"AID","Panel Member ID","SID","CID","Activity Outcome","Activity Value [uM]","Activity Type","Assay Name","Target GI","Target Name","Assay Type","PubMed ID","Gene Target if RNAi"
6408,"",103183980,1000,"inconclusive","","","Affinity for 5-hydroxytryptamine receptor was determined using male Dawley rat fundus preparation; Not determined","","","Literature",7069716,""
22830,"",103183980,1000,"unspecified","","","Vmax value was measured","","","Literature",3336016,""
155315,"",103183980,1000,"unspecified","","","Vmax was determined against bovine phenylethanolamine N-Methyltransferase (PNMT)","","","Literature",14695818,""
155338,"",103183980,1000,"unspecified","","","Km ratio for human and bovine Phenylethanolamine N-methyl-transferase",130374,"Phenylethanolamine N-methyltransferase","Literature",11412985,""
156061,"",103183980,1000,"unspecified","","","In vitro enzyme kinetics (PNMT)of the compound expressed as turnover rate isolated from bovine adrenal glands","","","Literature",3336033,""
185803,"",103183980,1000,"unspecified","","","Antiinflammatory activity in rats by using reverse passive Arthus reaction (RPAR) assay at dose level of 50 mg/Kg by peroral administration","","","Literature",6606708,""
230668,"",103183980,1000,"unspecified","","","Ratio of Vmax to Km of compound was determined","","","Literature",3336016,""
231212,"",103183980,1000,"unspecified","","","Activity of the substrate is measured as the ratio of 100*Vmax/Km","","","Literature",3336033,""
231931,"",103183980,1000,"unspecified","","","Ratio expressed as 100x Vmax/Km","","","Literature",3172133,""
232846,"",103183980,1000,"unspecified","","","Vmax/Km x100 value of the compound","","","Literature",7143357,""
232847,"",103183980,1000,"unspecified","","","Vmax/Km x100 value of the compound","","","Literature",7143356,""
155,"",75923,1001,"inactive","","","NCI Yeast Anticancer Drug Screen. Data for the rad50 strain","","","","",""
157,"",75923,1001,"inactive","","","NCI Yeast Anticancer Drug Screen. Data for the mec2-1 strain","","","","",""
161,"",75923,1001,"inactive","","","NCI Yeast Anticancer Drug Screen. Data for the sgs1 mgt1 strain","","","","",""
165,"",75923,1001,"inactive","","","NCI Yeast Anticancer Drug Screen. Data for the cln2 rad14 strain","","","","",""
167,"",75923,1001,"inactive","","","NCI Yeast Anticancer Drug Screen. Data for the bub3 strain","","","","",""
175,"",75923,1001,"inactive","","","NCI Yeast Anticancer Drug Screen. Data for the mlh1 rad18 strain","","","","",""
316,"",75923,1001,"inactive","","","NCI In Vivo Anticancer Drug Screen. Data for tumor model  P1534 Leukemia (intraperitoneal) in CD2F1 (CDF1) mice","","","","",""
330,"",75923,1001,"inactive","","","NCI In Vivo Anticancer Drug Screen. Data for tumor model  P388 Leukemia (intraperitoneal) in CD2F1 (CDF1) mice","","","","",""
342,"",75923,1001,"inactive","","","NCI In Vivo Anticancer Drug Screen. Data for tumor model  Sarcoma 180 (subcutaneous) in Swiss mice","","","","",""
880,"",26756723,1001,"inactive","","","qHTS Assay for Inhibitors of RGS12 GoLoco Motif Activity (Red Fluorophore)",3290016,"RGS12 [Homo sapiens]","confirmatory","",""
1030,"",26756723,1001,"inactive","","Potency","qHTS Assay for Inhibitors of Aldehyde Dehydrogenase 1 (ALDH1A1)",30582681,"aldehyde dehydrogenase 1 family, member A1 [Homo sapiens]","confirmatory","",""
1376,"",47193684,1001,"inactive","","IC50","Inhibitors of Mycobacterial Glucosamine-1-phosphate acetyl transferase (GlmU)",15608158,"UDP-N-acetylglucosamine pyrophosphorylase glmU [Mycobacterium tuberculosis H37Rv]","confirmatory","",""
1385,"",47193684,1001,"inactive","","","Homologous recombination - Rad 51",49168602,"RAD51 [Homo sapiens]","screening","",""
1422,"",47193684,1001,"inactive","","","Inhibitors of the EP2 Prostaglandin E2 Receptor - Primary Screen",31881630,"prostaglandin E receptor 2 (subtype EP2), 53kDa [Homo sapiens]","screening","",""
1457,"",26756723,1001,"inactive","","Potency","qHTS Assay for Identifying the Cell-Membrane Permeable IMPase Inhibitors: Potentiation with Lithium",44888968,"Inositol monophosphatase","confirmatory","",""
1458,"",26756723,1001,"inactive",14.1254,"Potency","qHTS Assay for Enhancers of SMN2 Splice Variant Expression",10937869,"survival motor neuron protein isoform d [Homo sapiens]","confirmatory","",""
1460,"",26756723,1001,"inactive","","Potency","qHTS for Inhibitors of Tau Fibril Formation, Thioflavin T Binding",92096784,"Microtubule-associated protein tau [Homo sapiens]","confirmatory","",""
1463,"",26756723,1001,"inactive","","Potency","Counterscreen qHTS for Inhibitors of Tau Fibril Formation, Fluorescence Polarization","","","confirmatory","",""
1465,"",47193684,1001,"inactive","","EC50","Screen for small molecule probes relevant to Friedreich's ataxia, Single Dose and Dose Response","","","confirmatory","",""
1468,"",26756723,1001,"inactive","","Potency","qHTS for Inhibitors of Tau Fibril Formation, Fluorescence Polarization",92096784,"Microtubule-associated protein tau [Homo sapiens]","confirmatory","",""
1469,"",26756723,1001,"inactive","","Potency","qHTS for Inhibitors of the Interaction of Thyroid Hormone Receptor and Steroid Receptor Coregulator 2",189491771,"thyroid hormone receptor beta [Homo sapiens]","confirmatory","",""
1471,"",26756723,1001,"inactive","","","qHTS Multiplex Assay to Identify Dual Action Probes in a Cell Model of Huntington: Cytoprotection (ATP)",90903231,"huntingtin [Homo sapiens]","confirmatory","",""
1477,"",26756723,1001,"inactive","","Potency","qHTS Assay for Compounds Blocking the Interaction Between CBF-beta and RUNX1 for the Treatment of Acute Myeloid Leukemia","","","confirmatory","",""
1479,"",26756723,1001,"inactive","","Potency","Total Fluorescence Counterscreen for Inhibitors of the Interaction of Thyroid Hormone Receptor and Steroid Receptor Coregulator 2",189491771,"thyroid hormone receptor beta [Homo sapiens]","confirmatory","",""
1490,"",26756723,1001,"inactive","","Potency","qHTS Assay for Inhibitors of Bacillus subtilis Sfp phosphopantetheinyl transferase (PPTase)",10954339,"phosphopantetheinyl transferase [Bacillus subtilis]","confirmatory","",""
1511,"",49718670,1001,"inactive","","","Primary cell-based high-throughput screening assay for identification of compounds that protect hERG from block by proarrhythmic agents",487738,"putative potassium channel subunit [Homo sapiens]","screening","",""
1529,"",47193684,1001,"inactive","","","Multiplex HTS Assay for Inhibitors of MEK Kinase PB1 Domains, specifically MEK5 MEK Kinase3 Wildtype",42794767,"mitogen-activated protein kinase kinase kinase 3 isoform 1 [Homo sapiens]","screening","",""
1530,"",47193684,1001,"inactive","","","Multiplex HTS Assay for Inhibitors of MEK Kinase PB1 Domains, specifically MEK5 MEK Kinase 2 mutant",22035600,"mitogen-activated protein kinase kinase kinase kinase 2 [Homo sapiens]","screening","",""
1531,"",47193684,1001,"inactive","","","Multiplex HTS Assay for Inhibitors of MEK Kinase PB1 Domains, specifically MEK5 binding to MEK Kinase 2 Wildtype",22035600,"mitogen-activated protein kinase kinase kinase kinase 2 [Homo sapiens]","screening","",""
1532,"",47193684,1001,"inactive","","","Rml C and D inhibition 384-well mixture HTS","","","screening","",""
1554,"",49718670,1001,"inactive","","","MLPCN Ras selective lethality-BJeLR viability","","","screening","",""
1621,"",47193684,1001,"inactive","","IC50","A Cell Based Assay for the Identification of Lead Compounds with Anti-Viral Activity Against West Nile Virus","","","confirmatory","",""
1626,"",47193684,1001,"inactive","","IC50","High Throughput Screen to Identify Inhibitors of Mycobacterium tuberculosis H37Rv","","","confirmatory","",""
1662,"",49718670,1001,"inactive","","","MLPCN Streptokinase Expression Inhibition",15675770,"streptokinase A precursor [Streptococcus pyogenes M1 GAS]","screening","",""
1663,"",49718670,1001,"inactive","","","MLPCN Platelet Activation -Dense Granule Release","","","screening","",""
1672,"",49718670,1001,"inactive","","","Primary cell-based high-throughput screening assay for identification of compounds that inhibit/block inward-rectifying potassium ion channel Kir2.1",6680530,"inward rectifier potassium channel 2 [Mus musculus]","screening","",""
1811,"",46393246,1001,"active","","","Experimentally measured binding affinity data derived from PDB",157833979,"Chain A, Prediction Of Novel Serine Protease Inhibitors","other",7634078,""
1811,"",46393335,1001,"active","","","Experimentally measured binding affinity data derived from PDB",42543835,"Chain A, Trypsin Specificity As Elucidated By Lie Calculations, X-Ray Structures And Association Con","other",18093984,""
1811,"",46393337,1001,"active","","","Experimentally measured binding affinity data derived from PDB",42543837,"Chain A, Trypsin Specificity As Elucidated By Lie Calculations, X-ray Structures And Association Con","other",18093984,""
1813,"",49718670,1001,"inactive","","","MLPCN Alpha-Synuclein 5'UTR - 5'-UTR binding - inhibitors","","","screening","",""
1814,"",49718670,1001,"inactive","","","MLPCN Alpha-Synuclein 5'UTR - 5'-UTR binding - activators","","","screening","",""
1832,"",49718670,1001,"inactive","","","MLPCN maternal gene expression-MEX-5 TCR-2 binding assay-Primary Screen",55976631,"Zinc finger protein mex-","screening","",""
1850,"",49718670,1001,"inactive","","IC50","A small molecule screen for inhibitors of the PhoP regulon in Salmonella typhi","","","confirmatory","",""
1863,"",49718670,1001,"inactive","","IC50","A small molecule screen for inhibitors of the PhoP regulon in Salmonella Typhimurium","","","confirmatory","",""
1865,"",26756723,1001,"inactive","","Potency","Quantitative High-Throughput Screen for Regulators of Epigenetic Control","","","confirmatory","",""
1875,"",49718670,1001,"inactive","","","Luminescence Cell-Based Primary HTS to Identify Inhibitors of Polyadenylation","","","screening","",""
1885,"",49718670,1001,"inactive","","","Luminescence Cell-Based/Microorganism Primary HTS to Identify Inhibitors of T.Cruzi Replication","","","screening","",""
1899,"",49718670,1001,"inactive","","","TR-FRET-based primary biochemical high-throughput screening assay to identify inhibitors of Hepatitis C Virus (HCV) core protein dimerization",83779224,"core protein [Hepatitis C virus]","screening","",""
1903,"",49718670,1001,"inactive","","IC50","Identification of SV40 T antigen inhibitors: A route to novel anti-viral reagents",297591903,"large T antigen [Simian virus 40]","confirmatory","",""
1906,"",49718670,1001,"inactive","","","QFRET-based counterscreen for PFM18AAP inhibitors: biochemical high throughput screening assay to identify inhibitors of the Cathepsin L proteinase (CTSL1).",55958172,"cathepsin L1 [Homo sapiens]","screening","",""
1910,"",49718670,1001,"inactive","","","Luminescence Cell-Based Primary HTS to Identify Transcriptional Activators of Hypoxia-Inducible Factor Pathway","","","screening","",""
1947,"",49718670,1001,"inactive","","","Fluorescence polarization-based counterscreen for RBBP9 inhibitors: primary biochemical high throughput screening assay to identify inhibitors of the serine hydrolase family member Fam108B.",21595511,"Fam108b protein [Mus musculus]","screening","",""
1950,"",49718670,1001,"inactive","","","Fluorescence polarization-based primary biochemical high throughput screening assay to identify inhibitors of the Epstein-Barr virus nuclear antigen 1 (EBNA-1).",23893623,"EBNA-1 protein [Human herpesvirus 4]","screening","",""
1956,"",47193684,1001,"inactive","","Conc @ Max Fold Increase","A high-throughput screen to identify small molecule compounds that augment HSV replication","","","confirmatory","",""
1962,"",49718670,1001,"inactive","","","Fluorescence polarization-based primary biochemical high throughput screening assay to identify inhibitors of tRNA 2'-phosphotransferase (TPT1).",68476498,"likely tRNA 2'-phosphotransferase [Candida albicans SC5314]","screening","",""
