2157664
1
2
3
4
5
6
7
8
9
10
11
12
13
14
15
16
17
18
19
20
21
22
23
24
25
26
27
28
29
30
31
32
33
34
35
36
37
38
39
40
41
42
43
44
45
46
47
48
49
17
16
8
8
8
7
7
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
2
2
2
2
5
6
6
6
7
7
7
8
8
9
9
10
11
12
12
12
13
13
13
14
14
15
15
16
16
17
17
18
20
21
21
22
22
23
23
24
25
25
26
26
27
27
28
28
29
29
30
20
3
4
8
13
19
10
11
12
19
25
41
9
11
10
14
15
31
16
32
33
19
34
35
17
36
18
37
20
21
18
38
39
22
23
40
24
42
24
43
44
26
27
28
45
29
46
30
47
30
48
49
1
2
2
1
1
2
1
1
1
1
1
1
1
2
1
2
2
1
1
1
1
1
1
1
1
1
1
1
1
2
2
1
1
2
1
1
1
1
2
1
1
2
1
1
1
2
1
2
1
1
1
1
2
5
10
1
2
3
4
5
6
7
8
9
10
11
12
13
14
15
16
17
18
19
20
21
22
23
24
25
26
27
28
29
30
31
32
33
34
35
36
37
38
39
40
41
42
43
44
45
46
47
48
49
1.7415
-3.2466
-4.6135
-2.8959
-0.8745
-0.7113
-0.5213
-2.2654
-2.3349
-1.3495
-1.2579
0.3797
-2.7467
-3.1441
-1.1318
1.7131
-2.9379
-1.9466
-1.2805
2.3894
2.2533
3.624
3.4878
4.1731
0.8824
1.4634
1.6455
2.8469
3.0289
3.6296
-0.918
0.2503
0.2786
-3.3421
-3.006
-3.9208
-0.3844
-3.5595
-1.8078
1.7522
-1.0133
4.1707
3.918
5.1364
0.8629
1.2569
3.314
3.64
4.7067
0.2078
-1.2407
-0.8206
-1.7848
-3.7105
1.6908
-1.9327
0.1297
1.0247
1.9947
0.5656
2.4412
-2.4281
1.103
3.0431
1.9335
2.1463
3.1003
-2.7866
0.9288
2.5007
0.4846
2.0562
1.0482
-1.941
-1.0047
-2.8854
-1.013
-2.8936
-1.9574
0.1763
3.4996
2.4084
-3.332
-2.0351
0.3693
3.8088
2.2121
3.9054
3.3003
-1.2178
-0.3002
2.4983
0.7056
-0.2639
-3.6399
-0.2871
-3.6278
-1.9643
-3.2317
-1.0086
-0.7193
-2.3172
-0.5674
-1.0167
0.9249
-0.7434
0.3607
0.1647
-1.5728
-1.6005
0.2263
1.5116
1.0658
-1.1223
2.4215
2.2001
0.1292
-1.8037
0.0261
-1.33
0.4997
-0.1783
1.1046
1.9439
0.438
2.1215
0.6158
1.4575
-2.5204
-1.3438
-2.6908
0.0617
1.2134
1.7057
0.8986
3.3106
2.9172
0.5594
1.4557
-1.8466
1.3935
0.1881
2.4645
-0.2295
2.7806
0.0986
1.5963
Conformer
ID
11
2.1
PubChem
ncbi.nlm.nih.gov
2009.12.11
0020EC6000000001
Energy
MMFF94 NoEstat
7
1.7.2
Szybki
openeye.com
2012.11.26
71.7176
Feature
Self Overlap
7
2.1
PubChem
ncbi.nlm.nih.gov
2012.11.26
45.78
Fingerprint
Shape
2
2.1
PubChem
ncbi.nlm.nih.gov
2012.11.26
10708813 3 18334292097810444428
11578080 2 11489571974626169373
12035759 4 18336265755278400747
12156800 1 17843142323572520038
12422481 6 17391026591727954368
12539773 59 17984672602919273247
12592029 89 17531526607014616839
12596599 1 18196078950829678630
12597179 24 16468939031899333881
12788726 201 18130792282597747009
13122387 1 17900810566420723258
131258 38 15882978486094135042
133893 2 17603875463821886220
1361 2 17038924167569069613
14068700 675 17981286132770311078
14787075 74 17766548428221824268
14955137 171 17761235222979683498
20600515 1 17831298676523911052
20775438 99 15534167291765016102
20905425 154 18260540156512629470
23419403 2 15886492250378189727
238 59 17168421653353363596
2818148 4 18043554766375614514
35225 105 17845942810011537145
