46820279
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13
28
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1
2
5
10
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-2.3016
3.2357
2.2353
-3.6003
-6.2012
3.3862
5.2722
-0.9076
4.5435
4.2621
5.2185
1.2359
5.7891
2.3132
5.8416
-0.143
-2.0653
-3.1299
7.3143
-0.7292
-2.8535
-4.4352
-3.8824
-5.1877
-5.464
-2.2407
-7.5059
4.689
3.3367
4.1738
5.7471
1.2242
1.4996
6.6904
5.9402
5.7051
6.0738
5.7386
5.2999
7.7312
7.8874
7.4572
-0.3248
-1.8229
-4.7214
-6.454
-1.8899
-1.5899
-2.2
-7.5563
-7.8577
-8.1863
3.1079
-1.0138
2.1304
-2.9268
-2.1399
1.5983
-1.0692
1.4772
1.0215
-0.4562
-2.4585
2.661
1.2072
2.112
-3.3793
2.6083
1.6293
0.654
-3.0814
3.6004
-0.6825
1.0487
-1.6245
-1.2298
0.1069
-3.2472
-1.6538
1.5032
1.5749
-2.7431
-2.5475
2.1013
3.6976
0.849
2.2657
0.6628
-0.5255
-4.4177
-3.2912
-3.8022
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-2.0801
4.5599
-0.9426
2.0757
0.4854
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-3.0623
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-1.2524
-0.9365
-2.511
0.8726
-0.2804
1.1779
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0.059
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0.8309
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0.1027
1.222
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0.0344
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0.0505
0.3384
-0.8149
0.3685
0.8391
-1.782
1.3884
2.177
-1.9063
-1.2046
-0.4807
-1.2266
-1.9355
1.1356
0.515
-0.7694
-0.7739
0.8667
-0.4813
0.6871
-0.4657
0.5389
0.5688
-1.721
0.0466
-1.0169
1.3864
-0.3808
0.3313
Conformer
ID
11
2.1
PubChem
ncbi.nlm.nih.gov
2010.07.16
02CA6BB70000000C
Energy
MMFF94 NoEstat
7
1.7.2
Szybki
openeye.com
2012.11.26
68.3056
Feature
Self Overlap
7
2.1
PubChem
ncbi.nlm.nih.gov
2012.11.26
50.752
Shape
Multipoles
8
1.8.3
OEShape
openeye.com
2012.11.26
521.08
18.54
5.02
0.92
8.38
0.63
-0.06
19.98
-1.76
1.86
-0.05
0.58
-0.13
-1.9
Shape
Self Overlap
7
2.1
PubChem
ncbi.nlm.nih.gov
2012.11.26
1067.157
Shape
Volume
7
1.8.3
OEShape
openeye.com
2012.11.26
304.4
Conformer
RMSD
7
2010.07.16
1
Diverse Conformer
ID List
6
2012.02.08
12
87
91
211
257
103
162
92
122
185
88
182
65
199
112
34
169
109
137
203
230
55
117
201
21
56
143
177
207
105
90
84
131
134
94
124
74
204
198
212
83
249
222
125
148
192
265
138
111
123
113
175
263
81
140
72
6
232
43
252
132
200
172
100
97
147
96
119
30
234
158
187
244
205
29
243
246
104
15
255
2
127
46
173
236
33
239
208
19
191
7
174
242
5
39
98
25
231
241
115
106
247
240
1
216
32
82
186
260
262
93
180
225
219
48
136
13
69
196
154
76
170
141
159
85
163
258
176
161
61
80
167
108
194
195
223
193
11
120
62
68
18
197
228
79
44
57
4
27
22
155
217
250
49
209
133
37
229
233
26
58
36
150
73
59
118
10
153
126
215
151
40
206
190
20
54
60
31
261
47
142
266
38
168
99
67
256
107
235
254
264
116
214
102
248
42
221
89
63
41
149
77
189
75
121
184
71
183
213
23
8
237
86
164
70
78
145
160
51
220
24
188
14
64
267
128
52
224
114
245
130
28
144
95
165
3
45
179
101
227
110
66
226
181
35
152
259
139
9
218
53
17
157
238
202
210
166
251
146
253
50
16
171
135
178
156
129
Charge
MMFF94 Partial
2
1.7.6
OEChem
openeye.com
2012.02.08
30
1 -0.08
10 0.57
11 0.3
12 0.24
14 0.57
16 0.05
17 0.33
18 0.05
2 -0.57
20 -0.11
21 -0.15
22 -0.15
23 0.08
24 0.08
25 -0.15
26 0.28
27 0.28
29 0.37
3 -0.57
37 0.37
4 -0.36
43 0.15
44 0.15
45 0.15
46 0.15
5 -0.36
6 -0.73
7 -0.73
8 -0.57
9 0.36
Count
Effective Rotor
7
1.7.6
OEChem
ncbi.nlm.nih.gov
2012.01.18
11
Features
Pharmacophore
2
ImplicitMillsDean merged
1.8.1
OEShape
openeye.com
2012.02.08
10
1 19 hydrophobe
1 2 acceptor
1 3 acceptor
1 4 acceptor
1 5 acceptor
1 6 donor
1 7 donor
1 8 acceptor
5 1 8 16 17 20 rings
6 18 21 22 23 24 25 rings
27
1
0
1
0
0
0
0
1
4