1974,"",49718670,1001,"inactive","","","Fluorescence polarization-based counterscreen for RBBP9 inhibitors: primary biochemical high throughput screening assay to identify inhibitors of the oxidoreductase glutathione S-transferase omega 1(GSTO1).",4758484,"glutathione S-transferase omega-1 isoform 1 [Homo sapiens]","screening","",""
1979,"",49718670,1001,"inactive","","","Fluorescence Cell-Based Primary HTS of C.albicans growth in the presence of Fluconazole and compound",994798,"heat shock protein 90 [Candida albicans]","screening","",""
1987,"",49718670,1001,"inactive","","","Fluorescence-based primary biochemical high throughput screening assay to identify inhibitors of Protein Phosphatase 5 (PP5).",37589898,"PPP5C protein [Homo sapiens]","screening","",""
2016,"",49718670,1001,"inactive","","","Multiplex HTS Screen of TOR pathway GFP-fusion proteins in Saccharomyes cerevisiae_specifically_ MEP2_MLPCN.",1302091,"MEP2 [Saccharomyces cerevisiae]","screening","",""
2023,"",49718670,1001,"inactive","","","Multiplex HTS Screen of TOR pathway GFP-fusion proteins in Saccharomyes cerevisiae_specifically_ LAP4_MLPCN.",486173,"LAP4 [Saccharomyces cerevisiae]","screening","",""
2025,"",49718670,1001,"inactive","","","Multiplex HTS Screen of TOR pathway GFP-fusion proteins in Saccharomyes cerevisiae_specifically_ RPL19A_MLPCN.",536029,"RPL19A [Saccharomyces cerevisiae]","screening","",""
2029,"",49718670,1001,"inactive","","","Multiplex HTS Screen of TOR pathway GFP-fusion proteins in Saccharomyes cerevisiae_specifically_ CIT2_MLPCN.",171229,"citrate synthase 2 [Saccharomyces cerevisiae]","screening","",""
2052,"",49718670,1001,"inactive","","","HTS for developing T Cell Immune Modulators",124486680,"integrin alpha-L [Mus musculus]","screening","",""
2057,"",49718670,1001,"inactive","","","Fluorescence polarization-based primary biochemical high throughput screening assay to identify inhibitors of myeloid cell leukemia sequence 1 (MCL1) interactions with BIM-BH3 peptide.",78070770,"Myeloid cell leukemia sequence 1 (BCL2-related) [Homo sapiens]","screening","",""
2066,"",49718670,1001,"inactive","","","Multiplex HTS Screen of TOR pathway GFP-fusion proteins in Saccharomyes cerevisiae_specifically_ AGP1_MLPCN.",85666113,"Agp1p [Saccharomyces cerevisiae S288c]","screening","",""
2094,"",49718670,1001,"inactive","","","Plate Read Microorganism-Based Primary HTS to Identify Modulators of the AI-2 Quorum Sensing System",67463988,"Chain A, Crystal Structure Of The Apo Form Of Vibrio Harveyi Luxp Complexed With The Periplasmic Dom","screening","",""
2097,"",49718670,1001,"inactive","","","Cell-Free Homogeneous Primary HTS to Identify Inhibitors of GSK3beta Activity",21361340,"GSK3B gene product [Homo sapiens]","screening","",""
2098,"",49718670,1001,"inactive","","","Luminescence Cell-Based Primary HTS to Identify Inhibitors of Heat Shock Factor 1 (HSF1).",62740231,"Hsf1 protein [Mus musculus]","screening","",""
2099,"",49718670,1001,"inactive","","","Fluorescence Biochemical Primary HTS to Identify Inhibitors of GASC-1 Activity","","","screening","",""
2101,"",26756723,1001,"inactive","","Potency","qHTS Assay for Inhibitors and Activators of N370S glucocerebrosidase as a Potential Chaperone Treatment of Gaucher Disease",496369,"glucocerebrosidase [Homo sapiens]","confirmatory","",""
2107,"",26756723,1001,"inactive","","Potency","qHTS Assay for Inhibitors and Activators of Human alpha-Galactosidase From Spleen Homogenate",757912,"alpha-galactosidase [Homo sapiens]","confirmatory","",""
2112,"",26756723,1001,"inactive","","Potency","qHTS Assay for Inhibitors and Activators of Human alpha-Glucosidase From Spleen Homogenate",119393891,"lysosomal alpha-glucosidase preproprotein [Homo sapiens]","confirmatory","",""
2129,"",49718670,1001,"inactive","","","Primary biochemical high throughput screening assay to identify inhibitors of BCL2-related protein, long isoform (BCLXL).",510901,"bcl-xL [Homo sapiens]","screening","",""
2130,"",49718670,1001,"inactive","","","Fluorescence polarization-based primary biochemical high throughput screening assay to identify inhibitors of Protein Phosphatase Methylesterase 1 (PME-1).",7706645,"protein phosphatase methylesterase 1 [Homo sapiens]","screening","",""
2156,"",49718670,1001,"inactive","","","Primary cell-based high-throughput screening assay for identification of compounds that inhibit KCNQ2 potassium channels",18959272,"Kcnq2 gene product [Rattus norvegicus]","screening","",""
2174,"",49718670,1001,"inactive","","","Counterscreen for PME1 inhibitors: fluorescence polarization-based primary biochemical high throughput screening assay to identify inhibitors of lysophospholipase 1 (LYPLA1).",5453722,"acyl-protein thioesterase 1 [Homo sapiens]","screening","",""
2177,"",49718670,1001,"inactive","","","Counterscreen for PME1 inhibitors: fluorescence polarization-based primary biochemical high throughput screening assay to identify inhibitors of lysophospholipase 2 (LYPLA2).",4581413,"lysophospholipase II [Homo sapiens]","screening","",""
2216,"",49718670,1001,"inactive","","","Fluorescence Cell-Free Homogeneous Primary HTS to Identify Inhibitors of the RanGTP-Importin-beta complex","","","screening","",""
2221,"",49718670,1001,"inactive","","","Fluorescence Cell-Free Homogenous Primary HTS to Identify Inhibitors of RecA Intein Splicing Activity",15609874,"DNA recombination protein RecA [Mycobacterium tuberculosis H37Rv]","screening","",""
2227,"",49718670,1001,"inactive","","","Primary cell-based high-throughput screening assay for identification of compounds that allosterically potentiate transient receptor potential cation channel C4 (TRPC4)",2935630,"alternatively spliced Trp4 [Mus musculus]","screening","",""
2234,"",49718670,1001,"inactive","","","Counterscreen for inhibitors of EBNA-1: fluorescence polarization-based biochemical high throughput primary assay to identify inhibitors of the Epstein-Barr virus-encoded protein, ZTA.",82503229,"BZLF1 [Human herpesvirus 4]","screening","",""
2235,"",49718670,1001,"inactive","","","Counterscreen for inhibitors of PP5: fluorescence-based biochemical high throughput primary assay to identify inhibitors of Protein Phosphatase 1 (PP1).",56790945,"PPP1CA gene product [Homo sapiens]","screening","",""
2237,"",49718670,1001,"inactive","","","Primary cell-based screen for identification of compounds that activate transient receptor potential cation channel C4 (TRPC4).",2935630,"alternatively spliced Trp4 [Mus musculus]","screening","",""
2239,"",49718670,1001,"inactive","","","Primary cell-based high-throughput screening assay for identification of compounds that potentiate KCNQ2 potassium channels",18959272,"Kcnq2 gene product [Rattus norvegicus]","screening","",""
2247,"",49718670,1001,"inactive","","","Primary cell-based screen for identification of compounds that inhibit transient receptor potential cation channel C4 (TRPC4).",2935630,"alternatively spliced Trp4 [Mus musculus]","screening","",""
2280,"",49718670,1001,"inactive","","","Fluorescence polarization-based primary biochemical high throughput screening assay to identify inhibitors of GLD-1 protein - TGE RNA interaction.",17507875,"defective in Germ Line Development family member (gld-1) [Caenorhabditis elegans]","screening","",""
2300,"",49718670,1001,"inactive","","","TR-FRET-based primary biochemical high throughput screening assay to identify agonists of nuclear receptor subfamily 2, group E, member 3 (NR2E3).",216409728,"photoreceptor-specific nuclear receptor [Homo sapiens]","screening","",""
2380,"",49718670,1001,"inactive","","","uHTS identification of small molecules that induce b-cell replication in the MIN-6 cell line","","","screening","",""
2391,"",49718670,1001,"inactive","","IC50","A Cell Based HTS Approach for the Discovery of New Inhibitors of Respiratory syncytial virus (RSV)","","","confirmatory","",""
2435,"",49718670,1001,"inactive","","","Fluorescence-based primary cell-based high throughput screening assay to identify agonists of the Oxytocin Receptor (OXTR).",32307152,"oxytocin receptor [Homo sapiens]","screening","",""
2445,"",49718670,1001,"inactive","","","Fluorescence-based primary cell-based high throughput screening assay to identify potentiators of Oxytocin Receptor (OXTR)",32307152,"oxytocin receptor [Homo sapiens]","screening","",""
2462,"",49718670,1001,"inactive","","","Luminescence Cell-Based Primary HTS to Identify Inhibitors of A1 Apoptosis.",20336315,"bcl-2-like protein 11 isoform 1 [Homo sapiens]","screening","",""
2517,"",26756723,1001,"inactive","","Potency","qHTS Assay for Inhibitors of the Human Apurinic/apyrimidinic Endonuclease 1 (APE1)",6980812,"Chain A, Human Ape1 Endonuclease With Bound Abasic Dna And Mn2+ Ion","confirmatory","",""
2520,"",49718670,1001,"inactive","","","uHTS identification of small molecule agonists of the APJ  receptor  via a luminescent beta-arrestin assay",4885057,"APLNR gene product [Homo sapiens]","screening","",""
2521,"",49718670,1001,"inactive","","","uHTS identification of small molecule antagonists of the APJ  receptor  via a luminescent beta-arrestin assay",4885057,"APLNR gene product [Homo sapiens]","screening","",""
2524,"",49718670,1001,"inactive","","","uHTS Luminescent assay for identification of activators of human intestinal alkaline phosphatase",124376142,"Alkaline phosphatase, intestinal [Homo sapiens]","screening","",""
2540,"",49718670,1001,"inactive","","","HTS Luminescent assay for identification of inhibitors of Sentrin-specific protease 8 (SENP8)",262118306,"SENP8 gene product [Homo sapiens]","screening","",""
2544,"",49718670,1001,"inactive","","","uHTS Luminescent assay for identification of inhibitors of human intestinal alkaline phosphatase",124376142,"Alkaline phosphatase, intestinal [Homo sapiens]","screening","",""
2549,"",26756723,1001,"inactive","","Potency","qHTS Assay for Inhibitors of RecQ-Like Dna Helicase 1 (RECQ1)",282403581,"Chain A, Structure Of Human Recq-Like Helicase In Complex With A Dna Substrate","confirmatory","",""
2550,"",49718670,1001,"inactive","","","High throughput screening of activators of transient receptor potential cation channel C6 (TRPC6)",160333370,"short transient receptor potential channel 6 [Mus musculus]","screening","",""
2553,"",49718670,1001,"inactive","","","High throughput screening of inhibitors of transient receptor potential cation channel C6 (TRPC6)",160333370,"short transient receptor potential channel 6 [Mus musculus]","screening","",""
2557,"",49718670,1001,"inactive","","","HTS for Identification of VLA-4 Allosteric Modulators from MLPCN library",67191027,"integrin alpha-4 precursor [Homo sapiens]","screening","",""
2563,"",49718670,1001,"inactive","","","Fluorescence Cell-Free Homogenous Primary HTS  to Identify Inhibitors of the Ras-converting Enzyme",6323930,"Rce1p [Saccharomyces cerevisiae S288c]","screening","",""
2599,"",49718670,1001,"inactive","","","uHTS Luminescent assay for identification of inhibitors of Sentrin-specific protease 6 (SENP6)",6166485,"SUMO-1-specific protease [Homo sapiens]","screening","",""
2606,"",49718670,1001,"inactive","","","Fluorescence polarization-based primary biochemical high throughput screening assay to identify inhibitors of the membrane-associated serine protease Rv3671c in M.tuberculosis",15610807,"membrane-associated serine protease [Mycobacterium tuberculosis H37Rv]","screening","",""
2629,"",49718670,1001,"inactive","","","Fluorescence Polarization Cell-Free Homogeneous Primary HTS to Identify Inhibitors of the LANA Histone H2A/H2B Interaction",139472804,"LANA [Human herpesvirus 8]","screening","",""
2642,"",49718670,1001,"inactive","","","Primary cell-based high-throughput screening assay for identification of compounds that inhibit KCNQ1 potassium channels",32479527,"KCNQ1 gene product [Homo sapiens]","screening","",""
