3596056
1
2
3
4
5
6
7
8
9
10
11
12
13
14
15
16
17
18
19
20
21
22
23
24
25
26
27
28
29
30
31
32
33
34
35
36
37
38
39
40
41
42
43
44
45
46
47
48
49
50
51
52
53
54
55
56
57
58
59
60
61
62
63
64
65
66
67
68
69
16
16
8
8
8
8
8
8
7
7
7
7
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
2
2
2
2
7
8
9
9
9
10
10
10
11
11
12
12
13
13
13
13
14
14
15
15
16
16
17
17
18
18
19
19
20
20
21
21
22
23
24
25
26
26
27
27
30
30
31
31
32
32
33
33
34
34
34
35
35
35
36
37
38
39
40
40
40
41
41
41
3
4
11
26
5
6
12
27
28
29
20
28
52
21
29
53
28
54
29
55
14
15
42
43
16
18
17
19
22
44
23
45
24
46
25
47
22
24
23
25
48
49
50
51
30
32
31
33
36
56
37
57
38
58
39
59
36
38
40
37
39
41
60
61
62
63
64
65
66
67
68
69
2
2
1
1
2
2
1
1
2
2
1
1
1
1
1
1
1
1
1
1
1
1
1
1
2
1
2
1
1
1
1
1
2
1
2
1
2
1
2
1
1
1
1
1
2
1
2
1
1
1
1
1
2
1
2
1
2
1
1
2
1
1
1
1
1
1
1
1
1
1
1
1
2
5
10
1
2
3
4
5
6
7
8
9
10
11
12
13
14
15
16
17
18
19
20
21
22
23
24
25
26
27
28
29
30
31
32
33
34
35
36
37
38
39
40
41
42
43
44
45
46
47
48
49
50
51
52
53
54
55
56
57
58
59
60
61
62
63
64
65
66
67
68
69
7.9914
-7.9682
8.9263
8.411
-8.9056
-8.3921
5.6621
-5.6297
4.5736
-4.557
6.5753
-6.5416
0.006
1.2254
-1.1926
1.4261
-1.4123
2.1086
-2.0948
3.4508
-3.4201
2.5485
-2.5336
3.2311
-3.2162
7.3607
-7.3776
5.5835
-5.5508
6.8819
-6.9045
7.357
-7.3784
6.3732
-6.4337
6.3843
-6.4326
6.8593
-6.9064
5.8417
-5.9298
-0.2334
0.2554
0.7296
-0.7183
1.9452
-1.9357
2.7074
-2.6951
3.8833
-3.8664
4.6667
-4.649
6.4645
-6.4315
6.8777
-6.8905
7.7253
-7.7366
6.009
-6.0677
6.8561
-6.9127
5.4019
5.0536
6.6467
-6.7486
-5.1443
-5.495
0.3859
0.3638
0.7156
-0.4267
0.662
-0.4781
-1.2209
-1.2146
-1.5069
-1.5152
-0.2861
-0.3003
-4.6045
-3.7774
-3.7929
-3.4036
-3.4203
-3.4167
-3.4063
-2.2681
-2.2847
-2.6422
-2.661
-2.6555
-2.6471
1.896
1.8637
-1.0383
-1.0459
1.9127
1.9032
3.034
3.0227
4.2613
4.2609
3.1046
3.1017
4.2257
4.2212
5.5357
5.5424
-5.2779
-5.2876
-3.6905
-3.7152
-3.7144
-3.6908
-2.3476
-2.3762
-2.405
-2.3872
-1.2619
-1.2816
-0.1954
-0.2161
1.024
1.0136
3.0241
3.0128
3.1197
3.1201
5.1202
5.1175
6.1616
5.3439
6.096
6.0863
5.3617
6.1792
-0.53
0.5479
-1.5884
0.5953
1.6227
-0.5625
0.7081
-0.7043
-1.3427
1.3478
-1.2137
1.228
-0.0149
-0.3694
0.3431
-1.6857
1.6693
0.6319
-0.6482
-1.0164
1.0083
-2.0121
2.0043
0.3055
-0.3133
0.1378
-0.1221
-0.5006
0.5064
1.4363
-1.4338
-0.6504
0.6542
1.1839
-1.1933
1.9636
-1.9694
-0.1233
0.1186
1.7476
-1.7661
-0.8498
0.8092
-2.468
2.452
1.6636
-1.6851
-3.0464
3.0402
1.1305
-1.1355
-2.3254
2.3334
-2.2315
2.2464
2.0594
-2.0569
-1.6716
1.6797
2.9835
-2.9929
-0.7405
0.7331
0.9636
2.4837
2.2334
-2.2474
-2.5078
-0.9882
Conformer
ID
11
2.1
PubChem
ncbi.nlm.nih.gov
2009.12.11
0036DF1800000001
Energy
MMFF94 NoEstat
7
1.7.2
Szybki
openeye.com
2012.11.26
80.3709
Feature
Self Overlap
7
2.1
PubChem
ncbi.nlm.nih.gov
2012.11.26
71.176
Fingerprint
Shape
2
2.1
PubChem
ncbi.nlm.nih.gov
2012.11.26
11421887 103 18410288116487409821
11478447 147 17775568667139356656
11578821 258 18342179925946755913
12013929 29 17908143175586437117
12888983 3 18410573989447081040
