4479938
1
2
3
4
5
6
7
8
9
10
11
12
13
14
15
16
17
18
19
20
21
22
23
24
25
26
27
28
29
30
31
32
33
34
35
36
37
38
39
40
41
42
43
53
8
8
8
7
7
7
7
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
2
2
3
4
5
5
6
6
7
8
8
8
9
9
10
10
11
11
11
12
12
13
13
14
15
16
16
16
17
17
18
18
19
19
20
21
22
23
23
26
26
27
27
28
22
5
24
24
25
9
37
7
10
25
17
42
43
12
13
14
15
18
19
25
14
29
15
30
31
32
22
23
24
20
21
20
33
21
34
35
36
26
27
38
28
39
28
40
41
1
1
1
2
2
1
1
2
1
1
1
1
1
2
1
2
1
2
1
1
1
1
2
1
1
1
1
2
1
2
1
1
1
2
1
1
1
2
1
1
1
1
2
1
1
2
5
10
1
2
3
4
5
6
7
8
9
10
11
12
13
14
15
16
17
18
19
20
21
22
23
24
25
26
27
28
29
30
31
32
33
34
35
36
37
38
39
40
41
42
43
6.547
3.5574
5.0932
-5.0441
2.6771
-2.5744
-3.2923
-8.1321
1.3549
-1.2556
-5.5255
0.4479
0.9535
-0.8607
-0.3551
5.6871
-7.2568
-5.0459
-6.8707
-5.9117
-7.7363
6.5041
5.6779
4.7698
-4.6226
7.3442
6.5181
7.3512
0.7486
1.6418
-1.5607
-0.6595
-4.0057
-7.2693
-5.5263
-8.7824
2.9283
5.0324
8.0026
6.5236
8.0052
-9.1079
-7.7857
-1.8587
-0.2187
-0.6668
-2.105
-1.0023
-1.9194
-0.9453
3.1541
-1.2347
-1.6903
-0.0038
-1.8736
-0.8241
-2.1021
-1.0524
0.7116
2.0933
1.1203
-0.0794
2.1688
0.9692
0.1813
2.064
-0.1392
-1.0967
1.0333
2.9159
2.4006
-2.1981
-0.3266
-2.601
-0.7302
1.2174
-0.9438
3.0398
0.8988
-1.2439
2.4742
0.6561
3.9805
3.0642
3.0987
3.9685
-1.2172
0.4205
2.082
-1.2564
1.1349
-0.574
-0.263
0.6043
0.7034
-0.1459
-0.3313
1.5489
-0.5676
1.1231
-0.9934
0.2303
0.2911
0.341
-0.6924
0.6522
-0.3813
-0.7486
0.5201
1.0289
-0.6568
-1.4658
-0.197
-1.1899
2.5418
-1.2457
1.788
-1.9857
0.6392
-1.2169
1.1762
-0.6684
2.087
1.2915
-2.2444
0.0177
-1.7481
0.3445
1.0937
Conformer
ID
11
2.1
PubChem
ncbi.nlm.nih.gov
2009.12.11
00445BC200000001
Energy
MMFF94 NoEstat
7
1.7.2
Szybki
openeye.com
2012.11.26
98.8401
Feature
Self Overlap
7
2.1
PubChem
ncbi.nlm.nih.gov
2012.11.26
45.671
Fingerprint
Shape
2
2.1
PubChem
ncbi.nlm.nih.gov
2012.11.26
10 15 14706925155214177766
10454371 7 18202285818565022713
10693767 8 11527943456644707284
10906281 52 18186805802884279810
11135609 127 18130218385558853512
11386260 185 15769766996836448384
11408170 253 18202007590668666697
11991303 11 16486967461728882285
12035758 1 15213301928277323643
12539765 74 18341054034065852287
12895837 130 18412262848856628379
13726171 33 15721105984367949100
13782708 43 9439412323918454622
14251757 52 18408602578520970072
14394314 77 18260831514130649149
14849402 71 18041562545980020517
14918687 75 10519993648111432124
15183329 4 17346606270141378714
15188451 53 10231763279773785238
15276724 80 18261669281612779580
15326921 28 11748864953067186391
15461852 350 17988919012254054287
15475509 8 18336271167485716206
1577012 14 18335697260559149379
15840311 113 18260268516794398093
16989713 51 17130414904321791615
16990366 60 7853275537413067253
16994733 274 18408599283801032665
1768 124 8790892886951023560
18603816 31 11891340894159947825
190975 80 11169918294512668646
2026 5 11311786059326077933
21424621 283 18334860519357347011
21585482 111 18188769427810052829
21637258 2 10015864284265658691
21781055 127 18335695036926491138
22149856 69 14924222660176070343
22224240 67 16732698355293664427
