3569151
1
2
3
4
5
6
7
8
9
10
11
12
13
14
15
16
17
18
19
20
21
22
23
24
25
26
27
28
29
30
31
32
33
34
35
16
16
8
8
8
8
8
7
7
6
6
6
6
6
6
6
6
6
6
6
6
6
6
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
2
2
2
2
7
8
9
9
10
10
11
12
12
13
13
14
14
15
16
17
17
18
18
19
19
20
20
21
21
22
23
23
23
3
4
8
10
5
6
8
11
16
9
16
26
11
12
13
14
24
15
25
15
27
28
17
18
19
20
29
21
30
22
23
22
31
32
33
34
35
2
2
1
1
2
2
1
1
2
1
1
1
1
2
2
1
1
1
1
2
1
1
1
1
2
2
1
1
1
1
1
2
1
1
1
1
1
2
5
10
1
2
3
4
5
6
7
8
9
10
11
12
13
14
15
16
17
18
19
20
21
22
23
24
25
26
27
28
29
30
31
32
33
34
35
1.7235
1.5057
1.663
1.5696
1.279
1.3181
-1.4115
0.7372
-0.6299
3.2443
3.14
4.4726
4.26
5.6141
5.5087
-1.6521
-3.0244
-4.0484
-3.272
-5.35
-4.5735
-5.6125
-6.4615
4.559
4.1835
-0.7684
6.5958
6.4101
-3.8473
-2.4969
-4.7794
-6.6221
-6.2912
-7.4185
-6.5446
1.4758
-1.3169
1.991
2.3128
-1.4118
-2.4311
-0.6296
0.0779
0.2933
0.6201
-0.7183
1.2098
-1.5159
0.4192
-0.9325
-0.102
0.1226
-0.6919
1.1456
-0.4784
1.3591
0.5471
-1.346
2.2503
-2.5606
0.671
0.8514
-1.5299
-1.4958
1.8176
2.1616
0.7237
-1.6598
-0.8136
-2.2379
0.2899
-0.4763
1.6412
-0.8814
-1.9031
0.4286
1.7121
0.1619
-0.235
0.1109
-0.2567
0.3463
-0.4029
0.1952
-0.1764
0.6244
0.1464
0.6062
-0.7568
0.1526
-1.2105
-0.7558
0.6391
0.639
-0.6832
-1.1657
0.37
-0.2847
1.3098
-1.1117
-1.9128
-1.1171
1.6746
0.6194
0.0102
Conformer
ID
11
2.1
PubChem
ncbi.nlm.nih.gov
2009.12.11
003675FF00000002
Energy
MMFF94 NoEstat
7
1.7.2
Szybki
openeye.com
2012.11.26
38.5913
Feature
Self Overlap
7
2.1
PubChem
ncbi.nlm.nih.gov
2012.11.26
45.753
Fingerprint
Shape
2
2.1
PubChem
ncbi.nlm.nih.gov
2012.11.26
10 15 18263073461705426152
10366900 7 15574428838998547945
11421498 54 16630253510690215539
11578080 2 13913762808024398772
11646440 116 18060421330579832072
12011746 2 18408327670623056118
12166972 35 18343024410431592384
12236239 1 16702303451069482705
12403259 415 18410285943507770985
12616971 3 16558750152686459001
13402501 40 18334293162899043429
13533116 47 16845577483323934422
14170010 4 18342174492153697792
14341114 176 18411422821250392511
14573314 32 18040715840004970525
14863182 85 17203339887951779990
15183329 4 18040712528680338921
15537594 2 15482672360425002631
15788980 27 18272365373882925485
17349148 13 17489872630697535499
17844677 252 18334300868297609069
19489759 90 17458063759775376667
200 152 17917711284162810097
20645477 70 18271811185789654902
21033648 29 18339345427524545681
21033650 10 16734966514215416772
21267235 1 18201728319304622382
21279426 13 18190738631242844068
21285901 2 18261393287393938932
21315763 129 18187363224913974733
21623969 137 18130794468657057271
21709351 56 18409722997917512309
221357 26 18410568470899304973
23402539 116 17530962479960698719
23557571 272 18114183034373703741
23559900 14 18261106392263724865
3004659 81 17313663738359435914
351380 180 18259703410809591813
3545911 37 18413389856047583195
4325135 7 18343017826900666967
46194498 28 18114464556004659549
465052 167 18341896264805298142
5104073 3 18270398282897992497
5283173 99 18188768332192114589
542803 24 15770058337041650921
59755656 215 18113050528759901475
7495541 125 18334579061496903077
9999458 23 17894630400702637566
Shape
Multipoles
8
1.8.3
OEShape
openeye.com
2012.11.26
441.72
14.42
1.95
1.15
9.66
0.1
0.02
-1.74
0.38
-0.94
0.07
0.38
0.06
1.57
Shape
Self Overlap
7
2.1
PubChem
ncbi.nlm.nih.gov
2012.11.26
933.903
Shape
Volume
7
1.8.3
OEShape
openeye.com
2012.11.26
246.2
Conformer
RMSD
7
2009.12.11
0.6
Diverse Conformer
ID List
6
2010.05.05
2
11
14
9
5
4
7
13
12
1
16
10
6
3
8
15
Charge
MMFF94 Partial
2
1.7.6
OEChem
openeye.com
2012.05.21
32
1 1.45
10 -0.01
11 -0.01
12 -0.15
13 -0.15
14 -0.15
15 -0.15
16 0.54
17 0.09
18 -0.15
19 -0.15
2 1.45
20 -0.14
21 -0.15
22 -0.15
23 0.14
24 0.15
25 0.15
26 0.37
27 0.15
28 0.15
29 0.15
3 -0.65
30 0.15
31 0.15
32 0.15
4 -0.65
5 -0.65
6 -0.65
7 -0.57
8 -0.36
9 -0.35
Count
Effective Rotor
7
1.7.6
OEChem
ncbi.nlm.nih.gov
2012.01.18
3.2
Features
Pharmacophore
2
ImplicitMillsDean merged
1.8.1
OEShape
openeye.com
2012.05.21
9
1 3 acceptor
1 4 acceptor
1 5 acceptor
1 6 acceptor
1 7 acceptor
1 9 donor
5 1 2 8 10 11 rings
6 10 11 12 13 14 15 rings
6 17 18 19 20 21 22 rings
23
0
0
0
0
0
0
0
1
2