2648,"",49718670,1001,"inactive","","","Primary cell-based high-throughput screening assay for identification of compounds that potentiate/activate KCNQ1 potassium channels",32479527,"KCNQ1 gene product [Homo sapiens]","screening","",""
2650,"",49718670,1001,"inactive","","","Luminescence Cell-Free  Homogenous Primary HTS to Identify Inhibitors of GSK-3 alpha",49574532,"GSK3A gene product [Homo sapiens]","screening","",""
2661,"",49718670,1001,"inactive","","","Luminescence Cell-Free  Homogenous Primary HTS to Identify Inhibitors of Serine/Threonine  Kinase 33  Activity",23943882,"serine/threonine-protein kinase 33 [Homo sapiens]","screening","",""
2690,"",49718670,1001,"inactive","","","A yeast HTS for caloric restriction mimetics that inhibit age-related superoxide","","","screening","",""
2716,"",49718670,1001,"inactive","","","Luminescence  Microorganism Primary HTS to Identify Inhibitors of the SUMOylation Pathway Using a Temperature Sensitive Growth Reversal Mutant Mot1-301","","","screening","",""
2717,"",49718670,1001,"inactive","","","Luminescence Cell-Based Primary HTS to Identify Inhibitors of Cancer Stem Cells","","","screening","",""
2718,"",49718670,1001,"inactive","","","Fluorescence Cell-Free Homogeneous Primary HTS to Identify Inhibitors of Histone Deacetylase 3",13128862,"histone deacetylase 3 [Homo sapiens]","screening","",""
2751,"",49718670,1001,"inactive","","","Fluorescence polarization-based primary biochemical high throughput screening assay to identify inhibitors of the prolyl oligopeptidase-like enzyme (PREPL)",153217451,"Prolyl endopeptidase-like [Homo sapiens]","screening","",""
2796,"",49718670,1001,"inactive","","","Luminescence-based primary cell-based high throughput screening assay to identify activators of the Aryl Hydrocarbon Receptor (AHR)",4502003,"aryl hydrocarbon receptor precursor [Homo sapiens]","screening","",""
2797,"",49718670,1001,"inactive","","","Counterscreen for Oxytocin Receptor (OXTR) agonists: Fluorescence-based primary cell-based high throughput assay to identify agonists of the vasopressin 1 receptor (V1R)",4502331,"vasopressin V1a receptor [Homo sapiens]","screening","",""
2805,"",49718670,1001,"inactive","","","uHTS Luminescent assay for identification of activators of mouse intestinal alkaline phosphatase",124487323,"intestinal alkaline phosphatase precursor [Mus musculus]","screening","",""
2806,"",49718670,1001,"inactive","","","uHTS Luminescent assay for identification of inhibitors of mouse intestinal alkaline phosphatase",124487323,"intestinal alkaline phosphatase precursor [Mus musculus]","screening","",""
2825,"",49718670,1001,"inactive","","","uHTS Luminescent assay for identification of inhibitors of NALP3 in yeast",219518789,"NLRP3 protein [Homo sapiens]","screening","",""
5354,"",103185023,1001,"active",16.8,"Ki","Binding affinity was performed using [3H]ketanserin as the radioligand and stably transfected NIH3T3 cells expressing the 5-hydroxytryptamine 2A receptor (GF-62 cells).","","","Literature",11931619,""
5516,"",103185023,1001,"active",16.82,"Ki","Binding affinity against 5-hydroxytryptamine 2A receptor expressed NIH3T3 cells using [3H]ketanserin",112808,"5-hydroxytryptamine receptor 2A","Literature",11229772,""
6406,"",103185023,1001,"active",5.49541,"Kd","Affinity against 5-hydroxytryptamine receptors in rat fundus model","","","Literature",7365744,""
6407,"",103185023,1001,"active",5.49541,"Kd","Affinity for 5-hydroxytryptamine receptor was determined using male Dawley rat fundus preparation","","","Literature",7069716,""
18736,"",103185023,1001,"unspecified","","","Selectivity of guest-induced changes in membrane potential at pH 5.0 for PVC matrix liquid membrane without any host","","","Literature",10476872,""
18737,"",103185023,1001,"unspecified","","","Selectivity of guest-induced changes in membrane potential at pH 5.0 for PVC matrix liquid membranes incorporated with o-Tolyloxy-acetic acid decyl ester polymer","","","Literature",10476872,""
18738,"",103185023,1001,"unspecified","","","Selectivity of guest-induced changes in membrane potential at pH 5.0 for PVC matrix liquid membranes incorporated with o-Tolyloxy-acetic acid ethyl ester polymer","","","Literature",10476872,""
18739,"",103185023,1001,"unspecified","","","Selectivity of guest-induced changes in membrane potential at pH 5.0 for PVC matrix liquid membranes incorporated with (2-Butoxy-5-tert-butyl-3-methyl-phenyl)-methanol polymer","","","Literature",10476872,""
18740,"",103185023,1001,"unspecified","","","Selectivity of guest-induced changes in membrane potential at pH 5.0 for PVC matrix liquid membranes incorporated with 6,7,9,10,17,18,20,21-Octahydro-5,8,11,16,19,22-hexaoxa-dibenzo[a,j]cyclooctadecene","","","Literature",10476872,""
23236,"",103185023,1001,"unspecified","","","Partition coefficient (logP)","","","Literature",10476872,""
25080,"",103185023,1001,"unspecified","","","pKA value in aqueous solution","","","","",""
61992,"",103185023,1001,"unspecified","","","Compound was evaluated as substrate for Dopamine beta hydroxylase (DBH) from bovine adrenals and the enzymatic kinetic constant was reported as Kcat","","","Literature",6481771,""
62142,"",103185023,1001,"unspecified",7000,"Km","Compound was evaluated as substrate for Dopamine beta hydroxylase (DBH) from bovine adrenals and the enzymatic kinetic constant was reported as Km","","","Literature",6481771,""
125213,"",103185023,1001,"unspecified","","","Compound was evaluated as substrate for monoamine oxidase (MAO) from bovine erythrocyte and the enzymatic kinetic constant was reported as Kcat","","","Literature",6481771,""
125217,"",103185023,1001,"unspecified",2200,"Km","Compound was evaluated as substrate for monoamine oxidase (MAO) from bovine erythrocyte and the enzymatic kinetic constant was reported as Km","","","Literature",6481771,""
145543,"",103185023,1001,"unspecified",467,"Ki","Inhibitory activity against Norepinephrine N-methyl-transferase of bovine adrenal glands","","","Literature",7143356,""
155169,"",103185023,1001,"unspecified",854,"Ki","In vitro inhibitory activity against bovine phenylethanolamine N-methyl-transferase","","","Literature",2913308,""
214878,"",103185023,1001,"active",11,"Ki","Binding affinity against bovine trypsin","","","Literature",12036355,""
215916,"",103185023,1001,"unspecified","","","Binding affinity against trypsin","","","Literature",12061879,""
226029,"",103185023,1001,"unspecified","","","Tested for the multidrug resistance reversal activity against P388 murine leukemia cell line, activity is expressed as RF(ED50 with no adriamycin (ADR)/ED50 with 200 nM ADR)","","","Literature",11087578,""
227718,"",103185023,1001,"unspecified","","","Binding energy by using the equation deltaG obsd = -RT ln KD","","","Literature",6094812,""
231141,"",103185023,1001,"unspecified","","","Ratio of the kinetic parameter Kcat to the Km on substrate dopamine beta-hydrolase from bovine adrenals","","","Literature",6481771,""
231142,"",103185023,1001,"unspecified","","","Ratio of the kinetic parameter Kcat to the Km on substrate dopamine monoamine oxidase","","","Literature",6481771,""
241172,"",103185023,1001,"active",4.41,"IC50","Inhibitory concentration against human cytochrome P450 2A6",308153612,"Cytochrome P450 2A6","Literature",15658857,""
241174,"",103185023,1001,"active",3,"IC50","Inhibitory concentration against mouse cytochrome P450 2A5","","","Literature",15658857,""
273097,"",103185023,1001,"unspecified","","","Activity of human SSAO measured as hydrogen peroxide production at 1 mM relative to benzylamine oxidation",2501336,"Membrane primary amine oxidase","Literature",17034126,""
273098,"",103185023,1001,"unspecified","","","Activity of mouse SSAO measured as hydrogen peroxide production at 100 uM relative to benzylamine oxidation",5902787,"Membrane primary amine oxidase","Literature",17034126,""
273099,"",103185023,1001,"unspecified",3725,"Km","Binding affinity to human SSAO",2501336,"Membrane primary amine oxidase","Literature",17034126,""
273100,"",103185023,1001,"active",34.8,"Km","Binding affinity to mouse SSAO",5902787,"Membrane primary amine oxidase","Literature",17034126,""
313558,"",103185023,1001,"unspecified",220,"Ki","Inhibition of bovine PNMT by radiochemical assay",130374,"Phenylethanolamine N-methyltransferase","Literature",18024134,""
313559,"",103185023,1001,"active",4,"Ki","Displacement of [3H]clonidine from adrenergic alpha-1 receptor in Sprague-Dawley rat cortex","","","Literature",18024134,""
313560,"",103185023,1001,"unspecified","","","Selectivity of Ki for bovine PNMT over Ki for rat alpha-2 adrenoceptor","","","Literature",18024134,""
341210,"",103185023,1001,"active",0.129,"EC50","Agonist activity at human trace amine associated receptor 1 expressed in RD-HGA16 CHO-K1 cells coexpressed with Galpha16 protein assessed as internal calcium mobilization by calcium 3 assay",38258636,"Trace amine-associated receptor 1","Literature",18602830,""
341211,"",103185023,1001,"unspecified","","","Agonist activity at human trace amine associated receptor 1 expressed in RD-HGA16 CHO-K1 cells coexpressed with Galpha16 protein assessed as internal calcium mobilization by calcium 3 assay relative to 2-phenylethanamine",38258636,"Trace amine-associated receptor 1","Literature",18602830,""
353103,"",103185023,1001,"unspecified",753,"Ki","Displacement of [3H]MK801 from NMDA receptor in rat brain neuronal membrane","","","Literature",19345586,""
353104,"",103185023,1001,"unspecified","","","Ratio of Ki for rat brain NMDA receptor in presence of 100 uM spermine to Ki for rat brain NMDA receptor in absence of spermine","","","Literature",19345586,""
369249,"",103185023,1001,"active","","","Increase in ompX-lacZ expression in Escherichia coli deltaompX mutant assessed as increase in beta-galactosidase activity after 60 mins relative to control","","","Literature",17606680,""
369250,"",103185023,1001,"active","","","Increase in ompX-lacZ expression in Escherichia coli JM109 assessed as ompX upregulation after 60 mins relative to control","","","Literature",17606680,""
369251,"",103185023,1001,"active","","","Increase in ompX-lacZ expression in Escherichia coli JM109 assessed as increase in beta-galactosidase activity after 60 mins relative to control","","","Literature",17606680,""
369252,"",103185023,1001,"active","","","Increase in ompX-lacZ expression in Enterobacter aerogenes ATCC 15038 assessed as ompX upregulation after 60 mins relative to control","","","Literature",17606680,""
369253,"",103185023,1001,"active","","","Increase in ompX-lacZ expression in Enterobacter aerogenes ATCC 15038 assessed as increase in beta-galactosidase activity after 60 mins relative to control","","","Literature",17606680,""
389734,"",103185023,1001,"active",16.8,"Ki","Displacement of [3H]ketanserin from 5HT2A receptor expressed in NIH3T3 cells","","","Literature",18847250,""
434955,"",49718670,1001,"inactive","","IC90","Screen to Identify Novel Compounds That Sensitize Mycobacterium Tuberculosis to Beta-lactam Antibiotics","","","confirmatory","",""
434962,"",49718670,1001,"inactive","","","Fluorescence polarization-based cell-based primary high throughput screening assay to identify inhibitors of insulin-degrading enzyme (IDE)",155969707,"IDE gene product [Homo sapiens]","screening","",""
434973,"",49718670,1001,"inactive","","","uHTS Luminescent assay for identification of inhibitors of Sentrin-specific protease 7 (SENP7)",120538355,"SUMO1/sentrin specific peptidase 7 [Homo sapiens]","screening","",""
434989,"",49718670,1001,"inactive","","","Fluorescence-based cell-based primary high throughput screening assay to identify antagonists of the orexin 1 receptor (OX1R; HCRTR1)",222080095,"orexin receptor type 1 [Homo sapiens]","screening","",""
435003,"",49718670,1001,"inactive","","","uHTS luminescence assay for the identification of chemical inhibitors of T-cell specific antigen receptor-induced NF-kB activation","","","screening","",""