392239 28 17911509115201563440
463206 1 18041271162101742296
469060 322 16807872093843343987
513532 50 17485630865488718919
539174 4 18188220813913437984
57527452 28 17607221423977073408
57527585 103 17386300903331097034
6287921 2 18197500614768940586
Shape
Multipoles
8
1.8.3
OEShape
openeye.com
2012.11.26
595.54
6.74
4.47
2.58
0.71
1.39
0.54
0.3
-0.67
-0.21
-1.11
0.07
-0.67
-3.13
Shape
Self Overlap
7
2.1
PubChem
ncbi.nlm.nih.gov
2012.11.26
1287.993
Shape
Volume
7
1.8.3
OEShape
openeye.com
2012.11.26
328.1
Conformer
RMSD
7
2009.12.11
0.8
Diverse Conformer
ID List
6
2012.02.08
1
37
61
289
96
177
278
88
243
84
246
142
262
211
381
390
271
342
259
135
20
60
304
52
209
218
286
276
274
23
312
194
321
350
280
117
341
319
383
201
267
16
384
163
204
349
175
104
2
62
197
58
234
223
245
398
249
120
281
162
113
268
164
212
156
144
372
378
295
178
252
5
221
344
293
273
86
225
153
261
371
393
346
75
217
397
166
360
182
169
244
357
93
90
339
152
77
367
308
103
198
402
287
171
302
74
183
184
141
59
238
148
395
189
388
114
196
125
327
317
7
157
307
47
138
160
168
51
26
369
109
130
108
355
190
216
154
387
251
365
392
292
406
70
57
358
294
310
377
410
347
303
343
44
408
229
340
46
143
136
282
394
235
224
241
95
176
240
239
227
170
147
3
185
14
187
126
334
285
389
92
409
100
181
131
167
316
233
18
379
247
66
65
256
386
83
298
6
296
165
78
318
82
272
362
39
277
375
230
404
356
290
129
299
330
373
364
361
72
351
405
191
338
33
399
101
266
236
385
115
353
407
122
214
311
91
380
53
354
25
264
17
132
265
155
8
151
112
21
315
301
24
283
203
329
322
359
42
231
19
192
89
332
270
71
12
80
85
102
118
38
403
150
237
106
275
324
352
328
31
391
188
258
242
326
396
179
309
45
13
127
128
116
254
370
206
411
139
180
79
10
305
314
366
323
133
32
81
149
105
269
193
28
284
99
279
333
110
27
228
48
401
219
55
248
202
145
29
107
291
260
313
11
137
336
173
257
215
376
73
146
34
54
172
64
306
161
49
134
368
205
186
297
4
111
94
374
124
210
220
140
56
67
159
119
22
413
200
348
40
98
226
345
382
222
253
76
208
207
300
331
199
30
213
174
195
69
337
325
320
35
123
363
288
63
250
97
232
400
68
335
50
15
255
158
121
263
412
9
36
41
87
43
Charge
MMFF94 Partial
2
1.7.6
OEChem
openeye.com
2012.02.08
44
1 -0.18
10 -0.15
11 -0.3
12 0.4
13 0.17
14 -0.15
15 -0.15
16 -0.14
17 -0.15
18 -0.15
19 0.57
2 1.26
20 0.18
21 -0.15
22 -0.15
23 -0.15
24 -0.15
25 0.12
26 -0.15
27 -0.15
28 -0.15
29 -0.15
3 -0.65
30 -0.15
31 0.15
36 0.15
37 0.15
38 0.15
39 0.15
4 -0.65
40 0.15
41 0.37
42 0.15
43 0.15
44 0.15
45 0.15
46 0.15
47 0.15
48 0.15
49 0.15
5 -0.57
6 0.05
7 -0.55
8 -0.06
Count
Effective Rotor
7
1.7.6
OEChem
ncbi.nlm.nih.gov
2012.01.18
7
Features
Pharmacophore
2
ImplicitMillsDean merged
1.8.1
OEShape
openeye.com
2012.02.08
9
1 3 acceptor
1 4 acceptor
1 5 acceptor
1 6 cation
1 7 donor
5 6 8 9 10 11 rings
6 16 20 21 22 23 24 rings
6 25 26 27 28 29 30 rings
6 9 10 14 15 17 18 rings
30
0
0
0
0
0
0
0
1
2