4141159
1
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9
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1
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1
1
1
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1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
5
1
1
2
3
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17
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33
8
10
13
35
12
17
46
16
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22
9
12
34
11
36
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11
38
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15
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16
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51
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28
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31
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29
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32
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32
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65
66
1
2
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1
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1
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1
1
2
1
1
1
1
1
1
8
5
9
12
34
3
1
14
16
17
18
47
3
1
16
7
14
20
51
3
1
2
5
10
1
2
3
4
5
6
7
8
9
10
11
12
13
14
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65
66
5.4173
-1.476
2.2949
0.6631
-4.4148
-1.8368
1.7637
-4.2051
-5.5683
-5.8799
-6.289
-3.108
-3.9033
0.1704
-4.0844
1.2839
-1.1301
0.5215
1.3093
2.3993
1.8342
2.2593
0.0292
1.6033
2.3315
3.4865
1.1592
0.3277
1.114
3.351
4.5061
4.4383
-0.3685
-3.9263
-3.8991
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-5.4992
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-6.4082
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-3.367
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-4.4501
-1.4332
0.0373
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0.8449
2.7039
3.0533
-0.5935
2.2151
1.4884
3.5813
0.3401
1.563
-0.0563
1.3452
3.2982
5.3534
0.0074
-0.7081
-1.2163
3.7005
-1.3587
-3.0034
-4.0518
1.1006
0.3724
-1.4704
0.9478
0.5114
0.8544
-0.075
-0.0796
2.388
0.3635
2.3806
-0.1241
-0.3107
0.1019
-1.0018
0.9077
-1.9173
-2.3153
0.941
-1.2559
1.8781
0.8809
-3.1893
0.6885
-0.4084
2.8215
1.8243
2.7946
-4.8965
1.9262
0.3396
1.3903
-0.1976
0.4037
1.8124
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-1.0948
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-1.0525
2.462
3.2121
1.2071
1.4473
2.4058
1.4991
3.2673
-0.2397
-1.6869
-2.956
1.796
-2.1045
1.9116
0.1432
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-3.7891
1.3454
-0.6056
3.5776
1.8035
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0.3182
1.2074
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0.032
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0.3106
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0.5963
0.1169
2.0984
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1.5558
1.9076
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0.8619
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2.566
3.2534
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3.9047
4.2474
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0.4954
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1.3013
0.2529
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0.3396
0.1261
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2.3875
2.5539
2.5321
-1.8306
-2.3219
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2.3144
3.5474
-2.6523
0.6937
-2.5013
-2.9404
4.6796
5.2901
-2.8717
0.4582
-2.4003