435005,"",49718670,1001,"inactive","","","Luminescence Cell-Based Primary HTS to Identify Inhibitors of Beta Cell Apoptosis.","","","screening","",""
435022,"",49718670,1001,"inactive","","","uHTS luminescence assay for the identification of chemical inhibitors of B-cell specific antigen receptor-induced NF-kB activation","","","screening","",""
435030,"",49718670,1001,"inactive","","","Absorbance-based primary bacterial cell-based high throughput screening assay to identify inhibitors of AddAB recombination protein complex",15645703,"hypothetical protein HP1089 [Helicobacter pylori 26695]","screening","",""
449728,"",49718670,1001,"inactive","","","Counterscreen for inhibitors of AddAB: absorbance-based bacterial cell-based high throughput screening assay to identify inhibitors of bacterial viability","","","screening","",""
449739,"",47193684,1001,"inactive","","","Inhibitors of Cav3 T-type Calcium Channels: Primary Screen",53832009,"voltage-dependent T-type calcium channel subunit alpha-1H isoform a [Homo sapiens]","screening","",""
449762,"",49718670,1001,"inactive","","IC50","High Throughput Screening Assay used to Identify Novel Compounds that Inhibit Mycobacterium Tuberculosis in 7H9 Media","","","confirmatory","",""
449763,"",49718670,1001,"inactive","","","uHTS identification of small molecule activators of the apoptotic arm of the Unfolded Protein response via a luminescent-based reporter assay","","","screening","",""
449768,"",47193684,1001,"inactive","","","High Throughput Screening for Cocaine Antagonists: Primary Screen",7108463,"dopamine transporter [Homo sapiens]","screening","",""
463079,"",49718670,1001,"inactive","","","Fluorescence-based counterscreen for orexin 1 receptor (OX1R) antagonists: cell-based assay to identify antagonists of the parental CHO cell line","","","screening","",""
463082,"",49718670,1001,"inactive","","","Fluorescence polarization-based primary biochemical high throughput screening assay to identify inhibitors of the plasma platelet activating factor acetylhydrolase (pPAFAH)",270133071,"PLA2G7 gene product [Homo sapiens]","screening","",""
463104,"",49718670,1001,"inactive","","","uHTS identification of small molecule activators of the adaptive arm of the Unfolded Protein response via a luminescent-based reporter assay","","","screening","",""
463111,"",49718670,1001,"inactive","","","Primary cell-based high-throughput screening assay for identification of compounds that potentiate/activate regulator of G-protein signaling 4 (RGS4)",5032039,"RGS4 gene product [Homo sapiens]","screening","",""
463141,"",49718670,1001,"inactive","","","Absorbance-based primary biochemical high throughput screening assay to identify activators of procaspase-3",14790119,"CASP3 gene product [Homo sapiens]","screening","",""
463165,"",49718670,1001,"inactive","","","Primary cell-based high-throughput screening assay for identification of compounds that inhibit regulator of   G-protein signaling 4 (RGS4)",5032039,"RGS4 gene product [Homo sapiens]","screening","",""
463190,"",49718670,1001,"inactive","","","uHTS identification of small molecule inhibitors of tim10-1 yeast via a luminescent assay",285809906,"TPA: Tim10p [Saccharomyces cerevisiae S288c]","screening","",""
463195,"",49718670,1001,"inactive","","","uHTS identification of small molecule inhibitors of tim10 yeast via a luminescent assay",285809906,"TPA: Tim10p [Saccharomyces cerevisiae S288c]","screening","",""
463210,"",49718670,1001,"inactive","","","Counterscreen for procaspase-3 activators: absorbance-based primary biochemical high throughput screening assay to identify activators of procaspase-7",55960760,"caspase 7, apoptosis-related cysteine peptidase [Homo sapiens]","screening","",""
463212,"",49718670,1001,"inactive","","","uHTS identification of small molecule inhibitors of tim23-1 yeast via a luminescent assay",285814664,"TPA: Tim23p [Saccharomyces cerevisiae S288c]","screening","",""
485270,"",49718670,1001,"inactive","","","FRET-based cell-based primary high throughput screening assay to identify antagonists of the orexin 1 receptor (OX1R; HCRTR1)",222080095,"orexin receptor type 1 [Homo sapiens]","screening","",""
485272,"",49718670,1001,"inactive","","","Fluorescence polarization-based primary biochemical high throughput screening assay to identify inhibitors of Protein Arginine Deiminase 4 (PAD4) (1536 HTS)",216548487,"protein-arginine deiminase type-4 [Homo sapiens]","screening","",""
485273,"",49718670,1001,"inactive","","","uHTS identification of UBC13 Polyubiquitin Inhibitors via a TR-FRET Assay",4507793,"UBE2N gene product [Homo sapiens]","screening","",""
485275,"",49718670,1001,"inactive","","","Phenotypic HTS multiplex for antifungal efflux pump inhibitors","","","screening","",""
485281,"",26756723,1001,"inactive","","Potency","qHTS Assay for Identification of Novel General Anesthetics",254220970,"Chain A, Horse Spleen Apoferritin","confirmatory","",""
485290,"",26756723,1001,"inactive","","Potency","qHTS Assay for Inhibitors of Tyrosyl-DNA Phosphodiesterase (TDP1)",20150581,"Chain A, Crystal Structure Of Human Tyrosyl-Dna Phosphodiesterase (Tdp1)","confirmatory","",""
485317,"",49718670,1001,"inactive","","","HTS-Luminescent assay for inhibitors of ALR by detection of hydrogen peroxide production Measured in Biochemical System Using Plate Reader - 2036-02_Inhibitor_SinglePoint_HTS",54112432,"FAD-linked sulfhydryl oxidase ALR [Homo sapiens]","screening","",""
485346,"",49718670,1001,"inactive","","","uHTS for identification of Inhibitors of Mdm2/MdmX interaction in luminescent format.",88702791,"protein Mdm4 isoform 1 [Homo sapiens]","screening","",""
488839,"",49718670,1001,"inactive","","","Development of CDK5 inhibitors   Measured in Biochemical System Using Plate Reader - 2083-01_Inhibitor_SinglePoint_HTS_Activity",20072248,"Cyclin-dependent kinase 5, regulatory subunit 1 (p35) [Homo sapiens]","screening","",""
488847,"",49718670,1001,"inactive","","","RNA aptamer-based HTS for inhibitors of GRK2",148539876,"beta-adrenergic receptor kinase 1 [Homo sapiens]","screening","",""
488862,"",49718670,1001,"inactive","","","Inhibitors of Prion Protein 5' UTR mRNA Measured in Cell-Based System Using Plate Reader - 2078-01_Inhibitor_SinglePoint_HTS_Activity","","","screening","",""
488890,"",49718670,1001,"inactive","","IC50","Elucidation of physiology of non-replicating, drug-tolerant Mycobacterium tuberculosis","","","confirmatory","",""
488895,"",49718670,1001,"inactive","","","High Throughput Screen for Tat Transport Inhibitors Measured in Microorganism System Using Plate Reader - 2093-01_Inhibitor_SinglePoint_HTS_Activity",90111653,"TatABCE protein translocation system subunit [Escherichia coli str. K-12 substr. MG1655]","screening","",""
488896,"",49718670,1001,"inactive","","","HTS using DiI-HDL to assay lipid transfer in ldlA[SR-BI] cells Measured in Cell-Based System Using Plate Reader - 2085-01_Inhibitor_SinglePoint_HTS_Activity",14389423,"Scarb1 gene product [Mus musculus]","screening","",""
488899,"",49718670,1001,"inactive","","","MITF Measured in Cell-Based System Using Plate Reader - 2084-01_Inhibitor_SinglePoint_HTS_Activity",40807040,"Microphthalmia-associated transcription factor [Homo sapiens]","screening","",""
488922,"",49718670,1001,"inactive","","","Primary cell-based screen for identification of compounds that inhibit the two-pore domain potassium channel KCNK9",7706135,"KCNK9 gene product [Homo sapiens]","screening","",""
488965,"",49718670,1001,"inactive","","","Fluorescent Biochemical Primary HTS to Identify Inhibitors of P. aeruginosa PvdQ acylase Measured in Biochemical System Using Plate Reader and Imaging Combination - 2091-01_Inhibitor_SinglePoint_HTS_Activity",218891639,"pvdQ gene product [Pseudomonas aeruginosa LESB58]","screening","",""
488966,"",49718670,1001,"inactive","","IC50","Primary and Confirmatory Screening for Inhibitors of Bacterial Capsule Biogenesis","","","confirmatory","",""
488975,"",49718670,1001,"inactive","","","Primary cell-based screen for identification of compounds that inhibit the Choline Transporter (CHT)",11141885,"SLC5A7 gene product [Homo sapiens]","screening","",""
488977,"",49718670,1001,"inactive","","","Primary cell-based screen for identification of compounds that allosterically activate the Choline Transporter (CHT)",11141885,"SLC5A7 gene product [Homo sapiens]","screening","",""
489030,"",49718670,1001,"inactive","","","uHTS Fluorescent assay for identification of inhibitors of Apaf-1",187952397,"Apoptotic peptidase activating factor 1 [Homo sapiens]","screening","",""
489031,"",49718670,1001,"inactive","","","uHTS Fluorescent assay for identification of activators of Apaf-1",187952397,"Apoptotic peptidase activating factor 1 [Homo sapiens]","screening","",""
492953,"",49718670,1001,"inactive","","","Fluorescence polarization-based primary biochemical high throughput screening assay to identify inhibitors of human platelet-activating factor acetylhydrolase 1b, catalytic subunit 2 (PAFAH1B2)",296080766,"platelet-activating factor acetylhydrolase IB subunit beta isoform b [Homo sapiens]","screening","",""
492956,"",49718670,1001,"inactive","","","Fluorescence polarization-based primary biochemical high throughput screening assay to identify inhibitors of human platelet activating factor acetylhydrolase 2 (PAFAH2)",4758878,"platelet-activating factor acetylhydrolase 2, cytoplasmic [Homo sapiens]","screening","",""
492972,"",49718670,1001,"inactive","","","Fluorescence polarization-based primary biochemical high throughput screening assay to identify inhibitors of human platelet-activating factor acetylhydrolase 1B, catalytic subunit 3 (PAFAH1B3)",225543099,"platelet-activating factor acetylhydrolase IB subunit gamma [Homo sapiens]","screening","",""
493005,"",49718670,1001,"inactive","","Potency","qHTS Assay for Iinhibitors of HIV-1 Budding by Blocking the Interaction of PTAP/TSG101",5454140,"TSG101 gene product [Homo sapiens]","confirmatory","",""
493008,"",49718670,1001,"inactive","","","Fluorescence-based biochemical primary high throughput screening assay to identify activators of the calcium sensitivity of cardiac Regulated Thin Filaments (RTF)",1927,"cardiac alpha tropomyosin [Sus scrofa]","screening","",""
493011,"",49718670,1001,"inactive","","","uHTS identification of APOBEC3A DNA Deaminase Inhibitors via a fluorescence-based single-stranded DNA deaminase assay",21955158,"APOBEC3A gene product [Homo sapiens]","screening","",""
493012,"",49718670,1001,"inactive","","","uHTS identification of APOBEC3G DNA Deaminase Inhibitors via a fluorescence-based single-stranded DNA deaminase assay",13399304,"APOBEC3G gene product [Homo sapiens]","screening","",""
493036,"",49718670,1001,"inactive","","","Image-Based HTS for Selective Agonists for NTR1",110611243,"NTSR1 gene product [Homo sapiens]","screening","",""
493087,"",49718670,1001,"inactive","","","Fluorescence polarization-based cell-based primary high throughput screening assay to identify activators of insulin-degrading enzyme (IDE)",155969707,"IDE gene product [Homo sapiens]","screening","",""
493091,"",49718670,1001,"inactive","","","uHTS Colorimetric assay for identification of inhibitors of Scp-1",10864009,"carboxy-terminal domain RNA polymerase II polypeptide A small phosphatase 1 isoform 1 [Homo sapiens]","screening","",""
493098,"",49718670,1001,"inactive","","","uHTS identification of small molecule antagonists of the CCR6 receptor via a luminescent beta-arrestin assay",37187860,"CCR6 gene product [Homo sapiens]","screening","",""
493131,"",49718670,1001,"inactive","","","Activator for delta FosB/delta FosB homodimer Measured in Biochemical System Using Plate Reader - 2072-01_Activator_SinglePoint_HTS_Activity",6679827,"protein fosB [Mus musculus]","screening","",""
493160,"",49718670,1001,"inactive","","","uHTS Fluorescent assay for identification of inhibitors of hexokinase domain containing  I (HKDC1)",156151420,"putative hexokinase HKDC1 [Homo sapiens]","screening","",""
