11157666
1
2
3
4
5
6
7
8
9
10
11
12
13
14
15
16
17
18
19
20
21
22
23
24
25
26
27
28
29
30
31
32
33
34
35
36
37
38
39
40
41
42
43
44
45
46
47
48
49
50
51
52
53
54
55
56
57
58
59
60
61
62
63
64
65
66
67
68
69
70
71
72
9
9
9
9
9
9
9
8
8
7
7
7
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
2
3
4
5
6
7
8
8
9
10
10
10
11
11
11
12
12
13
13
13
14
14
15
15
15
16
16
16
17
17
18
19
19
19
19
20
20
21
21
22
24
24
25
25
25
26
26
26
27
28
28
29
29
30
30
31
31
31
32
32
33
33
34
34
35
36
36
39
39
40
40
40
41
41
37
37
37
38
38
38
42
14
52
23
13
18
51
22
23
31
18
27
14
15
43
16
44
17
45
46
17
47
48
49
50
20
23
24
25
26
21
53
22
28
27
29
30
54
55
56
57
58
59
60
34
36
32
61
33
62
63
64
65
35
38
35
37
39
40
66
41
67
42
68
69
70
71
42
72
1
1
1
1
1
1
1
1
1
2
1
1
1
1
1
1
2
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
2
1
1
1
2
2
1
1
1
1
1
1
1
1
2
1
1
1
2
1
1
1
1
2
1
1
1
1
1
1
2
1
2
1
1
1
1
1
1
13
10
14
15
43
3
1
14
8
13
16
44
3
1
2
5
10
1
2
3
4
5
6
7
8
9
10
11
12
13
14
15
16
17
18
19
20
21
22
23
24
25
26
27
28
29
30
31
32
33
34
35
36
37
38
39
40
41
42
43
44
45
46
47
48
49
50
51
52
53
54
55
56
57
58
59
60
61
62
63
64
65
66
67
68
69
70
71
72
-5.3367
-5.554
-6.833
-2.8659
-5.0157
-3.7233
-2.3875
6.6822
0.6757
5.5167
0.304
4.0238
6.6872
6.973
7.9236
8.4559
8.7049
4.1968
-1.5107
3.1578
1.8572
1.6387
-0.0831
-2.627
-1.6865
-1.5819
2.7458
0.7528
-2.7192
-3.549
-0.5689
-3.7337
-4.5636
0.1824
-4.6559
0.2624
-5.5486
-3.8328
-0.8784
0.6821
-0.7985
-1.3689
6.5475
6.3738
7.6903
8.5344
9.0677
8.69
8.3013
9.7684
5.6167
6.952
3.3539
-0.9871
-2.6998
-1.4958
-2.4368
-1.6913
-0.6821
2.6453
-1.9916
-3.5075
-1.3292
0.0288
-1.0334
-5.4463
0.7037
-1.3329
1.7318
0.5734
0.119
-1.1786
-1.7197
0.4278
-0.9098
1.0761
1.1606
2.4841
4.2366
-1.9304
-2.3666
0.7158
-1.3248
-1.1407
-0.1343
-0.5552
0.6457
-0.2758
0.9518
0.1999
-2.7664
1.1155
0.6239
-0.7491
-2.1356
-1.7139
-3.5197
-3.8575
-1.5814
1.5627
-0.7661
-1.7048
-1.0301
0.1907
-0.7479
2.0553
0.1999
1.9732
-0.7374
1.2044
2.9584
1.6391
2.8765
3.3691
-0.9957
0.019
1.554
0.0025
-1.1219
-0.1018
1.847
1.1157
1.6739
-2.1658
2.1842
-4.3625
-3.9282
-2.8882
-4.5228
-3.5318
-4.4851
-2.6626
-0.7536
-2.4336
-0.3045
-0.6297
-1.9138
0.9465
1.6152
3.355
1.9216
0.5594
2.1216
3.1989
2.6942
2.4818
1.3401
-3.4623
-3.1875
-2.0442
0.8998
-1.0786
-1.3873
0.5947
0.651
0.5841
0.5559
-0.8928
1.0199
-1.1083
-0.2515
0.6096
-0.4542
0.649
0.6634
0.6382
-0.4351
-0.4244
-1.8038
0.641
0.5991
0.7048
-1.4438
0.6221
1.7952
-1.4163
0.6494
-0.469
-0.3697
1.9444
1.7689
-2.5059
-0.4031
-1.8152
2.0101
0.8364
1.2207
-1.6104
1.5849
1.6661
-0.7722
-2.163
-0.7392
-0.0561
0.2732
-1.9827
0.6687
-1.8756
-1.9061
-2.6789
0.4593
1.6709
0.6104
0.5885
-2.2503
1.4232
1.5046
2.6196
2.2044
-0.3481
2.8716
-1.3068
-1.9449
-1.9552
-2.622
2.9749
