2887498 1 2 3 4 5 6 7 8 9 10 11 12 13 14 15 16 17 18 19 20 21 22 23 24 25 26 27 28 29 30 31 32 33 34 35 36 37 38 39 40 41 42 43 44 45 46 47 48 49 50 51 52 53 16 16 8 8 8 8 7 7 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 2 3 3 4 4 5 6 7 7 7 8 8 8 9 9 9 10 10 10 11 11 11 12 12 13 14 14 15 15 16 16 16 17 17 17 21 21 21 22 22 22 23 24 24 25 25 26 26 27 27 28 28 29 13 18 20 9 14 19 21 19 23 18 20 42 20 23 45 10 11 30 12 31 32 16 17 33 13 15 14 34 35 18 19 36 37 38 39 40 41 22 43 44 46 47 48 24 25 26 27 49 28 50 29 51 29 52 53 1 1 2 1 1 1 1 2 2 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 2 1 1 1 1 2 1 1 1 1 1 1 1 1 1 1 1 1 1 1 2 1 1 1 2 1 2 1 1 1 1 9 3 10 11 30 3 1 1 5 255 1 2 3 4 5 6 7 8 9 10 11 12 13 14 15 16 17 18 19 20 21 22 23 24 25 26 27 28 29 30 31 32 33 34 35 36 37 38 39 40 41 42 43 44 45 46 47 48 49 50 51 52 53 6.4103 7.9939 3.732 6.0531 7.6995 9.4939 7.9939 9.4939 3.732 4.5981 2.866 5.4641 5.4641 4.5981 6.4103 2 2.866 6.9939 6.721 8.4939 6.3638 5.696 9.9939 10.9939 11.4939 11.4939 12.4939 12.4939 12.9939 3.1951 4.9966 4.1996 2.866 4.1996 4.9966 1.69 1.4631 2.31 3.486 2.866 2.246 8.3039 6.9107 6.7464 9.8039 6.1574 5.2819 5.2345 11.1839 11.1839 12.8039 12.8039 13.6139 -1.6029 -2.5302 -1.2982 1.7014 1.1633 -3.3962 -0.7982 -1.6642 -0.2982 0.2018 0.2018 -0.2982 -1.2982 -1.7982 0.0066 -0.2982 1.2018 -0.7982 0.9571 -1.6642 2.6519 3.3962 -2.5302 -2.5302 -3.3962 -1.6642 -3.3962 -1.6642 -2.5302 -0.6082 0.6768 0.6768 -0.4182 -2.2731 -2.2731 0.2388 -0.6082 -0.8351 1.2018 1.8218 1.2018 -0.2612 2.3599 3.1398 -1.1272 3.8103 3.8577 2.9822 -3.9332 -1.1272 -3.9332 -1.1272 -2.5302 8 8 3 8 8 8 8 8 8 8 8 8 1 1 9 12 12 15 24 24 25 26 27 28 13 18 11 13 15 18 25 26 27 28 29 29 0 Compound Canonicalized 5 2011.04.04 1 Compound Complexity 7 E_COMPLEXITY 3.396 Cactvs xemistry.com 2012.02.08 610 Count Hydrogen Bond Acceptor 5 E_NHACCEPTORS 3.396 Cactvs xemistry.com 2012.02.08 6 Count Hydrogen Bond Donor 5 E_NHDONORS 3.396 Cactvs xemistry.com 2012.02.08 2 Count Rotatable Bond 5 E_NROTBONDS 3.396 Cactvs xemistry.com 2012.02.08 6 Fingerprint SubStructure Keys 16 extended 2 E_SCREEN 3.396 Cactvs xemistry.com 2012.02.08 00000371E07B380060000000000000000000000000012000000034400000000000004801C000001E04100000000D14A1D802338982C004088C0221D25800830080650819088811004CC888263AE0B5998631886EC10368E9E798FC6ECE80000000000000000000000000000000000000000000 IUPAC Name Allowed 1 2.1.0 LexiChem openeye.com 2012.02.08 ethyl 2-(benzoylcarbamothioylamino)-5-isopropyl-5,7-dihydro-4H-thieno[2,3-c]pyran-3-carboxylate IUPAC Name CAS-like Style 1 2.1.0 LexiChem openeye.com 2012.02.08 2-[[benzamido(sulfanylidene)methyl]amino]-5-propan-2-yl-5,7-dihydro-4H-thieno[2,3-c]pyran-3-carboxylic acid ethyl ester IUPAC Name Preferred 1 2.1.0 LexiChem openeye.com 2012.02.08 ethyl 2-(benzoylcarbamothioylamino)-5-propan-2-yl-5,7-dihydro-4H-thieno[2,3-c]pyran-3-carboxylate IUPAC Name Systematic 1 2.1.0 LexiChem openeye.com 2012.02.08 ethyl 2-(phenylcarbonylcarbamothioylamino)-5-propan-2-yl-5,7-dihydro-4H-thieno[2,3-c]pyran-3-carboxylate IUPAC Name Traditional 1 2.1.0 LexiChem openeye.com 2012.02.08 2-(benzoylthiocarbamoylamino)-5-isopropyl-5,7-dihydro-4H-thieno[2,3-c]pyran-3-carboxylic acid ethyl ester InChI Standard 1 1.0.4 InChI nist.gov 2012.02.08 InChI=1S/C21H24N2O4S2/c1-4-26-20(25)17-14-10-15(12(2)3)27-11-16(14)29-19(17)23-21(28)22-18(24)13-8-6-5-7-9-13/h5-9,12,15H,4,10-11H2,1-3H3,(H2,22,23,24,28) InChIKey Standard 1 1.0.4 InChI nist.gov 2012.02.08 ZMKPIAINRVCEQF-UHFFFAOYSA-N Log P XLogP3-AA 7 3.0 sioc-ccbg.ac.cn 2012.02.08 4.9 Mass Exact 7 2.1 PubChem ncbi.nlm.nih.gov 2012.02.08 432.117749 Molecular Formula 1 2.1 PubChem ncbi.nlm.nih.gov 2012.02.08 C21H24N2O4S2 Molecular Weight 7 2.1 PubChem ncbi.nlm.nih.gov 2012.02.08 432.55626 SMILES Canonical 1 1.7.6 OEChem openeye.com 2012.02.08 CCOC(=O)C1=C(SC2=C1CC(OC2)C(C)C)NC(=S)NC(=O)C3=CC=CC=C3 SMILES Isomeric 1 1.7.6 OEChem openeye.com 2012.02.08 CCOC(=O)C1=C(SC2=C1CC(OC2)C(C)C)NC(=S)NC(=O)C3=CC=CC=C3 Topological Polar Surface Area 7 E_TPSA 3.396 Cactvs xemistry.com 2012.02.08 137 Weight MonoIsotopic 7 2.1 PubChem ncbi.nlm.nih.gov 2012.02.08 432.117749 29 1 0 1 0 0 0 0 1 11