493187,"",49718670,1001,"inactive","","","uHTS Fluorescent assay for identification of activators of hexokinase domain containing  I (HKDC1)",156151420,"putative hexokinase HKDC1 [Homo sapiens]","screening","",""
493244,"",49718670,1001,"inactive","","","Fluorescence-based biochemical primary high throughput screening assay to identify inhibitors of the calcium sensitivity of cardiac Regulated Thin Filaments (RTF)",1927,"cardiac alpha tropomyosin [Sus scrofa]","screening","",""
504326,"",49718670,1001,"inactive","","","Luminescence-based cell-based primary high throughput screening assay to identify agonists of heterodimerization of the mu 1 (OPRM1) and delta 1 (OPRD1) opioid receptors",63477962,"OPRD1 gene product [Homo sapiens]","screening","",""
504327,"",26756723,1001,"inactive","","Potency","qHTS Assay for Inhibitors of GCN5L2",153791535,"histone acetyltransferase KAT2A [Homo sapiens]","confirmatory","",""
504329,"",49718670,1001,"inactive","","IC50","Discovery of Small Molecule Probes for H1N1 Influenza NS1A",227977143,"nonstructural protein 1 [Influenza A virus (A/California/07/2009(H1N1))]","confirmatory","",""
504332,"",26756723,1001,"inactive","","Potency","qHTS Assay for Inhibitors of Histone Lysine Methyltransferase G9a",168985070,"euchromatic histone-lysine N-methyltransferase 2 [Homo sapiens]","confirmatory","",""
504339,"",49718670,1001,"inactive","","Potency","qHTS Assay for Inhibitors of JMJD2A-Tudor Domain",162330054,"Chain A, Jmjd2a Tandem Tudor Domains In Complex With A Trimethylated Histone H4-K20 Peptide","confirmatory","",""
504357,"",49718670,1001,"inactive","","","Luminescence-based cell-based primary high throughput screening assay to identify inverse agonists of heterodimerization of the mu 1 (OPRM1) and delta 1 (OPRD1) opioid receptors",63477962,"OPRD1 gene product [Homo sapiens]","screening","",""
504406,"",49718670,1001,"inactive","","","Inhibitors of Mycobacterium tuberculosis UDP-galactopyranose mutase (UGM) enzyme - High throughput screening using Fluorescent polarization assay Measured in Biochemical System Using Plate Reader - 2105-01_Inhibitor_SinglePoint_HTS_Activity_Set6",15610945,"glf gene product [Mycobacterium tuberculosis H37Rv]","screening","",""
504408,"",49718670,1001,"inactive","","","Heat Shock Factor-1 (HSF-1) Measured in Cell-Based System Using Plate Reader - 2038-01_Activator_SinglePoint_HTS_Activity","","","screening","",""
504411,"",49718670,1001,"inactive","","","Fluorescence-based primary biochemical high throughput screening assay to identify inhibitors of human diacylglycerol lipase, beta (DAGLB)",218931251,"sn1-specific diacylglycerol lipase beta isoform 1 [Homo sapiens]","screening","",""
504414,"",49718670,1001,"inactive","","","Fluorescence Polarization with Cer CAL-PDZ Measured in Biochemical System Using Plate Reader - 2109-01_Inhibitor_SinglePoint_HTS_Activity",9966877,"Golgi-associated PDZ and coiled-coil motif-containing protein isoform a [Homo sapiens]","screening","",""
504423,"",49718670,1001,"inactive","","","C-LANA FP assay Measured in Biochemical System Using Plate Reader - 2117-01_Inhibitor_SinglePoint_HTS_Activity",312275222,"LANA [Human herpesvirus 8]","screening","",""
504441,"",49718670,1001,"inactive","","","Dyrk1 A HTS Measured in Biochemical System Using Plate Reader - 2124-01_Inhibitor_SinglePoint_HTS_Activity",6978787,"dual specificity tyrosine-phosphorylation-regulated kinase 1A [Rattus norvegicus]","screening","",""
504444,"",49718670,1001,"inactive","","Potency","Nrf2 qHTS screen for inhibitors",224028257,"nuclear factor erythroid 2-related factor 2 isoform 2 [Homo sapiens]","confirmatory","",""
504454,"",49718670,1001,"inactive","","","HTS for Beta-2AR agonists via FAP method",4501969,"ADRB2 gene product [Homo sapiens]","screening","",""
504462,"",49718670,1001,"inactive","","","uHTS fluorescent assay for identification of inhibitors of ATG4B",47132611,"cysteine protease ATG4B isoform a [Homo sapiens]","screening","",""
504490,"",49718670,1001,"inactive","","","Assay for Inhibitors of the beta-Arrestin-Adaptor Protein 2 Interaction That Mediate GPCR Degradation and Recycling",13177715,"Arrestin, beta 1 [Homo sapiens]","screening","",""
504523,"",49718670,1001,"inactive","","","Fluorescence polarization to screen for inhibitors that disrupt the protein-protein interaction between Keap1 and Nrf2   Measured in Biochemical System Using Plate Reader - 2119-01_Inhibitor_SinglePoint_HTS_Activity",45269145,"KEAP1 gene product [Homo sapiens]","screening","",""
504558,"",49718670,1001,"inactive","","","Inhibitors of Epstein-Barr LMP1 inducible NF-kappaB luciferase reporter Measured in Cell-Based System Using Plate Reader - 2122-01_Inhibitor_SinglePoint_HTS_Activity",23893668,"LMP1 [Human herpesvirus 4]","screening","",""
504577,"",49718670,1001,"inactive","","","HTS of Small Molecules that Regulate V-ATPase Proton Transport in Yeast using pHLuorin",6325022,"Vma11p [Saccharomyces cerevisiae S288c]","screening","",""
504582,"",49718670,1001,"inactive","","","In vivo-based yeast HTS to detect compounds rescuing yeast growth/survival of Plasmodium Falciparum HSP40-mediated toxicity Measured in Whole Organism System Using Plate Reader - 2120-01_Inhibitor_SinglePoint_HTS_Activity",124809271,"HSP40, subfamily A, putative [Plasmodium falciparum 3D7]","screening","",""
504621,"",49718670,1001,"inactive","","","Anti-Malarial Hsp90 Inhibitors Measured in Microorganism System Using Plate Reader - 2121-01_Inhibitor_SinglePoint_HTS_Activity_Set2",124809506,"HSP90 [Plasmodium falciparum 3D7]","screening","",""
504634,"",49718670,1001,"inactive","","","Counterscreen for inverse agonists of OPRM1-OPRD1 heterodimerization: luminescence-based cell-based full-deck high throughput screening assay to identify inverse agonists of 5-hydroxytryptamine (serotonin) 5A receptor (HTR5A)",13236497,"HTR5A gene product [Homo sapiens]","screening","",""
504648,"",49718670,1001,"inactive","","Potency","Nrf2 qHTS screen for inhibitors: counterscreen for cytotoxicity","","","confirmatory","",""
504690,"",49718670,1001,"inactive","","","uHTS identification of small molecule inhibitors of Plasmodium falciparum Glucose-6-phosphate dehydrogenase via a fluorescence intensity assay",12381848,"glucose-6-phosphate dehydrogenase-6-phosphogluconolactonase [Plasmodium berghei]","screening","",""
504692,"",49718670,1001,"inactive","","","Counterscreen for agonists of OPRM1-OPRD1 heterodimerization: luminescence-based cell-based full-deck high throughput screening assay to identify agonists of 5-hydroxytryptamine (serotonin) 5A receptor (HTR5A)",13236497,"HTR5A gene product [Homo sapiens]","screening","",""
504700,"",49718670,1001,"inactive","","","Fluorescence polarization-based biochemical primary high throughput screening assay to identify activators of the Protein Kinase A-R2B (PKA-R2B) complex",46909587,"cAMP-dependent protein kinase catalytic subunit beta isoform 3 [Homo sapiens]","screening","",""
504707,"",49718670,1001,"inactive","","","Fluorescence polarization-based biochemical primary high throughput screening assay to identify activators of the Protein Kinase A-R1A (PKA-R1A) complex",6755076,"cAMP-dependent protein kinase catalytic subunit beta isoform 1 [Mus musculus]","screening","",""
504720,"",49718670,1001,"inactive","","","uHTS identification of MazEF TA System activators  via a fluorescence-based single-stranded RNase assay",16130689,"mRNA interferase toxin, antitoxin is MazE [Escherichia coli str. K-12 substr. MG1655]","screening","",""
504734,"",49718670,1001,"inactive","","","Fluorescence-based cell-based primary high throughput screening assay to identify inhibitors of TLR9-MyD88 binding.",194068499,"toll-like receptor 9 [Homo sapiens]","screening","",""
504766,"",49718670,1001,"inactive","","","Luminescence-based primary cell-based high throughput screening assay to identify inhibitors of the orphan nuclear receptor subfamily 0, group B, member 1 (DAX1; NR0B1)",5016090,"NR0B1 gene product [Homo sapiens]","screening","",""
504775,"",49718670,1001,"inactive","","","HTS using DiI-HDL to assay lipid transfer in ldlA[SR-BI] cells Measured in Cell-Based System Using Plate Reader - 2085-01_Activator_SinglePoint_HTS_Activity",14389423,"Scarb1 gene product [Mus musculus]","screening","",""
504803,"",49718670,1001,"inactive","","","Fluorescence polarization-based primary biochemical high throughput screening assay to identify inhibitors of the HTRA serine peptidase 1 (HTRA1)",121945198,"HTRA1 protein","screening","",""
504845,"",49718670,1001,"inactive","","Potency","Inhibitors of Regulator of G Protein Signaling (RGS) 4: qHTS",86301163,"regulator of G-protein signaling 4 [Homo sapiens]","confirmatory","",""
504845,"",26756723,1001,"inactive","","Potency","Inhibitors of Regulator of G Protein Signaling (RGS) 4: qHTS",86301163,"regulator of G-protein signaling 4 [Homo sapiens]","confirmatory","",""
504847,"",26756723,1001,"inactive","","Potency","Inhibitors of the vitamin D receptor (VDR): qHTS",63054845,"vitamin D3 receptor isoform VDRA [Homo sapiens]","confirmatory","",""
504847,"",49718670,1001,"inactive","","Potency","Inhibitors of the vitamin D receptor (VDR): qHTS",63054845,"vitamin D3 receptor isoform VDRA [Homo sapiens]","confirmatory","",""
504884,"",49718670,1001,"inactive","","","Inhibitors of Y. pestis Topo-I using cleavage product accumulation Measured in Biochemical System Using Plate Reader - 2123-01_Inhibitor_SinglePoint_HTS_Activity",115347926,"DNA topoisomerase I [Yersinia pestis CO92]","screening","",""
504891,"",49718670,1001,"inactive","","Potency","qHTS Assay to Find Inhibitors of Pin1",5453898,"PIN1 gene product [Homo sapiens]","confirmatory","",""
504894,"",49718670,1001,"inactive","","Potency","Activators of T cell receptors: qHTS campaign",553160,"T cell receptor [Homo sapiens]","confirmatory","",""
504937,"",49718670,1001,"inactive","","Potency","Inhibitors of Secretory Acid Sphingomyelinase (S-ASM): qHTS",179095,"acid sphingomyelinase [Homo sapiens]","confirmatory","",""
540253,"",49718670,1001,"inactive","","Potency","qHTS Assay for Inhibitors of RanGTP induced Rango (Ran-regulated importin-beta cargo) - Importin beta complex dissociation",5031833,"snurportin-1 [Homo sapiens]","confirmatory","",""
540263,"",49718670,1001,"inactive","","Potency","qHTS Assay for Inhibitors of Rango (Ran-regulated importin-beta cargo) - Importin beta complex formation",5031833,"snurportin-1 [Homo sapiens]","confirmatory","",""
540267,"",49718670,1001,"inactive","","","Small Molecules that selectively kill Giardia lamblia: qHTS","","","screening","",""
540295,"",49718670,1001,"inactive","","","TRFRET-based cell-based primary high throughput screening assay to identify biased ligands of the melanocortin 4 receptor (MC4R): antagonists of MC4R",119508433,"melanocortin receptor 4 [Homo sapiens]","screening","",""
540303,"",49718670,1001,"inactive","","Potency","qHTS for Inhibitors of Cell Surface uPA Generation",6679377,"urokinase-type plasminogen activator [Mus musculus]","confirmatory","",""
540308,"",49718670,1001,"inactive","","","Luminescence-based cell-based primary high throughput screening assay to identify biased ligands of the melanocortin 4 receptor (MC4R): agonists of MC4R",119508433,"melanocortin receptor 4 [Homo sapiens]","screening","",""
540317,"",49718670,1001,"inactive",2.8184,"Potency","HTS for Inhibitors of HP1-beta Chromodomain Interactions with Methylated Histone Tails",187960037,"chromobox protein homolog 1 [Homo sapiens]","confirmatory","",""
540336,"",49718670,1001,"inactive","","","Rtt109/Vps75 Measured in Biochemical System Using Plate Reader - 2106-01_Inhibitor_SinglePoint_HTS_Activity",68474550,"hypothetical protein CaO19.7491 [Candida albicans SC5314]","screening","",""
540364,"",49718670,1001,"inactive","","","Luminescence-based cell-based primary high throughput screening assay to identify activators of the GAA850 frataxin (FXN) promoter","","","screening","",""
