16064039 1 2 3 4 5 6 7 8 9 10 11 12 13 14 15 16 17 18 19 20 21 22 23 24 25 26 27 28 29 30 31 32 33 34 35 36 37 38 39 40 41 42 43 44 45 46 47 48 49 50 51 52 53 54 55 56 57 58 59 60 61 62 63 64 65 66 67 68 69 70 71 72 73 74 75 76 77 78 9 9 9 9 9 9 9 8 8 7 7 7 7 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 6 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 2 3 4 5 6 7 8 8 9 10 10 10 11 11 11 12 12 13 13 13 14 14 14 15 15 16 16 16 17 17 18 18 19 19 19 20 20 21 22 22 23 23 24 25 26 26 26 26 27 27 29 29 30 30 31 31 31 32 32 32 33 33 33 34 34 35 35 36 36 37 37 38 38 38 39 39 40 40 41 41 42 43 44 44 44 45 45 45 15 58 28 14 16 19 18 20 21 21 25 24 28 33 15 18 46 17 47 17 48 49 50 51 52 53 20 54 55 56 57 22 23 59 24 27 25 60 28 29 31 32 30 34 35 36 37 38 61 62 63 64 65 66 67 68 69 41 70 39 71 40 72 43 73 74 75 76 42 45 42 44 43 77 78 1 1 1 1 1 1 1 1 1 2 1 1 1 1 1 1 2 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 1 2 1 1 1 2 1 1 1 1 1 2 1 2 1 1 1 1 1 1 1 1 1 1 1 1 2 1 1 1 2 1 2 1 1 1 1 2 1 1 1 1 1 1 14 10 15 18 46 3 1 15 8 17 14 47 2 1 1 5 255 1 2 3 4 5 6 7 8 9 10 11 12 13 14 15 16 17 18 19 20 21 22 23 24 25 26 27 28 29 30 31 32 33 34 35 36 37 38 39 40 41 42 43 44 45 46 47 48 49 50 51 52 53 54 55 56 57 58 59 60 61 62 63 64 65 66 67 68 69 70 71 72 73 74 75 76 77 78 4.5981 4.5981 3.5981 5.5981 2 2.366 3.366 13.6492 8.0622 12.3923 10.6603 9.7942 7.1962 12.3923 13.3385 13.3385 13.9221 11.5263 11.5263 10.6603 9.7942 8.9282 8.0622 8.0622 8.9282 6.3301 7.1962 7.1962 5.4641 7.1962 6.8301 5.8301 6.3301 6.3301 4.5981 5.4641 6.3301 8.0622 3.732 4.5981 5.4641 3.732 5.4641 4.5981 2.866 12.4823 13.951 13.8759 13.0875 14.383 14.383 11.1278 11.9248 11.9248 11.1278 10.4482 10.0497 14.2559 8.9282 8.9282 6.2932 7.1401 7.3671 6.3671 5.5201 5.2932 6.6401 5.7932 6.0201 6.3301 4.5981 6.001 6.3301 8.3722 8.5991 7.7522 4.9272 3.1951 4.5 -4.5 -3.5 -3.5 0 -1.366 0.366 1.7448 -0.5 4 3 1.5 1 3 2.6953 4.3047 3.5 2.5 4.5 4 2.5 3 2.5 1.5 1 -0.5 3 0 -1 4 -1.366 0.366 1.5 2.5 -0.5 -2 4.5 4.5 -1 -2.5 3 -2 4 -3.5 -0.5 2.1548 2.5991 4.614 4.8716 3.0853 3.9147 2.025 2.025 4.975 4.975 4.5826 3.8923 1.6169 3.62 0.38 -1.676 -1.903 -1.056 0.676 0.903 0.056 2.0369 1.81 0.9631 1.88 0.12 -2.31 5.12 3.9631 4.81 5.0369 2.69 -2.31 8 8 3 6 8 8 8 8 8 8 8 8 8 8 8 8 8 8 8 8 12 12 14 15 21 22 23 24 27 27 29 29 30 34 35 36 37 39 40 41 21 25 46 8 22 23 24 25 30 34 35 36 37 41 39 40 43 42 42 43 0 Compound Canonicalized 5 2011.04.04 1 Compound Complexity 7 E_COMPLEXITY 3.402 Cactvs xemistry.com 2012.05.21 1020 Count Hydrogen Bond Acceptor 5 E_NHACCEPTORS 3.402 Cactvs xemistry.com 2012.05.21 12 Count Hydrogen Bond Donor 5 E_NHDONORS 3.402 Cactvs xemistry.com 2012.05.21 1 