0.57
30 0.1
31 0.1
32 0.1
33 0.1
34 0.37
35 0.15
36 0.15
37 0.37
38 0.15
39 0.15
4 -0.58
42 0.15
43 0.15
44 0.15
48 0.15
49 0.15
5 -0.55
6 -0.62
7 0.05
8 -0.2
9 -0.2
Count
Effective Rotor
7
1.7.6
OEChem
ncbi.nlm.nih.gov
2012.01.18
8.6
Features
Pharmacophore
2
ImplicitMillsDean merged
1.8.1
OEShape
openeye.com
2012.02.08
8
1 2 acceptor
1 3 acceptor
1 4 donor
1 5 donor
1 6 acceptor
6 11 12 13 14 15 16 rings
6 17 20 24 25 27 28 rings
6 6 17 19 20 22 23 rings
28
0
0
0
0
0
0
0
1
5