588334,"",49718670,1001,"inactive","","","MITF Measured in Cell-Based System Using Plate Reader - 2084-01_Activator_SinglePoint_HTS_Activity","","","screening","",""
588335,"",49718670,1001,"inactive","","","Counterscreen for inhibitors of the fructose-bisphosphate aldolase (FBA) of M. tuberculosis: Absorbance-based biochemical high throughput Glycerophosphate Dehydrogenase-Triosephosphate Isomerase (GDH-TPI) full deck assay to identify assay artifacts","","","screening","",""
588352,"",49718670,1001,"inactive","","","Luminescence-based cell-based primary high throughput screening assay to identify inhibitors of the Steroid Receptor Coactivator 3 (SRC3; NCOA3)",32307126,"nuclear receptor coactivator 3 isoform a [Homo sapiens]","screening","",""
588354,"",49718670,1001,"inactive","","","Luminescence-based cell-based primary high throughput screening assay to identify inhibitors of the Steroid Receptor Coactivator 1 (SRC1; NCOA1)",22538455,"nuclear receptor coactivator 1 isoform 1 [Homo sapiens]","screening","",""
588358,"",49718670,1001,"inactive","","","HTS to Find Inhibitors of Pathogenic Pemphigus Antibodies","","","screening","",""
588405,"",49718670,1001,"inactive","","","HTS Assay for Peg3 Promoter Inhibitors",78486550,"Ppp1r15a gene product [Rattus norvegicus]","screening","",""
588413,"",49718670,1001,"inactive","","","uHTS identification of Gli-Sufu Antagonists in a luminescence reporter assay",6009644,"Gli1 [Mus musculus]","screening","",""
588436,"",49718670,1001,"inactive","","","Cholera Quorum: HTS for inducers of light production in the absence ofautoinducers using BH1578 (luxS deficient, cqsA deficient) Measured in Microorganism System Using Plate Reader - 2132-01_Agonist_SinglePoint_HTS_Activity","","","screening","",""
588453,"",49718670,1001,"inactive","","Potency","qHTS Assay for Inhibitors of Mammalian Selenoprotein Thioredoxin Reductase 1 (TrxR1): qHTS",8659577,"thioredoxin reductase [Rattus norvegicus]","confirmatory","",""
588456,"",49718670,1001,"inactive","","Potency","qHTS Assay for Substrates of Mammalian Selenoprotein Thioredoxin Reductase 1 (TrxR1): qHTS",8659577,"thioredoxin reductase [Rattus norvegicus]","confirmatory","",""
588458,"",49718670,1001,"inactive","","","uHTS identification of DNMT1 inhibitors in a Fluorescent Molecular Beacon assay",4503351,"DNA (cytosine-5)-methyltransferase 1 isoform b [Homo sapiens]","screening","",""
588473,"",49718670,1001,"inactive","","","uHTS identification of agonists of the CRF-binding protein and CRF-R2 receptor complex",30219,"corticotropin releasing factor-binding protein [Homo sapiens]","screening","",""
588475,"",49718670,1001,"inactive","","","uHTS identification of antagonists of the CRF-binding protein and CRF-R2 receptor complex",30219,"corticotropin releasing factor-binding protein [Homo sapiens]","screening","",""
588478,"",124811907,1001,"inactive","","","A screen for small molecule inhibitors of the human deubiquitinating enzyme, UCH37",4877999,"ubiquitin C-terminal hydrolase UCH37 [Homo sapiens]","other","",""
588489,"",49718670,1001,"inactive","","","uHTS identification of microRNA-mediated mRNA deadenylation inhibitors by fluoresence polarization assay",46367787,"polyadenylate-binding protein 1 [Homo sapiens]","screening","",""
588492,"",49718670,1001,"inactive","","","uHTS identification of small molecule modulators of myocardial damage","","","screening","",""
588493,"",49718670,1001,"inactive","","","uHTS identification of inhibitors of Rpn11 in a Fluorescent Polarization assay",16306916,"PSMD14 protein [Homo sapiens]","screening","",""
588497,"",49718670,1001,"inactive","","","High-throughput multiplex microsphere screening for inhibitors of toxin protease, specifically Botulinum neurotoxin light chain F protease, MLPCN compound set",168184763,"botulinum neurotoxin type F, BoNT/F [Clostridium botulinum Bf]","screening",16604538,""
588499,"",49718670,1001,"inactive","","","High-throughput multiplex microsphere screening for inhibitors of toxin protease, specifically Botulinum neurotoxin light chain A protease, MLPCN compound set",148378801,"botulinum neurotoxin type A [Clostridium botulinum A str. ATCC 3502]","screening",16604538,""
588501,"",49718670,1001,"inactive","","","High-throughput multiplex microsphere screening for inhibitors of toxin protease, specifically Lethal Factor Protease, MLPCN compound set",21392848,"lethal factor [Bacillus anthracis str. A2012]","screening",16604538,""
588511,"",49718670,1001,"inactive","","","Primary cell-based high-throughput screening for identification of compounds that inhibit/block calcium-activated chloride channels (TMEM16A)",334278898,"Ano1 gene product [Mus musculus]","screening","",""
588549,"",49718670,1001,"inactive","","","Fluorescence polarization to screen for inhibitor that competite the binding of FadD28 to bisubstrate Measured in Biochemical System Using Plate Reader - 2147-01_Inhibitor_SinglePoint_HTS_Activity",1781172,"FATTY-ACID-CoA LIGASE FADD28 (FATTY-ACID-CoA SYNTHETASE) (FATTY-ACID-CoA SYNTHASE) [Mycobacterium tu","screening","",""
588579,"",49718670,1001,"inactive","","Potency","qHTS for Inhibitors of Polymerase Kappa",7705344,"DNA polymerase kappa [Homo sapiens]","confirmatory","",""
588579,"",26756723,1001,"inactive","","Potency","qHTS for Inhibitors of Polymerase Kappa",7705344,"DNA polymerase kappa [Homo sapiens]","confirmatory","",""
588590,"",49718670,1001,"inactive","","Potency","qHTS for Inhibitors of Polymerase Iota",154350220,"DNA polymerase iota [Homo sapiens]","confirmatory","",""
588591,"",49718670,1001,"inactive","","Potency","qHTS for Inhibitors of Polymerase Eta",5729982,"DNA polymerase eta [Homo sapiens]","confirmatory","",""
588621,"",49718670,1001,"inactive","","","uHTS identification of small molecule inhibitors of Striatal-Enriched Phosphatase via a fluorescence intensity assay",90652859,"PTPN5 gene product [Homo sapiens]","screening","",""
588627,"",49718670,1001,"inactive","","","Primary cell-based high-throughput screening for identification of compounds that activate MrgX1 receptor signaling",195969650,"MAS-related GPR member X1 [Homo sapiens]","screening","",""
588664,"",49718670,1001,"inactive","","","TRFRET-based biochemical primary high throughput screening assay to identify inhibitors of the interaction of the Ras and Rab interactor 1 protein (Rin1) and the c-abl oncogene 1, non-receptor tyrosine kinase (Abl)",62362414,"ABL1 gene product [Homo sapiens]","screening","",""
588674,"",49718670,1001,"inactive","","","Schnurri-3 Inhibitors: specific inducers of adult bone formation Measured in Cell-Based System Using Plate Reader - 2134-01_Inhibitor_SinglePoint_HTS_Activity_Set2","","","screening","",""
588675,"",49718670,1001,"inactive","","","Primary cell-based high-throughput screening for identification of compounds that allosterically activate MrgX1 receptor signaling",195969650,"MAS-related GPR member X1 [Homo sapiens]","screening","",""
588676,"",49718670,1001,"inactive","","","Primary cell-based high-throughput screening for identification of compounds that antagonize MrgX1 receptor signaling",195969650,"MAS-related GPR member X1 [Homo sapiens]","screening","",""
588689,"",49718670,1001,"inactive","","IC50","Primary and Confirmatory Screening for Flavivirus Genomic Capping Enzyme Inhibition",219689243,"Chain A, Crystal Structure Of Dengue-2 Virus Methyltransferase Complexed With S-Adenosyl-L-Homocyste","confirmatory","",""
588692,"",49718670,1001,"inactive","","","Luciferase Reporter Cell Based HTS to identify inhibitors of N-linked Glycosylation Measured in Cell-Based System Using Plate Reader - 2146-01_Inhibitor_SinglePoint_HTS_Activity_Set2","","","screening","",""
588726,"",49718670,1001,"inactive","","","Fluorescence-based biochemical primary high throughput screening assay to identify inhibitors of the fructose-bisphosphate aldolase (FBA) of M. tuberculosis",15607504,"Probable fructose-bisphosphate aldolase Fba [Mycobacterium tuberculosis H37Rv]","screening","",""
588727,"",49718670,1001,"inactive","","IC50","A Cell-Based Confirmatory Screen for Compounds that Inhibit VEEV, TC-83","","","confirmatory","",""
588795,"",49718670,1001,"inactive","","Potency","qHTS Assay for the Inhibitors of Human Flap endonuclease 1 (FEN1).",4758356,"flap endonuclease 1 [Homo sapiens]","confirmatory","",""
588814,"",49718670,1001,"inactive","","","Fluorescence-based cell-based primary high throughput screening assay to identify agonists of the human cholinergic receptor, muscarinic 1 (CHRM1)",37622910,"CHRM1 gene product [Homo sapiens]","screening","",""
588819,"",49718670,1001,"inactive","","","Fluorescence-based cell-based primary high throughput screening assay to identify positive allosteric modulators (PAMs) of the human M1 muscarinic receptor (CHRM1).",37622910,"CHRM1 gene product [Homo sapiens]","screening","",""
588832,"",49718670,1001,"inactive","","","Hedgehog Measured in Biochemical System Using Plate Reader - 2070-01_Inhibitor_SinglePoint_HTS_Activity",7300964,"hedgehog, isoform A [Drosophila melanogaster]","screening","",""
588850,"",49718670,1001,"inactive","","","uHTS identification of cystic fibrosis induced NFkb Inhibitors in a fluoresence assay",90421313,"CFTR gene product [Homo sapiens]","screening","",""
588852,"",49718670,1001,"inactive","","","Fluorescence-based cell-based primary high throughput screening assay to identify antagonists of the human M1 muscarinic receptor (CHRM1)",37622910,"CHRM1 gene product [Homo sapiens]","screening","",""
588855,"",49718670,1001,"inactive","","Potency","qHTS for Inhibitors of TGF-b",18418623,"Smad3 [Homo sapiens]","confirmatory","",""
588856,"",49718670,1001,"inactive","","Potency","qHTS for Inhibitors of TGF-b: Cytotox Counterscreen","","","confirmatory","",""
602123,"",49718670,1001,"inactive","","","Fluorescence polarization-based primary biochemical high throughput screening assay to identify inhibitors of Escherichia coli DNA-binding ATP-dependent protease La (eLon)",16128424,"DNA-binding ATP-dependent protease La [Escherichia coli str. K-12 substr. MG1655]","screening","",""
602141,"",49718670,1001,"inactive","","","uHTS determination of small molecule cytotoxicity in a fluorescence assay to identify cystic fibrosis induced NFkb Inhibitors","","","screening","",""
602162,"",49718670,1001,"inactive","","","Flow Cytometric HTS Screen for inhibitors of the ABC transporter ABCB6 for MLPCN Compound Set",9955963,"ABCB6 gene product [Homo sapiens]","screening","",""
602163,"",49718670,1001,"inactive","","","Absorbance-based biochemical primary high throughput screening assay to identify activators of Methionine sulfoxide reductase A (MsrA)",73586699,"MSRA protein [Bos taurus]","screening","",""
602179,"",49718670,1001,"inactive","","Potency","qHTS for Inhibitors of mutant isocitrate dehydrogenase 1 (IDH1): qHTS",89573979,"isocitrate dehydrogenase 1 [Homo sapiens]","confirmatory","",""
602229,"",49718670,1001,"inactive","","","Luminescence-based cell-based high throughput primary screening assay to identify agonists of nuclear receptor subfamily 2, group E, member 3 (NR2E3)",216409728,"photoreceptor-specific nuclear receptor [Homo sapiens]","screening","",""
602233,"",49718670,1001,"inactive","","Potency","qHTS Assay to Find Inhibitors of Phosphoglycerate Kinase",115503961,"phosphoglycerate kinase [Trypanosoma brucei]","confirmatory","",""
602244,"",49718670,1001,"inactive","","","uHTS identification of CXCR6 Inhibitors in a B-arrestin luminescence assay",5730106,"CXCR6 gene product [Homo sapiens]","screening","",""
602247,"",49718670,1001,"inactive","","","Full deck counterscreen for positive allosteric modulators (PAMs) of the human M1 muscarinic receptor (CHRM1): Fluorescence-based cell-based high throughput screening assay to identify nonselective activators and assay artifacts using the parental CHOK1 cell line","","","screening","",""
