222284
1
2
3
4
5
6
7
8
9
10
11
12
13
14
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16
17
18
19
20
21
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32
33
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65
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71
72
73
74
75
76
77
78
79
80
8
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
2
2
2
2
3
3
3
4
4
4
5
5
5
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27
28
28
28
29
29
29
30
30
30
22
68
3
6
7
14
4
9
31
5
12
32
8
10
33
11
13
34
10
35
36
15
16
18
11
37
38
39
40
41
42
17
43
44
20
23
45
46
47
48
17
19
21
49
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51
52
53
54
22
55
56
24
57
58
22
59
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61
62
63
64
25
65
66
26
27
67
28
29
69
30
70
71
72
73
74
75
76
77
78
79
80
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
2
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
2
3
6
7
14
1
1
3
2
9
4
31
2
1
4
3
5
12
32
1
1
5
4
8
10
33
1
1
6
2
13
11
34
2
1
8
5
16
15
18
2
1
13
6
20
23
45
1
1
22
1
21
19
61
2
1
25
24
27
26
67
2
1
2
5
10
1
2
3
4
5
6
7
8
9
10
11
12
13
14
15
16
17
18
19
20
21
22
23
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31
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37
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41
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43
44
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51
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61
62
63
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76
77
78
79
80
8.4283
-0.2872
0.6661
2.0573
2.6946
-1.5629
0.3166
4.1197
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1.732
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2.9596
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-0.5351
4.9489
4.8561
4.4124
4.0026
6.4322
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6.3411
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0.8136
1.9672
2.8515
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0.3699
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0.1827
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1.6465
2.1451
-2.2573
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2.6516
2.8391
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0.3921
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4.7706
4.3763
5.0548
3.3961
3.5533
4.9777
6.9544
6.6032
-4.1226
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6.475
6.7975
7.0668
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8.8822
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0.6445
0.0123
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0.3603
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1.3472
0.518
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1.5493
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0.2524
0.0425
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1.7012
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0.8086
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1.8086
0.503
1.7731
0.3345
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2.4548
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1.737
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0.0298
0.8977
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1.596
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1.3861
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0.8845
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2.862
2.6604
3.0059
0.975
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0.1257
0.5847
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0.4526
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0.3
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0.8277
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0.1096
1.3735
0.0453
-2.2378
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Conformer
ID
11
2.1
PubChem
ncbi.nlm.nih.gov
2009.12.11
0003644C00000001
Energy
MMFF94 NoEstat
7
1.7.2
Szybki
openeye.com
2012.11.26
90.9091
Feature
Self Overlap
7
2.1
PubChem
ncbi.nlm.nih.gov
2012.11.26
50.849
Fingerprint
Shape
2
2.1
PubChem
ncbi.nlm.nih.gov
2012.11.26
10 15 17894912962691494840
10076449 9 11383835982963215482
10411042 1 17832142720078186058
11135609 187 18410853248584332891
11135926 11 18259699000522354623
11315181 36 17632860837383960579
12082328 90 18409166619981770583
12236239 1 17989208144091680235
12838862 33 18337379509782536968
13533116 47 18342458102240903018
13690498 29 17987786524120535047
13782708 43 13542465341568485693
14117953 113 18261119573829353044
14251764 18 18343302578599469754
14251764 46 18259704502385562184
14856354 85 16343703249310428493
15131766 46 15794290607525213190
15142383 8 17240198846641461188
15183329 4 18060137631200354107
15352257 5 12103842359007724805
15439362 3 17982163732782906712
15461852 350 18202004364841154580
1577012 14 18411976954032003219
15849732 13 18260832609109029677
18681886 176 17917702539820496131
20105231 36 10159704616242060456
20157964 124 18410014308169195138
21150785 3 17490151919498884705
21298829 104 18334577940605644357
21792934 111 18335973174265083016
23559900 14 18339078314701993961
255183 451 17912371927388375470
2838139 119 18261111898427590197
335352 9 18410580587724291966
350125 39 18335420144953151713
3633792 109 18340491071152922336
4073 2 18113343033286644251
4325135 7 18272370863067426989
4760202 170 18340195333234445469
5104073 3 18189347787725460544
54039377 194 17917145131061195975
59755656 215 18334859398264945875
6009941 240 17385730222093131690
6086070 43 17632293527242487011
6328613 192 18411699885675543795
Shape
Multipoles
8
1.8.3
OEShape
openeye.com
2012.11.26
611.52
23.14
2.24
1.21
14.41
0.26
-0.49
-6.8
-4.35
0.18
0.08
1.18
0.2
-0.94
Shape
Self Overlap
7
2.1
PubChem
ncbi.nlm.nih.gov
2012.11.26
1259.421
Shape
Volume
7
1.8.3
OEShape
openeye.com
2012.11.26
351.6
Conformer
RMSD
7
2009.12.11
1
Diverse Conformer
ID List
6
2012.02.08
1
7
8
4
9
6
2
3
5
Charge
MMFF94 Partial
2
1.7.6
OEChem
openeye.com
2012.02.08
9
1 -0.68
12 0.14
15 -0.28
17 -0.29
19 0.14
22 0.28
51 0.15
68 0.4
8 0.14
Count
Effective Rotor
7
1.7.6
OEChem
ncbi.nlm.nih.gov
2012.01.18
8
Features
Pharmacophore
2
ImplicitMillsDean merged
1.8.1
OEShape
openeye.com
2012.02.08
10
1 1 acceptor
1 1 donor
1 23 hydrophobe
1 30 hydrophobe
3 26 28 29 hydrophobe
5 2 3 6 9 11 rings
6 13 20 24 25 26 27 hydrophobe
6 2 3 4 5 7 10 rings
6 4 5 8 12 15 17 rings
6 8 15 16 19 21 22 rings
30
9
9
0
0
0
0
0
1
1