3550101
1
2
3
4
5
6
7
8
9
10
11
12
13
14
15
16
17
18
19
20
21
22
23
24
25
26
27
28
29
30
31
32
33
34
35
36
37
38
39
40
41
42
43
44
45
46
47
48
49
50
51
52
53
54
55
8
8
8
8
8
8
8
8
8
8
8
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
2
2
3
3
4
4
5
5
6
6
7
7
8
8
9
10
10
11
11
12
12
12
13
13
14
14
15
15
16
17
17
17
18
18
19
20
20
21
22
22
24
25
25
26
27
27
28
28
28
29
29
30
30
31
32
32
15
16
16
18
12
42
13
43
14
44
21
25
19
28
23
47
24
31
54
33
55
13
14
34
15
35
16
36
17
37
38
39
40
41
19
20
23
21
45
22
23
24
26
26
27
46
29
30
48
49
50
31
51
32
52
33
33
53
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
2
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
2
1
1
2
1
1
2
1
1
2
1
1
2
1
1
1
1
1
1
2
1
2
1
1
12
3
13
14
34
3
1
13
4
12
15
35
3
1
14
5
12
16
36
3
1
15
1
13
17
37
3
1
16
1
2
14
38
3
1
2
5
10
1
2
3
4
5
6
7
8
9
10
11
12
13
14
15
16
17
18
19
20
21
22
23
24
25
26
27
28
29
30
31
32
33
34
35
36
37
38
39
40
41
42
43
44
45
46
47
48
49
50
51
52
53
54
55
-3.3904
-2.7239
-6.2266
-5.3386
-5.4287
1.9233
-2.7565
-0.4652
2.0903
4.9941
7.5412
-4.9531
-5.0712
-4.4498
-3.767
-3.1604
-3.9078
-1.5781
-1.5898
-0.39
0.7869
0.7732
-0.4141
2.0288
3.1069
3.2227
4.2674
-3.0549
4.0882
5.5496
5.1845
6.6458
6.4632
-4.2684
-5.9202
-4.3114
-2.9535
-2.3973
-4.6858
-2.9747
-4.1521
-6.5183
-4.5938
-5.4333
-0.3637
4.1464
0.4089
-4.008
-2.2802
-3.1517
3.1007
5.7308
7.6362
5.8583
8.3415
-0.5277
0.4863
-2.821
-3.5659
-0.1486
0.1066
3.0365
4.1484
3.8422
-3.856
-2.8026
-2.4678
-2.2994
-1.1805
-1.7347
-0.7236
-1.4103
1.0428
2.3284
0.3129
0.8717
2.1558
2.8899
2.7213
0.6333
1.8576
-0.2702
3.8582
-1.6548
0.256
-2.508
-0.5974
-1.9793
-3.2918
-1.6477
-1.313
-2.4652
-1.5006
-0.6563
-0.9855
-2.3003
-3.6297
-4.1572
0.1302
-0.6815
2.2622
4.427
4.3609
4.6185
3.2504
-2.0878
1.3255
-0.1727
-4.291
-2.2616
-0.7596
1.2495
1.1994
-1.4471
1.1623
0.3794
0.175
-0.8049
-1.2379
0.046
0.3939
0.6667
-0.8503
1.3194
-1.4305
0.6376
-2.9143
0.7594
0.2164
0.8054
0.3066
-0.2352
-0.2829
-0.7523
-0.1149
-0.6531
0.0186
1.3007
-0.0308
0.1941
0.0944
0.3195
0.2697
0.9029
-1.0878
2.3972
-1.3274
0.7744
-3.0771
-3.3003
-3.5016
0.7447
-1.2443
0.2311
1.2428
-1.0501
-1.1171
1.1147
1.4406
2.206
-0.1748
0.2602
0.4605
0.1495
0.5073
Conformer
ID
11
2.1
PubChem
ncbi.nlm.nih.gov
2009.12.11
00362B950000000B
Energy
MMFF94 NoEstat
7
1.7.2
Szybki
openeye.com
2012.11.26
119.667
Feature
Self Overlap
7
2.1
PubChem
ncbi.nlm.nih.gov
2012.11.26
91.454
Fingerprint
Shape
2
2.1
PubChem
ncbi.nlm.nih.gov
2012.11.26
10050765 1 18408891732794600904
10411042 1 18334862718623163280
10622 236 18410569591516224766
10693767 8 18194956564317347755
11135926 11 17974014143585337876
11409948 35 18192714678127575667
11410812 94 16153973666063025814
11497681 19 18412831266583200558
117089 54 18192439777870004499
12107183 9 18340220609263974505
12166972 35 17676774248838126854
12342043 65 17098359772215781507
12422481 6 17418101991904039726
12633257 1 16200151044751069267
13540713 5 18263667154344441324
13782708 43 18201716229045764762