602248,"",49718670,1001,"inactive","","","Full deck counterscreen for agonists of the human M1 muscarinic receptor (CHRM1): Fluorescence-based cell-based high throughput screening assay to identify nonselective activators and assay artifacts using the parental CHOK1 cell line","","","screening","",""
602250,"",49718670,1001,"inactive","","","Full deck counterscreen for antagonists of the human M1 muscarinic receptor (CHRM1): Fluorescence-based cell-based high throughput screening assay to identify nonselective inhibitors and assay artifacts using the parental CHOK1 cell line","","","screening","",""
602252,"",49718670,1001,"inactive","","","Fluorescence Polarization with CAL-PDZ Measured in Biochemical System Using Plate Reader - 2109-02_Inhibitor_SinglePoint_HTS_Activity",62868213,"Golgi-associated PDZ and coiled-coil motif-containing protein isoform b [Homo sapiens]","screening","",""
602261,"",49718670,1001,"inactive","","","uHTS identification of small molecule inhibitors of  the thioesterase domain of fatty acid synthase via a fluorescence intensity assay",41872631,"FASN gene product [Homo sapiens]","screening","",""
602274,"",49718670,1001,"inactive","","","uHTS luminescent assay for identification of compounds that enhance the survival of human induced pluripotent stem cells when cultured as single cells","","","screening","",""
602281,"",49718670,1001,"inactive","","","Luminescence-based biochemical primary high throughput screening assay to identify inhibitors of the interaction of the lipase co-activator protein, abhydrolase domain containing 5 (ABHD5) with perilipin-5 (MLDP; PLIN5)",31542303,"ABHD5 gene product [Homo sapiens]","screening","",""
602310,"",49718670,1001,"inactive","","Potency","qHTS for Inhibitors of Vif-A3G Interactions: qHTS",13399304,"APOBEC3G gene product [Homo sapiens]","confirmatory","",""
602313,"",49718670,1001,"inactive","","Potency","qHTS for Inhibitors of Vif-A3F Interactions: qHTS",22907044,"APOBEC3F gene product [Homo sapiens]","confirmatory","",""
602329,"",49718670,1001,"inactive","","","Identification of inhibitors of RAD54 Measured in Biochemical System Using Plate Reader - 2159-01_Inhibitor_SinglePoint_HTS_Activity",216548193,"RAD54L gene product [Homo sapiens]","screening","",""
602332,"",49718670,1001,"inactive","","Potency","qHTS for Inducers of the Endoplasmic Reticulum Stress Response (ERSR) in Human Glioma: qHTS",168984549,"heat shock 70kDa protein 5 (glucose-regulated protein, 78kDa) [Homo sapiens]","confirmatory","",""
602332,"",26756723,1001,"inactive","","Potency","qHTS for Inducers of the Endoplasmic Reticulum Stress Response (ERSR) in Human Glioma: qHTS",168984549,"heat shock 70kDa protein 5 (glucose-regulated protein, 78kDa) [Homo sapiens]","confirmatory","",""
602340,"",49718670,1001,"inactive","","","HTS for suppressors of simvastatin-induced mytoxicity in differentiated C2C12 cells Measured in Cell-Based System Using Plate Reader - 2112-01_Suppressor_SinglePoint_HTS_Activity","","","screening","",""
602342,"",49718670,1001,"inactive","","","Small molecule inhibitors of miR122  Measured in Cell-Based System Using Plate Reader - 2144-01_Inhibitor_SinglePoint_HTS_Activity","","","screening","",""
602346,"",49718670,1001,"inactive","","","Identification of VIF Inhibitors Measured in Cell-Based System Using Imaging - 2108-01_Inhibitor_SinglePoint_HTS_Activity",9629361,"Vif [Human immunodeficiency virus 1]","screening","",""
602363,"",49718670,1001,"inactive","","","Whole cell Yeast HTS to identify compounds modulating the fidelity of the start codon recognition in eukaryotes. Measured in Whole Organism System Using Plate Reader - 2155-01_Other_SinglePoint_HTS_Activity","","","screening","",""
602393,"",49718670,1001,"inactive","","","Screen for inhibitors of the SWI/SNF chromatin remodeling complex (esBAF) in mouse embryonic stem cells with Luciferase reporter assay Measured in Cell-Based System Using Plate Reader - 2141-01_Inhibitor_SinglePoint_HTS_Activity",291463269,"transcription activator BRG1 isoform 1 [Mus musculus]","screening","",""
602396,"",49718670,1001,"inactive","","","Luminescence-based cell-based primary high throughput screening assay to identify inverse agonists of the liver receptor homolog-1 (LRH-1; NR5A2)",4504343,"NR5A2 gene product [Homo sapiens]","screening","",""
602399,"",49718670,1001,"inactive","","","uHTS identification of inhibitors of NadD in a Colorimetric assay",15927174,"hypothetical protein SA1422 [Staphylococcus aureus subsp. aureus N315]","screening","",""
602405,"",49718670,1001,"inactive","","","PgID: DNTB colorimetric HTS to detect inhibitor of PgID Measured in Biochemical System Using Plate Reader - 2164-01_Inhibitor_SinglePoint_HTS_Activity",75495260,"WlaI protein (PglD)","screening","",""
602410,"",49718670,1001,"inactive","","","Primary cell-based screen for identification of compounds that inhibit the two-pore domain potassium channel KCNK3",11093520,"Kcnk3 channel [Homo sapiens]","screening","",""
602429,"",49718670,1001,"inactive","","","uHTS identification of SUMO1-mediated protein-protein interactions",1762973,"SUMO-1 [Homo sapiens]","screening","",""
602438,"",49718670,1001,"inactive","","","uHTS identification of modulators of interaction between CendR and NRP-1 using Fluorescence Polarization assay",160877737,"Chain A, Crystal Structure Of The B1b2 Domains From Human Neuropilin- 1","screening","",""
602440,"",49718670,1001,"inactive","","","uHTS Fluorescent Assay Using Nedd8 Protein Substrate for Identification of Inhibitors of Sentrin-Specific Protease 8 (SENP8)",262118306,"SENP8 gene product [Homo sapiens]","screening","",""
602449,"",49718670,1001,"inactive","","","uHTS identification of small molecule inhibitors of the mitochondrial permeability transition pore via an absorbance assay","","","screening","",""
602481,"",49718670,1001,"inactive","","","Mycobacterium tuberculosis BioA enzyme inhibitor Measured in Biochemical System Using Plate Reader - 2163-01_Inhibitor_SinglePoint_HTS_Activity",378544807,"bioA [Mycobacterium tuberculosis UT205]","screening","",""
623870,"",49718670,1001,"inactive","","","ARNT-TAC3: AlphaScreen HTS to detect disruption of ARNT/TAC3 interactions Measured in Biochemical System Using Plate Reader - 2158-01_Inhibitor_SinglePoint_HTS_Activity",2702319,"aryl hydrocarbon receptor nuclear translocator [Homo sapiens]","screening","",""
623877,"",49718670,1001,"inactive","","","Primary cell-based high-throughput screening for identification of compounds that activate/potentiate calcium-activated chloride channels (TMEM16A)",334278898,"Ano1 gene product [Mus musculus]","screening","",""
623901,"",49718670,1001,"inactive","","","Small molecule inhibitors of miR122  Measured in Cell-Based System Using Plate Reader - 2144-01_Activator_SinglePoint_HTS_Activity","","","screening","",""
624037,"",49718670,1001,"inactive","","","Fluorescence-based cell-based primary high throughput screening assay to identify agonists of the human cholinergic receptor, muscarinic 5 (CHRM5)",7108336,"CHRM5 gene product [Homo sapiens]","screening","",""
624038,"",49718670,1001,"inactive","","","Fluorescence-based cell-based primary high throughput screening assay to identify positive allosteric modulators (PAMs) of the human cholinergic receptor, muscarinic 5 (CHRM5)",7108336,"CHRM5 gene product [Homo sapiens]","screening","",""
624040,"",49718670,1001,"inactive","","","Fluorescence-based cell-based primary high throughput screening assay to identify antagonists of the human cholinergic receptor, muscarinic 5 (CHRM5)",7108336,"CHRM5 gene product [Homo sapiens]","screening","",""
624125,"",49718670,1001,"inactive","","","Fluorescence-based cell-based primary high throughput screening assay to identify antagonists of the human cholinergic receptor, muscarinic 4 (CHRM4)",52426748,"CHRM4 gene product [Homo sapiens]","screening","",""
624126,"",49718670,1001,"inactive","","","Fluorescence-based cell-based primary high throughput screening assay to identify positive allosteric modulators (PAMs) of the human cholinergic receptor, muscarinic 4 (CHRM4)",52426748,"CHRM4 gene product [Homo sapiens]","screening","",""
624127,"",49718670,1001,"inactive","","","Fluorescence-based cell-based primary high throughput screening assay to identify agonists of the human cholinergic receptor, muscarinic 4 (CHRM4)",52426748,"CHRM4 gene product [Homo sapiens]","screening","",""
624168,"",49718670,1001,"inactive","","","uHTS identification of small molecule activators of alpha dystroglycan glycosylation",47678551,"LARGE [Homo sapiens]","screening","",""
624169,"",49718670,1001,"inactive","","","Luminescence-based cell-based primary high throughput screening assay to identify agonists of the mouse 5-hydroxytryptamine (serotonin) receptor 2A (HTR2A)",27753985,"Htr2a gene product [Mus musculus]","screening","",""
624170,"",49718670,1001,"inactive","","Potency","qHTS for Inhibitors of Glutaminase (GLS)",71051501,"GLS protein [Homo sapiens]","confirmatory","",""
624171,"",49718670,1001,"inactive","","Potency","qHTS of Nrf2 Activators",693842,"Nrf2 [Homo sapiens]","confirmatory","",""
624172,"",49718670,1001,"inactive","","Potency","qHTS of GLP-1 Receptor Agonists",1724069,"glp-1 receptor [Homo sapiens]","confirmatory","",""
624173,"",49718670,1001,"inactive","","Potency","qHTS of Trypanosoma Brucei Inhibitors",62359610,"hypothetical protein, conserved [Trypanosoma brucei]","confirmatory","",""
624178,"",49718670,1001,"unspecified","","Potency","qHTS for Inhibitors of Human Acid Sphingomyelinase Assay: Native Substrate",179095,"acid sphingomyelinase [Homo sapiens]","confirmatory","",""
624202,"",49718670,1001,"inactive","","Potency","qHTS Assay to Identify Small Molecule Activators of BRCA1 Expression",1698399,"BRCA1 [Homo sapiens]","confirmatory","",""
624204,"",49718670,1001,"inactive","","","uHTS identification of small molecule inhibitors of the catalytic domain of the SUMO protease, SENP1 in a FRET assay",7657550,"SENP1 gene product [Homo sapiens]","screening","",""
624246,"",49718670,1001,"inactive","","Potency","qHTS for Small Molecule Inhibitors of the ERG Ets/DNA interaction",343478176,"ERG gene product [Homo sapiens]","confirmatory","",""
624256,"",49718670,1001,"inactive","","","HTS to identify compounds that promote myeloid differentiation with MLPCN compound set","","","screening","",""
624263,"",49718670,1001,"inactive","","Potency","A Quantitative High throughput Screen to Identify Chemical Modulators of PINK1 Expression",3063388,"Parkin [Homo sapiens]","confirmatory","",""
624267,"",49718670,1001,"inactive","","","Fluorescence-based cell-based primary high throughput screening assay to identify inhibitors of the interaction of nucleotide-binding oligomerization domain containing 2 (NOD2) and the receptor-interacting serine-threonine kinase 2 (RIPK2)",4506537,"RIPK2 gene product [Homo sapiens]","screening","",""
624268,"",49718670,1001,"inactive","","","Luminescence-based biochemical primary high throughput screening assay to identify inhibitors of Trypanosoma brucei methionyl tRNA synthetase (MetRS)",71746704,"methionyl-tRNA synthetase [Trypanosoma brucei brucei strain 927/4 GUTat10.1]","screening","",""
624288,"",49718670,1001,"inactive","","Potency","qHTS for Antagonists of gsp, the Etiologic Mutation Responsible for Fibrous Dysplasia/McCune-Albright Syndrome: qHTS",52000961,"Guanine nucleotide-binding protein G(s) subunit alpha isoforms short","confirmatory","",""
624291,"",49718670,1001,"inactive","","Potency","qHTS for Activators of Integrin-Mediated Alleviation for Muscular Dystrophy",121312,"Glycoprotein hormones alpha chain","confirmatory","",""
624296,"",49718670,1001,"inactive","","Potency","A quantitative high throughput screen for small molecules that induce DNA re-replication in MCF 10a normal breast cells.",7705682,"GMNN gene product [Homo sapiens]","confirmatory","",""
