475100
1
2
3
4
5
6
7
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9
10
11
12
13
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47
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51
52
53
54
55
56
57
58
9
8
8
8
7
7
7
7
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
2
2
3
3
4
5
5
5
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19
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21
21
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23
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28
28
29
29
30
30
31
7
26
19
56
24
12
13
14
18
22
24
15
22
25
10
11
15
32
12
33
34
13
35
36
37
38
39
40
16
41
42
23
17
43
44
24
25
19
45
46
20
47
21
48
49
22
50
51
26
27
28
29
30
52
53
54
55
31
57
31
58
1
1
1
1
1
2
1
1
1
1
1
1
2
2
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
2
1
1
1
1
1
1
1
1
1
1
1
2
1
1
1
2
1
1
1
1
2
1
1
1
19
3
18
20
47
3
1
2
5
10
1
2
3
4
5
6
7
8
9
10
11
12
13
14
15
16
17
18
19
20
21
22
23
24
25
26
27
28
29
30
31
32
33
34
35
36
37
38
39
40
41
42
43
44
45
46
47
48
49
50
51
52
53
54
55
56
57
58
-9.7216
-6.1097
7.9293
3.9683
-0.2004
5.6849
-4.7301
5.2045
-3.111
-2.2583
-2.3964
-0.8279
-0.9606
1.1837
-4.5259
1.9728
3.397
6.6691
8.0166
8.4869
7.4786
6.0406
-5.7142
4.361
3.8835
-6.6943
-6.0948
3.0134
-8.0591
-7.462
-8.4241
-3.1699
-2.7126
-2.2322
-2.3799
-2.9474
-0.3256
-0.8289
-0.9748
-0.4841
1.6426
1.2247
1.9252
1.5781
6.8022
6.2288
8.7413
8.6247
9.4535
7.7409
7.5163
-5.3605
3.2002
3.2465
1.9434
8.8071
-8.7969
-7.7789
-1.0546
1.7971
1.0256
1.9248
0.5169
0.3924
1.7073
-1.9232
0.1513
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1.1478
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0.7035
0.1488
0.571
0.0125
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1.4807
1.0996
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0.7639
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0.7144
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0.804
2.1475
1.2435
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1.4772
0.9312
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0.9441
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1.8318
2.3068
1.889
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0.7743
1.1154
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0.9564
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0.5292
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0.1639
0.8171
0.2493
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1.0793
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0.7083
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0.1538
0.8462
0.5667
0.0951
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0.0882
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0.4166
0.4731
0.3746
-0.8085
0.5769
0.3105
-0.8919
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1.6892
1.7068
-0.6484
-2.0466
1.6727
0.2243
-1.9873
-2.0083
-1.0666
-1.027
1.4246
1.5193
1.1263
-0.4763
-0.2655
1.1713
-0.3418
0.3745
-1.2555
-1.2403
1.5268
-0.2366
0.5083
-2.2494
0.7394
-1.3924
Conformer
ID
11
2.1
PubChem
ncbi.nlm.nih.gov
2009.12.11
00073FDC00000001
Energy
MMFF94 NoEstat
7
1.7.2
Szybki
openeye.com
2012.11.26
56.5535
Feature
Self Overlap
7
2.1
PubChem
ncbi.nlm.nih.gov
2012.11.26
50.874
Fingerprint
Shape
2
2.1
PubChem
ncbi.nlm.nih.gov
2012.11.26
10 15 17418372506767411941
10299344 5 18343018886971410311
10391435 84 17240486939714441147
10595046 47 18340768148341493851