14268113 111 18409447016152297044
15320295 198 18199478821640757226
20691028 202 18267867366799346602
3525247 18 18410572885641116124
3862424 121 9727639436042779786
3918712 181 18413671296770161474
4760202 170 18273222985276000630
6289498 60 18335702715125366080
636775 72 18334299751906681927
Shape
Multipoles
8
1.8.3
OEShape
openeye.com
2012.11.26
796.32
33.77
9.11
1.89
0.36
7.15
0
45.47
0
0.04
0.03
0.04
0.57
7.6
Shape
Self Overlap
7
2.1
PubChem
ncbi.nlm.nih.gov
2012.11.26
1689.637
Shape
Volume
7
1.8.3
OEShape
openeye.com
2012.11.26
443.6
Conformer
RMSD
7
2009.12.11
1.2
Diverse Conformer
ID List
6
2012.02.08
1
202
43
77
314
233
21
327
201
100
132
248
156
222
273
60
226
61
219
243
363
334
7
221
179
92
24
165
195
255
369
246
6
158
305
296
331
261
303
251
224
197
122
281
183
217
354
124
365
182
294
113
159
257
306
8
254
332
128
351
229
293
249
323
194
220
307
362
38
326
30
336
315
131
150
360
223
343
177
284
15
88
247
49
71
104
366
143
112
285
173
312
174
213
190
141
178
211
212
200
26
297
115
176
368
338
101
72
87
44
70
272
227
130
280
164
102
218
52
207
86
230
250
322
214
58
3
345
10
357
203
189
55
149
320
89
67
232
265
69
169
11
93
50
51
253
271
148
299
318
328
215
329
295
225
267
234
168
282
310
186
270
166
56
152
301
79
210
133
342
140
262
66
116
135
344
304
107
205
319
244
108
185
278
27
105
231
292
119
147
198
372
171
91
340
126
181
339
117
309
279
154
287
19
288
316
99
216
228
42
206
317
184
290
175
353
240
123
35
114
333
39
367
98
125
311
356
269
41
302
335
68
264
103
236
298
358
121
300
110
161
361
172
145
90
346
34
94
350
57
64
308
16
330
374
359
337
142
258
155
106
138
204
187
170
18
192
139
48
324
347
191
256
268
237
81
375
29
188
239
78
196
370
85
74
371
83
80
355
37
241
242
127
352
259
364
76
109
341
252
276
95
62
160
260
286
111
283
274
263
82
36
348
40
180
53
54
167
349
28
136
373
153
163
12
325
321
97
162
157
22
134
208
151
313
14
75
275
65
291
25
17
32
118
137
238
31
20
129
45
209
235
245
146
289
33
277
144
73
266
59
46
120
63
199
96
84
193
23
47
9
5
4
2
13
Charge
MMFF94 Partial
2
1.7.6
OEChem
openeye.com
2012.02.08
61
1 1.45
10 -0.55
11 -0.79
12 -0.79
13 0.29
14 -0.14
15 -0.14
16 -0.15
17 -0.15
18 -0.15
19 -0.15
2 1.45
20 0.12
21 0.12
22 -0.15
23 -0.15
24 -0.15
25 -0.15
26 -0.01
27 -0.01
28 0.87
29 0.87
3 -0.65
30 -0.15
31 -0.15
32 -0.15
33 -0.15
34 -0.14
35 -0.14
36 -0.15
37 -0.15
38 -0.15
39 -0.15
4 -0.65
40 0.14
41 0.14
44 0.15
45 0.15
46 0.15
47 0.15
48 0.15
49 0.15
5 -0.65
50 0.15
51 0.15
52 0.37
53 0.37
54 0.42
55 0.42
56 0.15
57 0.15
58 0.15
59 0.15
6 -0.65
60 0.15
61 0.15
62 0.15
63 0.15
7 -0.57
8 -0.57
9 -0.55
Count
Effective Rotor
7
1.7.6
OEChem
ncbi.nlm.nih.gov
2012.01.18
12
Features
Pharmacophore
2
ImplicitMillsDean merged
1.8.1
OEShape
openeye.com
2012.02.08
14
1 10 donor
1 11 donor
1 12 donor
1 3 acceptor
1 4 acceptor
1 5 acceptor
1 6 acceptor
1 7 acceptor
1 8 acceptor
1 9 donor
6 14 16 18 20 22 24 rings
6 15 17 19 21 23 25 rings
6 26 30 32 34 36 38 rings
6 27 31 33 35 37 39 rings
41
0
0
0
0
0
0
0
1
6