46919619
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82
83
17
17
8
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36
23
26
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32
10
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32
11
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17
13
44
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27
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41
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83
1
1
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2
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2
1
1
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1
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1
1
1
2
1
2
1
1
1
1
23
3
21
24
25
1
1
2
5
10
1
2
3
4
5
6
7
8
9
10
11
12
13
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15
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83
-2.6
-2.8561
-2.67
4.4335
-3.8907
5.16
1.2177
4.7846
-3.8803
3.9968
2.8135
3.6315
1.5117
2.2986
4.8378
6.3084
4.4228
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7.5477
6.0291
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6.0037
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Conformer
ID
11
2.1
PubChem
ncbi.nlm.nih.gov
2010.09.21
02CBEFC300000001
Energy
MMFF94 NoEstat
7
1.7.2
Szybki
openeye.com
2012.11.26
131.1038
Feature
Self Overlap
7
2.1
PubChem
ncbi.nlm.nih.gov
2012.11.26
50.749
Fingerprint
Shape
2
2.1
PubChem
ncbi.nlm.nih.gov
2012.01.18
10675989 125 17611181950400939649
11059845 2 18339657732250728376
11062273 23 18343301427918298675
11136131 41 17909272726104614409
11763715 3 17764283078012361799
12788726 201 18339656538234956755
12988421 55 18127425655334556949
14068700 675 18052545365682204551
14950920 106 16988267755321641664
15200665 1 18411411796439161363
15320294 125 18059012903245278572
15513586 35 17559374886698783269
16114785 44 18334298695460739283
16990350 14 17689151631357493913
18393751 57 18268977839336649513
18470217 77 18118142285060519035
19053607 189 17910101744350025285
21033648 29 18265328585212212841
21120745 212 18051956044956087799
21133410 221 17533531995517256880
3383291 50 18409733972007781457
3418910 222 17977670801685020112
376196 1 17897168142117025639
4144715 1 18410012105478505530
44249763 50 17604447252940029804
4616759 239 18189075147876337938
508706 21 18187377510006979872
5219985 13 18264485277389990789
6058803 2 18131065988231534478
6371380 46 17975967979979624662
6700243 42 17756669037199393166
9555976 147 18341067237406775882
9896288 288 18342170090477150531
Shape
Multipoles
8
1.8.3
OEShape
openeye.com
2012.11.26
809.97
16.92
9.71
2.46
30.73
5.55
0.08
-12.92
-5.43
-26.59
-2.01
3.72
0.07
-1.87
Shape
Self Overlap
7
2.1
PubChem
ncbi.nlm.nih.gov
2012.11.26
1706.934
Shape
Volume
7
1.8.3
OEShape
openeye.com
2012.11.26
454.9
Conformer
RMSD
7
2010.09.21
1.2
Diverse Conformer
ID List
6
2012.02.08
1
248
255
3
210
229
320
295
168
178
224
242
325
92
261
233
180
296
15
108
31
294
155
288
273
253
198
324
34
286
22
79
291
106
81
206
149
175
70
303
202
280
129
260
177
72
270
226
292
272
185
247
76
156
216
172
317
148
217
69
240
267
130
222
313
238
134
117
152
283
140
265
262
67
204
87
277
213
269
302
147
173
164
315
298
125
321
246
212
74
309
116
86
227
142
287
27
166
151
176
100
50
257
28
316
158
256
221
163
322
41
193
241
274
49
190
104
80
218
235
207
329
170
167
209
65
249
254
11
162
205
75
5
208
12
214
244
171
107
143
115
159
144
94
78
199
201
251
230
300
138
10
84
307
239
195
326
197
33
23
109
91
112
157
299
276
189
282
85
183
121
82
128
21
306
252
278
188
304
211
234
245
186
102
46
182
215
279
97
88
8
305
301
150
133
73
118
141
228
53
139
96
103
77
114
225
271
56
293
312
318
323
268
122
243
24
290
289
66
196
184
258
57
220
308
42
47
99
44
39
284
59
71
123
263
281
203
113
9
16
297
154
310
29
58
275
119
127
165
64
48
25
169
124
63
191
330
192
14
132
18
194
259
93
161
35
327
52
314
20
328
237
231
98
120
111
43
236
51
36
174
90
223
62
89
200
219
285
136
55
153
319
30
131
181
37
110
135
95
266
19
126
179
232
45
40
2
54
101
137
60
187
250
17
160
7
83
105
26
13
6
145
38
32
311
68
61
4
146
264
Charge
MMFF94 Partial
2
1.7.6
OEChem
openeye.com
2012.02.08
43
1 -0.18
10 0.33
13 0.27
14 0.27
15 0.27
16 0.27
17 0.57
18 0.27
2 -0.18
23 0.42
24 0.3
25 -0.14
26 0.28
27 0.3
28 0.3
29 0.3
3 -0.56
30 -0.15
31 -0.15
32 0.54
33 0.18
34 -0.15
35 0.09
36 0.18
37 -0.15
38 -0.15
39 -0.15
4 -0.57
40 -0.15
41 -0.15
5 -0.57
6 -0.81
7 -0.81
76 0.15
77 0.15
78 0.15
79 0.15
8 -0.66
80 0.15
81 0.15
82 0.15
83 0.15
9 -0.66
Count
Effective Rotor
7
1.7.6
OEChem
ncbi.nlm.nih.gov
2012.01.18
12.6
Features
Pharmacophore
2
ImplicitMillsDean merged
1.8.1
OEShape
openeye.com
2012.02.08
10
1 3 acceptor
1 4 acceptor
1 5 acceptor
1 6 cation
1 7 cation
6 25 30 31 33 34 36 rings
6 3 9 23 24 26 27 rings
6 35 37 38 39 40 41 rings
6 6 15 16 19 20 22 rings
6 7 10 11 12 13 14 rings
41
1
1
0
0
0
0
0
1
1