23081809 10 18336532898071077146
23569943 247 11167681879039957389
255183 313 14634868677978556611
3014063 24 11023832773210188200
3711267 37 18411427232082546880
394071 54 17240482559422740892
397830 11 12179847212347430614
3986486 107 18337404829058073540
406291 66 10663826269149478876
4073 2 18334297582669214011
4107672 100 17917147312028759119
4403749 210 17458062682298320451
445580 37 18130790062194275569
4756326 101 17201064046009236608
5718773 13 10015863180495564489
5758199 1 17967532380768409795
5911458 16 18408044013333941373
59682541 35 17022626381935832689
59682541 52 17275108310753608958
6328613 192 18410292536060868161
9689198 14 18335426763687503083
Shape
Multipoles
8
1.8.3
OEShape
openeye.com
2012.11.26
550.63
28.22
3.13
1.39
13.34
1.66
-0.25
22.36
6.37
0.06
-0.02
-1.73
-0.48
-1.77
Shape
Self Overlap
7
2.1
PubChem
ncbi.nlm.nih.gov
2012.11.26
1174.084
Shape
Volume
7
1.8.3
OEShape
openeye.com
2012.11.26
310.4
Conformer
RMSD
7
2009.12.11
0.8
Diverse Conformer
ID List
6
2012.02.08
1
289
326
374
71
222
370
140
21
287
46
298
244
285
77
343
179
304
82
344
362
330
282
95
313
299
27
139
125
256
357
268
35
40
273
158
24
358
301
333
126
122
120
156
162
371
84
45
342
34
281
152
316
8
81
14
375
317
16
160
217
80
323
240
13
28
159
350
15
203
128
43
266
219
276
227
328
10
51
356
230
180
250
7
270
116
300
196
25
117
58
65
279
31
234
307
61
191
311
238
137
50
106
245
292
48
199
147
306
23
9
349
214
79
98
142
100
30
369
154
57
315
109
141
172
352
297
138
264
314
44
94
36
325
26
99
257
111
206
293
114
318
365
337
29
283
377
56
295
218
255
200
267
224
33
2
226
175
127
47
4
78
72
359
367
144
284
17
339
136
165
68
178
309
145
113
90
163
296
11
85
3
205
305
340
280
118
155
89
182
64
204
60
263
88
6
53
91
338
73
41
241
332
272
166
243
20
18
346
290
192
39
55
252
376
146
67
211
167
334
265
278
215
331
37
107
5
327
233
52
151
364
207
174
212
286
104
373
102
360
223
216
176
32
194
195
121
76
112
312
42
105
101
119
143
221
115
148
92
93
220
324
69
59
190
124
237
22
347
249
225
38
12
231
153
308
361
242
351
336
75
83
185
208
103
123
229
131
157
302
288
348
201
329
70
150
181
66
108
63
345
74
303
202
173
129
96
87
253
149
368
260
19
184
259
86
239
169
130
258
248
321
372
188
291
341
363
275
232
183
322
171
274
269
320
193
277
235
170
197
261
251
246
54
378
254
209
310
354
135
49
262
97
210
133
335
247
228
132
236
168
271
110
355
187
62
164
134
213
177
186
353
198
319
189
161
294
366
Charge
MMFF94 Partial
2
1.7.6
OEChem
openeye.com
2012.02.08
43
1 -0.08
10 0.18
11 0.09
12 -0.15
13 -0.15
14 -0.15
15 -0.15
16 0.09
17 0.1
18 -0.15
19 -0.15
2 -0.13
20 -0.15
21 -0.15
22 0.08
23 -0.15
24 0.63
25 0.69
26 -0.15
27 -0.15
28 -0.15
29 0.15
3 -0.57
30 0.15
31 0.15
32 0.15
33 0.15
34 0.15
35 0.15
36 0.15
37 0.4
38 0.15
39 0.15
4 -0.57
40 0.15
41 0.15
42 0.4
43 0.4
5 -0.52
6 -0.18
7 -0.21
8 -0.9
9 0.1
Count
Effective Rotor
7
1.7.6
OEChem
ncbi.nlm.nih.gov
2012.01.18
7
Features
Pharmacophore
2
ImplicitMillsDean merged
1.8.1
OEShape
openeye.com
2012.02.08
9
1 1 hydrophobe
1 3 acceptor
1 4 acceptor
1 7 donor
1 8 cation
1 8 donor
6 11 17 18 19 20 21 rings
6 16 22 23 26 27 28 rings
6 9 10 12 13 14 15 rings
28
0
0
0
0
0
0
0
1
5