11135609 127 18263647428772720692
11315181 36 18411700977193433465
11456790 92 10447930580939945182
11497681 19 18410849997473444463
11524674 6 15626218044780602983
12013929 94 18340487867872651843
12082328 90 17989207014895336317
12089408 11 18342176652880664369
12664476 115 17967812761314716644
12838862 33 16081361985913315217
14118638 360 16660636302805038400
14142895 15 18335143128553174276
14251764 18 18410855464423135588
14251764 46 18410573993741392242
14444916 359 14764349340529342749
14856354 85 17560797762994117327
14933364 13 18341894082302483257
15183329 4 18410855447333009299
15419008 47 16081361968981620293
15461852 350 18343023302830624469
15728490 51 18409166641029501487
1577012 14 18341050727214788713
15840311 113 18411140264955202324
15849732 13 17894911841272501063
15980000 95 17676489445378690805
16120349 18 18186522129205917948
18335252 98 18408886230835155203
18365409 1 18263367052342468630
19301679 30 17273986740305429022
20105231 36 16128659651925372430
20771845 140 17131543944081900294
21095086 128 18413387631212345438
21150785 3 18408322189675119683
21315763 28 18343301452848838816
21360443 126 17895197740239898810
21772524 286 17487913207527764249
21781051 124 16558752359756278822
21792934 111 12179841732116717958
21792938 703 17968944218793286963
21792961 116 16415483723088747305
22224240 67 18113336414588858514
232437 2 18343019978742539918
23516275 137 17986974988964460695
24771293 8 17967819327338393973
335507 130 18060137656864819135
395649 100 18187084005254478819
4073 2 18113905987171237450
4325135 7 18342454850844969839
4625314 4 18409446990196759877
5758199 1 18334576836735531538
6057620 51 18409450284294452625
6081469 158 15647048245245271126
67123 10 18341894103761209504
9663363 56 16298382474354592637
9831232 110 18055918684599634630
Shape
Multipoles
8
1.8.3
OEShape
openeye.com
2012.11.26
593.16
31.4
1.88
1.05
11.92
0.65
-0.22
1.75
-4.49
-1.35
0.12
0.01
-0.18
-1.79
Shape
Self Overlap
7
2.1
PubChem
ncbi.nlm.nih.gov
2012.11.26
1288.314
Shape
Volume
7
1.8.3
OEShape
openeye.com
2012.11.26
324.8
Conformer
RMSD
7
2009.12.11
0.8
Diverse Conformer
ID List
6
2012.02.08
1
142
105
153
4
102
181
132
72
95
12
104
175
130
139
106
69
147
174
141
131
159
37
119
107
180
26
78
52
112
14
94
66
75
83
21
23
157
183
170
74
9
164
116
148
123
121
71
45
31
81
3
127
100
108
77
176
47
56
160
122
152
154
8
30
70
167
64
128
10
73
93
34
46
82
84
101
156
125
103
133
44
79
2
161
134
155
7
158
113
145
182
140
90
42
49
151
138
166
11
50
48
177
118
16
86
61
59
117
6
58
89
19
20
80
173
27
143
88
179
13
68
172
18
76
65
169
28
92
149
178
98
136
33
41
162
144
163
109
135
24
60
91
126
96
53
43
150
97
85
120
110
51
38
165
171
129
29
63
32
114
168
35
39
40
55
36
99
137
17
57
15
146
87
54
124
22
62
67
25
5
115
111
Charge
MMFF94 Partial
2
1.7.6
OEChem
openeye.com
2012.02.08
31
1 -0.19
12 0.27
13 0.27
14 0.27
15 0.11
16 0.14
17 -0.12
18 0.3
19 0.28
2 -0.02
21 0.06
22 0.45
24 0.62
25 0.03
26 0.14
27 -0.15
28 0.14
29 -0.15
3 -0.68
30 -0.15
31 0.19
4 -0.57
5 -0.81
52 0.15
56 0.4
57 0.15
58 0.15
6 -0.42
7 -0.41
8 -0.62
9 0.18
Count
Effective Rotor
7
1.7.6
OEChem
ncbi.nlm.nih.gov
2012.01.18
6
Features
Pharmacophore
2
ImplicitMillsDean merged
1.8.1
OEShape
openeye.com
2012.02.08
10
1 3 acceptor
1 3 donor
1 4 acceptor
1 5 cation
1 7 acceptor
5 2 7 15 23 26 rings
6 23 26 27 29 30 31 rings
6 5 9 10 11 12 13 rings
6 6 18 19 20 21 22 rings
6 6 8 17 22 24 25 rings
31
1
0
1
0
0
0
0
1
1