Count Rotatable Bond 5 E_NROTBONDS 3.402 Cactvs xemistry.com 2012.05.21 5 Fingerprint SubStructure Keys 16 extended 2 E_SCREEN 3.402 Cactvs xemistry.com 2012.05.21 00000371F07FB1C00000000000000000000000000001600000003C788100000000005801D000001F00000800000E3CE19A1E3FF093081200A8023777740082802931122009D8213874988A7072C09D919460086A8602D8C8271888C08F80000200001000000000040000200000000000000000 IUPAC Name Allowed 1 2.1.0 LexiChem openeye.com 2012.05.21 2-[3,5-bis(trifluoromethyl)phenyl]-N-[4-(4-fluoro-2-methyl-phenyl)-6-[(8S)-8-hydroxy-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]-3-pyridyl]-N,2-dimethyl-propanamide IUPAC Name CAS-like Style 1 2.1.0 LexiChem openeye.com 2012.05.21 2-[3,5-bis(trifluoromethyl)phenyl]-N-[4-(4-fluoro-2-methylphenyl)-6-[(8S)-8-hydroxy-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]-3-pyridinyl]-N,2-dimethylpropanamide IUPAC Name Preferred 1 2.1.0 LexiChem openeye.com 2012.05.21 2-[3,5-bis(trifluoromethyl)phenyl]-N-[4-(4-fluoro-2-methylphenyl)-6-[(8S)-8-hydroxy-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]pyridin-3-yl]-N,2-dimethylpropanamide IUPAC Name Systematic 1 2.1.0 LexiChem openeye.com 2012.05.21 2-[3,5-bis(trifluoromethyl)phenyl]-N-[4-(4-fluoranyl-2-methyl-phenyl)-6-[(8S)-8-oxidanyl-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]pyridin-3-yl]-N,2-dimethyl-propanamide IUPAC Name Traditional 1 2.1.0 LexiChem openeye.com 2012.05.21 2-[3,5-bis(trifluoromethyl)phenyl]-N-[4-(4-fluoro-2-methyl-phenyl)-6-[(8S)-8-hydroxy-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]-3-pyridyl]-N,2-dimethyl-propionamide InChI Standard 1 1.0.4 InChI iupac.org 2012.05.21 InChI=1S/C32H33F7N4O2/c1-18-11-22(33)5-6-23(18)24-15-28(43-10-9-42-8-7-27(44)26(42)17-43)40-16-25(24)41(4)29(45)30(2,3)19-12-20(31(34,35)36)14-21(13-19)32(37,38)39/h5-6,11-16,26-27,44H,7-10,17H2,1-4H3/t26?,27-/m0/s1 InChIKey Standard 1 1.0.4 InChI iupac.org 2012.05.21 FUEBLCGUMDEZGV-GEVKEYJPSA-N Log P XLogP3-AA 7 3.0 sioc-ccbg.ac.cn 2012.05.21 6.4 Mass Exact 7 2.1 PubChem ncbi.nlm.nih.gov 2012.05.21 638.249174 Molecular Formula 1 2.1 PubChem ncbi.nlm.nih.gov 2012.05.21 C32H33F7N4O2 Molecular Weight 7 2.1 PubChem ncbi.nlm.nih.gov 2012.05.21 638.618842 SMILES Canonical 1 1.7.6 OEChem openeye.com 2012.05.21 CC1=C(C=CC(=C1)F)C2=CC(=NC=C2N(C)C(=O)C(C)(C)C3=CC(=CC(=C3)C(F)(F)F)C(F)(F)F)N4CCN5CCC(C5C4)O SMILES Isomeric 1 1.7.6 OEChem openeye.com 2012.05.21 CC1=C(C=CC(=C1)F)C2=CC(=NC=C2N(C)C(=O)C(C)(C)C3=CC(=CC(=C3)C(F)(F)F)C(F)(F)F)N4CCN5CC[C@@H](C5C4)O Topological Polar Surface Area 7 E_TPSA 3.402 Cactvs xemistry.com 2012.05.21 59.9 Weight MonoIsotopic 7 2.1 PubChem ncbi.nlm.nih.gov 2012.05.21 638.249174 45 2 1 1 0 0 0 0 1 1