24415312 1 2 3 4 5 6 7 8 9 10 11 12 13 14 15 16 17 18 19 20 21 22 23 24 25 26 27 28 29 30 31 32 33 34 35 36 37 38 39 40 41 42 43 44 45 46 47 48 49 50 51 17 16 8 8 8 7 7 7 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 2 2 3 3 4 4 5 6 6 7 7 7 8 9 9 9 10 10 11 12 13 13 14 14 15 16 16 17 18 19 20 20 20 21 21 22 22 24 24 25 26 26 27 28 28 29 29 30 30 32 32 32 33 27 14 18 10 20 11 32 23 15 18 23 26 44 31 12 13 16 11 17 12 34 17 35 15 21 22 19 36 37 19 31 23 38 39 24 40 25 41 25 42 43 27 28 29 30 45 33 46 33 47 48 49 50 51 1 1 1 1 1 1 1 2 1 2 1 1 1 3 2 1 1 2 1 1 1 2 1 1 2 2 2 1 1 1 1 1 1 1 1 1 1 1 2 1 1 1 2 2 1 1 1 1 2 1 1 1 1 1 16 9 36 19 31 18 2 1 1 5 255 1 2 3 4 5 6 7 8 9 10 11 12 13 14 15 16 17 18 19 20 21 22 23 24 25 26 27 28 29 30 31 32 33 34 35 36 37 38 39 40 41 42 43 44 45 46 47 48 49 50 51 13.7619 4.6783 10.7619 9.7619 12.7619 4.6783 12.7619 7.2619 7.7619 9.7619 9.2619 8.2619 8.2619 3.732 3.732 6.7619 9.2619 5.2619 6.2619 11.2619 2.866 2.866 12.2619 2 2 13.7619 14.2619 14.2619 15.2619 15.2619 6.7619 9.2619 15.7619 7.9519 7.9519 6.4519 9.5719 11.3695 10.6793 2.866 2.866 1.4631 1.4631 12.4519 13.9519 15.5719 15.5719 8.7249 8.9519 9.7988 16.3819 0 1.6708 0 -1.732 0 0.0613 1.732 2.5981 0 0 -0.866 -0.866 0.866 1.366 0.366 0 0.866 0.866 0.866 0.866 1.866 -0.134 0.866 1.366 0.366 1.732 0.866 2.5981 0.866 2.5981 1.732 -2.5981 1.732 -1.403 1.403 -0.5369 1.403 1.4766 1.0781 2.486 -0.754 1.676 0.056 2.269 3.135 0.3291 3.135 -2.2881 -3.135 -2.9081 1.732 8 8 8 8 8 8 8 8 8 8 8 8 8 8 8 8 8 8 8 8 8 8 2 2 6 6 9 9 10 10 11 13 14 14 15 21 22 24 26 26 27 28 29 30 14 18 15 18 12 13 11 17 12 17 15 21 22 24 25 25 27 28 29 30 33 33 0 Compound Canonicalized 5 2011.04.04 1 Compound Complexity 7 E_COMPLEXITY 3.402 Cactvs xemistry.com 2012.05.21 756 Count Hydrogen Bond Acceptor 5 E_NHACCEPTORS 3.402 Cactvs xemistry.com 2012.05.21 6 Count Hydrogen Bond Donor 5 E_NHDONORS 3.402 Cactvs xemistry.com 2012.05.21 1 Count Rotatable Bond 5 E_NROTBONDS 3.402 Cactvs xemistry.com 2012.05.21 7 Fingerprint SubStructure Keys 16 extended 2 E_SCREEN 3.402 Cactvs xemistry.com 2012.05.21 00000371E07B30004400000000000000000000000001600000003060C000000000005801F400001E06100000000C0EA1DE2232C7B2C81408BC0725725402A3F8A0612F3848983C76EE980FA6A2E5B39FC7382AE4D411FAE80790C0100E20000100000041104000020000008220000000000000 IUPAC Name Allowed 1 2.1.0 LexiChem openeye.com 2012.05.21 2-[4-[(E)-2-(1,3-benzothiazol-2-yl)-2-cyano-vinyl]-2-methoxy-phenoxy]-N-(2-chlorophenyl)acetamide IUPAC Name CAS-like Style 1 2.1.0 LexiChem openeye.com 2012.05.21 2-[4-[(E)-2-(1,3-benzothiazol-2-yl)-2-cyanoethenyl]-2-methoxyphenoxy]-N-(2-chlorophenyl)acetamide IUPAC Name Preferred 1 2.1.0 LexiChem openeye.com 2012.05.21 2-[4-[(E)-2-(1,3-benzothiazol-2-yl)-2-cyanoethenyl]-2-methoxyphenoxy]-N-(2-chlorophenyl)acetamide IUPAC Name Systematic 1 2.1.0 LexiChem openeye.com 2012.05.21 2-[4-[(E)-2-(1,3-benzothiazol-2-yl)-2-cyano-ethenyl]-2-methoxy-phenoxy]-N-(2-chlorophenyl)ethanamide IUPAC Name Traditional 1 2.1.0 LexiChem openeye.com 2012.05.21 2-[4-[(E)-2-(1,3-benzothiazol-2-yl)-2-cyano-vinyl]-2-methoxy-phenoxy]-N-(2-chlorophenyl)acetamide InChI Standard 1 1.0.4 InChI iupac.org 2012.05.21 InChI=1S/C25H18ClN3O3S/c1-31-22-13-16(12-17(14-27)25-29-20-8-4-5-9-23(20)33-25)10-11-21(22)32-15-24(30)28-19-7-3-2-6-18(19)26/h2-13H,15H2,1H3,(H,28,30)/b17-12+ InChIKey Standard 1 1.0.4 InChI iupac.org 2012.05.21 OPGXANVADFMWHG-SFQUDFHCSA-N Log P XLogP3-AA 7 3.0 sioc-ccbg.ac.cn 2012.05.21 5.7 Mass Exact 7 2.1 PubChem ncbi.nlm.nih.gov 2012.05.21 475.07574 Molecular Formula 1 2.1 PubChem ncbi.nlm.nih.gov 2012.05.21 C25H18ClN3O3S Molecular Weight 7 2.1 PubChem ncbi.nlm.nih.gov 2012.05.21 475.94672 SMILES Canonical 1 1.7.6 OEChem openeye.com 2012.05.21 COC1=C(C=CC(=C1)C=C(C#N)C2=NC3=CC=CC=C3S2)OCC(=O)NC4=CC=CC=C4Cl SMILES Isomeric 1 1.7.6 OEChem openeye.com 2012.05.21 COC1=C(C=CC(=C1)/C=C(\C#N)/C2=NC3=CC=CC=C3S2)OCC(=O)NC4=CC=CC=C4Cl Topological Polar Surface Area 7 E_TPSA 3.402 Cactvs xemistry.com 2012.05.21 113 Weight MonoIsotopic 7 2.1 PubChem ncbi.nlm.nih.gov 2012.05.21 475.07574 33 0 0 0 1 1 0 0 1 3