10133
1
2
3
4
5
6
7
8
9
10
11
12
13
14
15
16
17
18
19
20
21
22
23
24
25
26
27
28
29
30
31
32
33
34
35
36
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41
42
43
44
45
46
47
48
49
50
51
52
53
54
55
56
57
58
59
60
61
62
63
64
65
66
67
68
8
8
8
8
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
6
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
2
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27
14
61
24
65
28
68
28
6
7
15
29
10
12
19
8
14
30
9
13
31
11
18
22
16
20
32
17
21
33
13
34
35
36
37
17
38
16
39
40
41
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43
44
23
45
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47
48
49
25
26
50
24
51
52
53
54
55
24
56
57
58
27
59
60
62
63
64
28
66
67
1
1
1
1
1
1
2
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
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1
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1
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1
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1
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1
1
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1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
1
5
6
15
7
29
2
1
6
5
10
12
19
1
1
7
5
8
14
30
1
1
8
7
9
13
31
1
1
9
8
18
11
22
2
1
10
6
20
16
32
2
1
11
9
21
17
33
2
1
14
1
7
17
38
1
1
20
10
25
26
50
1
1
24
2
21
23
58
1
1
2
5
10
1
2
3
4
5
6
7
8
9
10
11
12
13
14
15
16
17
18
19
20
21
22
23
24
25
26
27
28
29
30
31
32
33
34
35
36
37
38
39
40
41
42
43
44
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46
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52
53
54
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56
57
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64
65
66
67
68
-2.2896
-5.8692
7.4191
6.4579
0.1029
1.0947
-1.2183
-1.8961
-3.2643
2.2896
-4.2036
0.4464
-0.9164
-2.1535
0.9434
2.3454
-3.5316
-3.9948
1.4967
3.6237
-4.7745
-3.0453
-4.5198
-5.4614
4.7126
3.4804
6.0756
6.6501
-0.1462
-0.993
-2.1194
2.0232
-5.074
0.2986
1.0447
-0.7533
-1.3593
-1.7105
0.5585
0.9811
3.0875
2.6046
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-3.353
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0.6346
2.0261
2.1509
3.9353
-3.9969
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-2.5099
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-3.6916
-6.3619
4.8358
4.3955
-1.478
2.9475
2.9867
4.4427
-5.0762
6.7825
6.0434
7.7917
2.2896
-0.907
-1.2919
0.7449
1.0201
-0.1011
0.9436
-0.4362
-0.5935
0.314
0.6035
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-1.6244
2.1264
2.2901
1.8516
1.9716
-1.9254
-0.118
-0.359
0.5021
-0.6179
-1.9962
-0.8348
0.1934
-1.8802
-0.4801
-0.2459
0.9
1.0044
-0.4416
0.1069
0.5656
-1.4951
-2.3056
-1.8001
-2.5434
3.0551
3.098
2.6641
2.1695
2.3264
2.1311
2.7641
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0.792
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0.6457
1.3119
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0.2584
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-2.943
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1.2717
0.0605
2.7008
-2.1739
-2.3012
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-0.0361
-1.5476
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1.1329
2.3628
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0.1893
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0.7057
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0.1895
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0.0892
0.5504
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0.4169
0.7403
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0.7141
1.0006
1.3594
0.5334
1.188
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1.2567
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0.7858
1.754
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1.2757
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0.7184
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1.5033
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1.4967
0.9135
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0.8674
1.4327
0.3819
1.2047
2.4016
1.4721
1.4433
-0.343
0.5437
2.9202
1.8995
1.4167
-1.4884
Conformer
ID
11
2.1
PubChem
ncbi.nlm.nih.gov
2009.12.11
0000279500000001
Energy
MMFF94 NoEstat
7
1.7.2
Szybki
openeye.com
2012.11.26
98.3711
Feature
Self Overlap
7
2.1
PubChem
ncbi.nlm.nih.gov
2012.11.26
61.077
Fingerprint
Shape
2
2.1
PubChem
ncbi.nlm.nih.gov
2012.11.26
10675989 125 16825575996399212613
11089746 13 11095882653218022170
11135609 12 18113905944363332721
12166972 35 17676492774114792876
12236239 1 17748825198893703508
12422481 6 17917714608119298557
12596602 18 17458340827941685736
12633257 1 17489305330380158329
12788726 201 18057880247892638216
13009979 54 18041002847016188125
13140716 1 18196369445095455147
13224815 77 18336262440175454533
13583140 156 18336815425662356797
13782708 43 16733255781987481274
13914758 101 13398638221106775274
14341114 176 18341891917976569768
14787075 74 18186517701025726176
14856354 85 18336831982450540439
14955137 171 18131071554298621256
15183329 4 18411412909019904334
15537594 2 18343297059424511446
15685185 35 17244723492047349196
16110190 28 18271806873199299985
17349148 13 17749107794324115408
17844677 252 17418086625249616992
1813 80 17386005014728457414
18608769 82 18334580182610487946
18927931 339 18409443696257686631
21033648 29 16773213142600101938
21150785 3 15502378945862797010
21267235 1 18410856576830240751
21859007 373 13181923366664697712
22182313 1 18059299746930421109
23081809 10 14908170985123800248
23402539 116 18200861946289631308
23522609 53 18194710204692854544
23559900 14 18129082559138727104
23569914 152 11968107609434555034
23569943 247 17773877494003226286
2838139 119 12247682656075574267
3004659 81 18335698301133426498
335352 9 18411129230730414845
34797466 226 18341904017574448724
350125 39 18409730677045074744
392239 28 18410016572075799035
4015057 19 13695881332409705102
5104073 3 18268419153905685826
59755656 215 18272647914096090622
999808 66 18260836998449795650
Shape
Multipoles
8
1.8.3
OEShape
openeye.com
2012.11.26
552.75
15.16
2.23
1.55
19.34
0.58
-0.21
-4.97
2.83
-1.4
0.16
-1.46
-0.27
0.43
Shape
Self Overlap
7
2.1
PubChem
ncbi.nlm.nih.gov
2012.11.26
1158.271
Shape
Volume
7
1.8.3
OEShape
openeye.com
2012.11.26
310.5
Conformer
RMSD
7
2009.12.11
0.8
Diverse Conformer
ID List
6
2010.05.05
1
5
3
4
2
Charge
MMFF94 Partial
2
1.7.6
OEChem
openeye.com
2012.05.21
11
1 -0.68
14 0.28
2 -0.68
24 0.28
27 0.06
28 0.66
3 -0.65
4 -0.57
61 0.4
65 0.4
68 0.5
Count
Effective Rotor
7
1.7.6
OEChem
ncbi.nlm.nih.gov
2012.01.18
6.2
Features
Pharmacophore
2
ImplicitMillsDean merged
1.8.1
OEShape
openeye.com
2012.05.21
12
1 1 acceptor
1 1 donor
1 2 acceptor
1 2 donor
1 26 hydrophobe
1 3 acceptor
1 4 acceptor
3 3 4 28 anion
5 5 6 10 15 16 rings
6 5 6 7 8 12 13 rings
6 7 8 9 11 14 17 rings
6 9 11 18 21 23 24 rings
28
10
10
0
0
0
0
0
1
1