-0.7741
-1.9445
Conformer
ID
11
2.1
PubChem
ncbi.nlm.nih.gov
2009.12.11
003F306700000001
Energy
MMFF94 NoEstat
7
1.7.2
Szybki
openeye.com
2012.11.26
78.3505
Feature
Self Overlap
7
2.1
PubChem
ncbi.nlm.nih.gov
2012.11.26
50.773
Fingerprint
Shape
2
2.1
PubChem
ncbi.nlm.nih.gov
2012.11.26
10074138 170 16084473754250123104
10764073 3 14563624679675027088
11421498 54 18130793321758455409
11443803 9 18119234302123506308
11582403 64 18041281079418755208
12058002 1 18126014762857445098
12156800 1 17765123444230164178
12788726 201 16199047001927872257
14040222 75 15896948855383000071
14068700 675 17558552392309313070
14955137 171 16953072246450637922
15815584 197 17095249103101548429
16114785 44 17320147832995250536
17492 54 15337992165233328944
21033650 10 17273721843101322548
21716022 299 17488475070131057718
266924 78 17838380390468494214
376196 1 17968940936631105468
394222 165 18335421270704023586
59444896 2 17898825080549212722
Shape
Multipoles
8
1.8.3
OEShape
openeye.com
2012.11.26
639.3
10.32
4.33
3.72
15.56
4.79
4.56
-9.21
-6.17
-4.11
-2.74
-1.89
-0.74
-3.05
Shape
Self Overlap
7
2.1
PubChem
ncbi.nlm.nih.gov
2012.11.26
1357.355
Shape
Volume
7
1.8.3
OEShape
openeye.com
2012.11.26
359.3
Conformer
RMSD
7
2009.12.11
1
Diverse Conformer
ID List
6
2012.02.08
1
177
291
142
361
346
276
199
366
120
150
274
415
144
328
362
164
62
101
345
93
168
273
391
427
194
128
342
379
287
141
195
383
381
327
43
424
268
417
58
373
208
262
187
279
23
14
209
426
296
98
314
243
305
176
365
352
398
240
261
309
428
264
236
67
244
247
385
335
13
293
375
88
225
393
299
245
33
405
387
119
354
158
409
127
49
35
136
197
224
306
402
133
367
27
283
201
223
270
285
60
344
317
252
338
108
336
430
184
100
280
132
234
413
289
81
172
432
229
407
272
125
429
422
65
82
111
22
384
348
310
241
84
265
255
61
242
337
340
99
75
271
109
394
115
318
278
316
55
230
311
298
374
235
396
91
320
246
202
412
290
52
357
239
70
9
302
389
135
369
390
79
170
214
353
152
418
266
307
129
200
380
83
329
222
122
248
94
363
425
260
107
392
38
411
397
315
419
139
42
376
292
174
6
54
166
421
251
388
347
17
227
404
254
339
69
7
423
137
351
250
216
153
382
74
372
171
395
319
157
210
238
324
161
370
181
217
89
308
269
26
138
85
155
211
182
331
178
147
408
175
16
39
212
249
180
53
377
193
410
162
349
183
267
112
117
66
321
297
215
356
163
114
221
123
368
312
59
323
286
359
154
326
189
322
220
206
386
41
341
131
406
226
281
72
256
18
431
334
15
364
258
403
37
371
36
294
358
301
148
237
86
192
190
118
5
414
205
10
80
218
140
169
399
116
343
333
186
350
231
300
77
8
400
253
378
87
40
145
203
207
330
124
355
71
282
219
360
275
3
92
97
56
24
198
213
32
173
284
188
126
96
64
106
149
105
48
143
185
295
233
416
28
325
179
288
263
113
257
63
401
121
204
51
103
167
73
110
102
50
34
165
146
232
228
25
130
95
19
45
304
20
104
12
21
159
277
332
44
68
78
156
2
151
196
134
303
160
90
420
259
31
191
11
46
313
30
29
4
57
76
47
Charge
MMFF94 Partial
2
1.7.6
OEChem
openeye.com
2012.02.08
40
1 -0.19
10 0.5
12 0.3
13 0.5
14 0.2
16 0.44
17 0.57
18 -0.14
19 0.09
2 -0.57
20 -0.14
21 0.54
22 0.3
23 -0.15
24 -0.15
25 -0.15
26 -0.15
27 0.28
28 -0.15
29 -0.15
3 -0.57
30 -0.15
31 -0.15
32 0.19
33 0.28
35 0.45
4 -0.56
46 0.37
5 -0.96
54 0.15
55 0.15
56 0.15
57 0.15
6 -0.73
60 0.15
61 0.15
62 0.15
63 0.15
7 -0.66
8 0.5
Count
Effective Rotor
7
1.7.6
OEChem
ncbi.nlm.nih.gov
2012.01.18
10.6
Features
Pharmacophore
2
ImplicitMillsDean merged
1.8.1
OEShape
openeye.com
2012.02.08
10
1 2 acceptor
1 3 acceptor
1 4 acceptor
1 5 cation
1 5 donor
1 6 donor
5 5 8 9 10 11 rings
6 18 19 23 24 28 29 rings
6 20 25 26 30 31 32 rings
6 7 14 16 18 19 21 rings
33
3
0
3
0
0
0
0
1
2