Conformer
ID
11
2.1
PubChem
ncbi.nlm.nih.gov
2009.12.11
00AA40A200000001
Energy
MMFF94 NoEstat
7
1.7.2
Szybki
openeye.com
2012.11.26
150.315
Feature
Self Overlap
7
2.1
PubChem
ncbi.nlm.nih.gov
2012.11.26
50.746
Fingerprint
Shape
2
2.1
PubChem
ncbi.nlm.nih.gov
2012.11.26
10076449 9 18409736196504961016
10165383 225 18408037412707438767
10190206 1 18412261710632519660
10290309 65 18261950747952881474
11135926 11 18273211989695466382
11513181 2 17773026462774479255
11756154 5 18335144240696789235
12107698 1 16805325522108356861
12156800 1 16762598311585865037
12788726 201 18201423737002796344
13726171 33 17896031040777673829
13911987 19 18339626868257374415
14114207 22 15122967092527172541
14856354 85 18271530887354350351
14930077 153 17749676276929066716
14931854 50 18197753558483801741
14955137 171 18266750249525358451
15183329 4 18202278105088602238
15274700 242 18263640671833746034
15276724 80 18272656714837689574
15328829 1 18040438802737103748
15849732 13 18271253797528959219
16087824 20 18341056225116228497
18603816 31 16272204181167248542
19311894 1 18128811022352355390
19958102 18 18340483362525577950
21792961 116 18259979354095577522
23559900 14 18200301247764515944
2818148 4 17609221500163289839
469060 322 17168436964748211013
5265222 85 18114741642120346934
70634741 139 18408320012886836724
7226269 152 18411694405191811482
9896288 288 17700991954412958465
Shape
Multipoles
8
1.8.3
OEShape
openeye.com
2012.11.26
786.74
17.73
3.91
2.42
38.07
0.61
-1.1
-1.97
-0.15
-3.44
0.09
-4.36
0.7
1.74
Shape
Self Overlap
7
2.1
PubChem
ncbi.nlm.nih.gov
2012.11.26
1708.467
Shape
Volume
7
1.8.3
OEShape
openeye.com
2012.11.26
434.6
Conformer
RMSD
7
2009.12.11
1.2
Diverse Conformer
ID List
6
2012.02.08
1
75
23
59
77
43
11
14
60
73
25
45
56
44
42
53
46
65
39
47
66
72
41
17
80
31
81
67
57
74
10
79
7
48
68
37
19
82
61
15
62
49
40
33
5
64
58
71
18
28
70
34
50
51
52
22
78
35
55
13
63
26
76
12
36
32
54
29
38
69
8
27
20
24
30
6
9
3
21
2
4
16
Charge
MMFF94 Partial
2
1.7.6
OEChem
openeye.com
2012.02.08
45
1 -0.34
10 -0.87
11 -0.48
12 -0.62
13 0.37
14 0.28
18 0.41
19 0.2
2 -0.34
20 -0.15
22 0.12
23 0.57
24 -0.14
27 0.16
29 -0.15
3 -0.34
30 -0.15
31 0.3
32 -0.14
33 -0.14
34 -0.14
35 -0.15
36 -0.15
37 1.16
38 1.16
39 -0.15
4 -0.34
40 0.14
41 -0.15
42 0.19
5 -0.34
51 0.4
52 0.4
53 0.15
6 -0.34
60 0.15
61 0.15
62 0.15
66 0.15
67 0.15
68 0.15
7 -0.19
72 0.15
8 -0.68
9 -0.57
Count
Effective Rotor
7
1.7.6
OEChem
ncbi.nlm.nih.gov
2012.01.18
10
Features
Pharmacophore
2
ImplicitMillsDean merged
1.8.1
OEShape
openeye.com
2012.02.08
10
1 10 donor
1 8 acceptor
1 8 donor
1 9 acceptor
3 10 12 18 cation
3 19 25 26 hydrophobe
5 13 14 15 16 17 rings
6 12 18 20 21 22 27 rings
6 24 29 30 32 33 35 rings
6 28 34 36 39 41 42 rings
42
2
0
2
0
0
0
0
1
2