13911987 19 17322973590437067813
14347332 77 18409735062132701009
14429380 30 18335423465485377338
1454969 45 18335986471906265852
14950920 106 16917061183325135290
15320294 125 17845947307438752159
15361156 5 17971496026261335252
15803439 3 16885231202064302085
17492 89 18408889563466104376
17686467 74 18409722968701995816
18393751 57 17693922395869433176
19141452 34 18195532484992881728
19246450 95 18200333043750384635
19301676 85 17687457971281421791
19301679 30 18339935878411902747
19303781 99 18334569174767836418
19315092 285 17703227459030252688
19319366 153 17691128557511704396
208703 8 18408322206966252675
21703447 108 18337098064681180864
23522609 53 18052855599776006744
23536364 44 18040986337456690319
23559900 14 18408317791729439816
23569914 152 18049406363717857847
24771750 20 16957898350819847044
34797466 226 16009874025336062895
3504750 166 18272652311926356195
38570 142 8430326778694167768
397830 11 18059842953953008314
4015057 19 18116157842639486793
46194498 28 17024590225029004045
50009960 94 17825086136182067066
5080951 261 18193820575215562468
513202 73 18411700954727053983
56633871 153 18192726548229550640
5937810 71 9006188319401207442
6058803 2 18265357103732371716
6431902 208 18410290302936720390
6691757 9 17916028945663540673
70251023 43 18336264651646113153
7970288 3 18339079423020255955
Shape
Multipoles
8
1.8.3
OEShape
openeye.com
2012.11.26
614.56
16.67
5.24
1.42
12.96
2.19
-0.73
-21.24
1.73
-1.35
-0.74
-2.64
-0.4
-2.29
Shape
Self Overlap
7
2.1
PubChem
ncbi.nlm.nih.gov
2012.11.26
1348.155
Shape
Volume
7
1.8.3
OEShape
openeye.com
2012.11.26
329.3
Conformer
RMSD
7
2009.12.11
1
Diverse Conformer
ID List
6
2012.02.08
11
466
545
555
523
140
704
348
535
237
232
455
594
336
251
590
552
413
509
531
35
36
411
600
696
493
539
365
544
414
449
27
275
82
517
412
146
417
387
432
520
498
264
663
439
383
309
32
354
253
667
102
147
55
300
24
440
371
118
279
87
226
109
222
174
39
491
2
14
62
515
434
583
532
164
88
702
112
175
26
40
205
46
13
290
669
495
366
57
323
104
4
558
93
56
12
660
540
74
138
59
98
123
34
81
391
7
95
126
3
60
45
144
16
1
538
249
92
68
145
33
65
121
124
6
459
238
169
128
10
148
91
41
5
Charge
MMFF94 Partial
2
1.7.6
OEChem
openeye.com
2012.02.08
43
1 -0.56
10 -0.53
11 -0.53
12 0.28
13 0.28
14 0.28
15 0.28
16 0.56
18 0.08
19 0.08
2 -0.36
20 -0.15
21 0.08
22 0.09
23 0.08
24 0.47
25 0.05
26 -0.14
27 0.03
28 0.28
29 -0.15
3 -0.68
30 -0.15
31 0.08
32 -0.15
33 0.08
4 -0.68
42 0.4
43 0.4
44 0.4
45 0.15
46 0.15
47 0.45
5 -0.68
51 0.15
52 0.15
53 0.15
54 0.45
55 0.45
6 -0.16
7 -0.36
8 -0.53
9 -0.57
Count
Effective Rotor
7
1.7.6
OEChem
ncbi.nlm.nih.gov
2012.01.18
5.2
Features
Pharmacophore
2
ImplicitMillsDean merged
1.8.1
OEShape
openeye.com
2012.02.08
18
1 1 acceptor
1 10 donor
1 11 donor
1 2 acceptor
1 3 acceptor
1 3 donor
1 4 acceptor
1 4 donor
1 5 acceptor
1 5 donor
1 6 acceptor
1 7 acceptor
1 8 donor
1 9 acceptor
6 1 12 13 14 15 16 rings
6 18 19 20 21 22 23 rings
6 27 29 30 31 32 33 rings
6 6 21 22 24 25 26 rings
33
5
0
5
0
0
0
0
1
57