624297,"",49718670,1001,"inactive","","Potency","A quantitative high throughput screen for small molecules that induce DNA re-replication in SW480 colon adenocarcinoma cells.",7705682,"GMNN gene product [Homo sapiens]","confirmatory","",""
624304,"",49718670,1001,"inactive","","","uHTS identification of SKN-1 Inhibitors in a fluoresence assay",25148072,"Protein SKN-1, isoform b [Caenorhabditis elegans]","screening","",""
624330,"",49718670,1001,"inactive","","IC50","Discovery of small molecule inhibitors of the oncogenic and cytokinetic protein MgcRacGAP -  Primary and Confirmatory Screens",21361397,"RACGAP1 gene product [Homo sapiens]","confirmatory","",""
624352,"",49718670,1001,"inactive","","","uHTS identification of HIF-2a Inhibitors in a luminesence assay",40254439,"EPAS1 gene product [Homo sapiens]","screening","",""
624354,"",49718670,1001,"inactive","","","uHTS identification of Caspase-8 TRAIL sensitizers in a luminesence assay",224494019,"TNFRSF10B gene product [Homo sapiens]","screening","",""
624377,"",49718670,1001,"inactive","","","Fluorescence polarization-based biochemical primary high throughput screening assay to identify inhibitors of ArfGAP with SH3 domain, ankyrin repeat and PH domain 1 (ASAP1)",351542238,"ASAP1 gene product [Homo sapiens]","screening","",""
624416,"",49718670,1001,"inactive","","","TRFRET-based biochemical primary high throughput screening assay to identify small molecules that bind to the HIV-1-gp120 binding antibody, PG9",9629363,"Envelope surface glycoprotein gp160, precursor [Human immunodeficiency virus 1]","screening","",""
624417,"",49718670,1001,"inactive","","Potency","qHTS of GLP-1 Receptor Inverse Agonists (Inhibition Mode)",1724069,"glp-1 receptor [Homo sapiens]","confirmatory","",""
624418,"",49718670,1001,"inactive","","Potency","qHTS of GLP-1 Receptor Inverse Agonists: Cytotox Screen","","","confirmatory","",""
624463,"",49718670,1001,"inactive","","","Beta-Arrestin HTS for Positive Allosteric Modulators of the Human D2 Dopamine Receptor: Antagonists",4503385,"DRD2 gene product [Homo sapiens]","other","",""
624464,"",49718670,1001,"inactive","","","Beta-Arrestin HTS for Positive Allosteric Modulators of the Human D2 Dopamine Receptor: Potentiators",4503385,"DRD2 gene product [Homo sapiens]","other","",""
624465,"",49718670,1001,"inactive","","","Beta-Arrestin HTS for Positive Allosteric Modulators of the Human D2 Dopamine Receptor: Agonists",4503385,"DRD2 gene product [Homo sapiens]","other","",""
624466,"",49718670,1001,"active","","","Fluorescence-based cell-based primary high throughput screening assay to identify antagonists of the human trace amine associated receptor 1 (TAAR1)",21264324,"TAAR1 gene product [Homo sapiens]","screening","",""
624467,"",49718670,1001,"active","","","Fluorescence-based cell-based primary high throughput screening assay to identify agonists of the human trace amine associated receptor 1 (TAAR1)",21264324,"TAAR1 gene product [Homo sapiens]","screening","",""
624483,"",49718670,1001,"inactive","","","Counterscreen of compound fluorescence effects on High-throughput multiplex microsphere screening for inhibitors of toxin protease","","","screening","",""
635291,"",103185023,1001,"active",0.209,"EC50","Activation of rat TAAR1 expressed in Syrian hamster AV12-664 cells assessed as accumulation of cAMP after 30 mins using cAMP XS EA/CL as substrate by luminescence method",38258290,"Trace amine-associated receptor 1","Literature",22037049,""
635295,"",103185023,1001,"active",0.106,"EC50","Activation of human TAAR1 expressed in Syrian hamster AV12-664 cells co-expressing GalphaS protein assessed as accumulation of cAMP after 30 mins using cAMP XS EA/CL as substrate by luminescence method in presence of RX821002 and alprenolol",38258636,"Trace amine-associated receptor 1","Literature",22037049,""
651550,"",49718670,1001,"inactive","","","HTS Assay for Inhibitors of Akt Phophorylation: Primary Screen",60391226,"RAC-alpha serine/threonine-protein kinase","screening","",""
651560,"",49718670,1001,"inactive","","","uHTS identification of small molecule inhibitors of Low Molecular Weight Protein Tyrosine Phosphatase, LMPTP, via a fluorescence intensity assay",1709543,"Low molecular weight phosphotyrosine protein phosphatase","screening","",""
651572,"",49718670,1001,"inactive","","","Fluorescence polarization-based biochemical primary high throughput screening assay to identify inhibitors of ADP-ribosylation factor GTPase activating protein 1 (ARFGAP1)",21489979,"Arfgap1 gene product [Rattus norvegicus]","screening","",""
651602,"",49718670,1001,"inactive","","","Absorbance-based primary bacterial cell-based high throughput screening assay to identify inhibitors of RecBCD (with phage)",16130723,"exonuclease V (RecBCD complex), alpha chain [Escherichia coli str. K-12 substr. MG1655]","screening","",""
651635,"",49718670,1001,"inactive","","Potency","qHTS for Inhibitors of ATXN expression",171543895,"ATXN2 gene product [Homo sapiens]","confirmatory","",""
651636,"",49718670,1001,"inactive","","","uHTS identification of small molecule antagonists of the EBI2 receptor via a luminescent beta-arrestin assay",4826706,"GPR183 gene product [Homo sapiens]","screening","",""
651640,"",49718670,1001,"active","","","DENV2 CPE-Based HTS Measured in Cell-Based and Microorganism Combination System Using Plate Reader - 2149-01_Other_SinglePoint_HTS_Activity","","","screening","",""
651644,"",49718670,1001,"inactive","","Potency","qHTS Assay for Inhibitors of the HIV-1 protein Vpr",28872817,"Vpr [Human immunodeficiency virus 1]","confirmatory","",""
651647,"",49718670,1001,"inactive","","","uHTS identification of inhibitors of MT1-MMP activation in a fluoresence assay",4826834,"MMP14 gene product [Homo sapiens]","screening","",""
651654,"",49718670,1001,"inactive","","","HTS for the detection of C. neoformans cell lysis via adenylate kinase (AK) release Measured in Microorganism System Using Plate Reader - 2162-01_Inhibitor_SinglePoint_HTS_Activity","","","screening","",""
651658,"",49718670,1001,"inactive","","","Small Molecule Inhibitors of FGF22-Mediated Excitatory Synaptogenesis & Epilepsy Measured in Biochemical System Using RT-PCR - 7012-01_Inhibitor_SinglePoint_HTS_Activity",10190672,"FGF22 gene product [Homo sapiens]","screening","",""
651661,"",49718670,1001,"inactive","","","Luminescence Cell-Based Primary HTS to identify inhibitors of the oncoprotein EWS/Fli transcriptional activity Measured in Cell-Based System Using Plate Reader - 7014-01_Inhibitor_SinglePoint_HTS_Activity","","","screening","",""
651687,"",49718670,1001,"inactive","","","MLPCN PGC1a Modulators Measured in Cell-Based System Using Plate Reader - 2139-01_Inhibitor_SinglePoint_HTS_Activity","","","screening","",""
651699,"",49718670,1001,"inactive","","","uHTS identification of inhibitors of cullin neddylation in a TR-FRET assay",4502169,"NAE1 gene product [Homo sapiens]","screening","",""
651702,"",49718670,1001,"inactive","","","Flow Cytometric HTS Screening for Inhibitors of Lytic Granule Exocytosis with MLPCN Compound Library","","","screening","",""
651704,"",49718670,1001,"inactive","","","Inhibition of the MLL-AF4-AF9 Interaction in Pediatric Leukemia Measured in Biochemical System Using Plate Reader - 2160-01_Inhibitor_SinglePoint_HTS_Activity",156104889,"MLLT3 gene product [Homo sapiens]","screening","",""
651710,"",49718670,1001,"inactive","","","FRET-based HTS for detection of RAD52 Inhibitors Measured in Biochemical System Using Plate Reader - 7018-01_Inhibitor_SinglePoint_HTS_Activity_Set2",109637798,"RAD52 gene product [Homo sapiens]","screening","",""
651711,"",49718670,1001,"inactive","","","Turbidometric Biochemical  Primary HTS  to identify inhibitors of ERp5 Measured in Biochemical System Using Plate Reader - 7002-01_Inhibitor_SinglePoint_HTS_Activity",2501205,"Protein disulfide-isomerase A6","screening","",""
651718,"",49718670,1001,"inactive","","","Absorbance-based biochemical primary high throughput screening assay to identify inhibitors of Methionine sulfoxide reductase A (MsrA)",73586699,"MSRA protein [Bos taurus]","screening","",""
651719,"",49718670,1001,"inactive","","","Fluorescence-based cell-based primary high throughput screening assay to identify antagonists of the Galanin Receptor 3 (GalR3)",4503907,"GALR3 gene product [Homo sapiens]","screening","",""
651723,"",49718670,1001,"inactive","","","MLPCN PGC1a Modulators Measured in Cell-Based System Using Plate Reader - 2139-01_Activator_SinglePoint_HTS_Activity","","","screening","",""
651724,"",49718670,1001,"inactive","","","qHTS Assay for Inhibitors of the CtBP/E1A Interaction",1730321,"CtBP interacting protein CtIP [Homo sapiens]","screening","",""
651725,"",49718670,1001,"inactive","","","qHTS Assay for Inhibitors of the Six1/Eya2 Interaction",1246761,"six1 [Homo sapiens]","screening","",""
651768,"",49718670,1001,"inactive","","Potency","qHTS for Inhibitors of WRN Helicase",3719421,"WRN [Homo sapiens]","confirmatory","",""
651800,"",49718670,1001,"inactive","","","Fluorescence-based biochemical primary high throughput assay to identify inhibitors of T-cell receptor (TCR)-CD3 interaction using a TAMRA-labeled TCR probe",2358024,"TCRAV4S1 [Homo sapiens]","screening","",""
651819,"",49718670,1001,"inactive","","","High-Throughput Screening for Modulators of Cytosolic Chaperonin Activity",83758679,"TRIC [Homo sapiens]","screening","",""
651820,"",49718670,1001,"inactive","","Potency","qHTS Assay for Inhibitors of Hepatitis C Virus (HCV)","","","confirmatory","",""
651821,"",49718670,1001,"inactive","","","Fluorescence-based biochemical primary high throughput screening assay to identify molecules that bind r(CAG) RNA repeats","","","screening","",""
651957,"",49718670,1001,"inactive","","","Luminescence-based cell-based primary high throughput screening assay to identify inhibitors of the Steroid Receptor Coactivator 2 (SRC2; NCOA2)",5729858,"NCOA2 gene product [Homo sapiens]","screening","",""
651958,"",49718670,1001,"inactive","","","Fluorescence-based biochemical high throughput screening primary assay to identify inhibitors of Crimean-Congo Hemorrhagic Fever (CCHF) viral ovarian tumor domain protease (vOTU): Pep-AMC substrate",76364066,"putative polyprotein [Crimean-Congo hemorrhagic fever virus]","screening","",""
651965,"",49718670,1001,"inactive","","Potency","qHTS Assay for Activators of ClpP",2668494,"ClpP [Bacillus subtilis]","confirmatory","",""
651999,"",49718670,1001,"inactive","","","uHTS identification of small molecule inhibitors of Csn-mediated Deneddylation of Cullin-Ring Ligases, vis a fluorescence polarization assay","","","screening","",""
652010,"",49718670,1001,"inactive","","","Luminescence-based cell-based primary high throughput screening assay for inhibitors of the orphan nuclear receptor subfamily 0, group B, member 1 (DAX1; NR0B1): repression of SF-1 (NR5A1) activated StAR promoter by full-length DAX-1","","","screening","",""
652017,"",49718670,1001,"inactive","","","Luminescence-based cell-based primary high throughput screening assay to identify activators of the function of SWI/SNF related, matrix associated, actin dependent regulator of chromatin, subfamily a, member 2 (SMARCA2, BRM)","","","screening","",""
652025,"",49718670,1001,"inactive","","Potency","qHTS of IL-2 Activators","","","confirmatory","",""
652039,"",49718670,1001,"inactive","","","Fluorescence Intensity-based biochemical primary high throughput screening assay to identify activators of kallikrein-7 (K7) zymogen","","","screening","",""
652048,"",49718670,1001,"inactive","","","qHTS of D3 Dopamine Receptor Agonist: qHTS",89191863,"DRD3 gene product [Homo sapiens]","screening","",""
652051,"",49718670,1001,"inactive","","","qHTS of D3 Dopamine Receptor Potentiators: qHTS","","","screening","",""
652054,"",49718670,1001,"inactive","","","qHTS of D3 Dopamine Receptor Antagonist: qHTS","","","screening","",""
652067,"",49718670,1001,"inactive","","","Luminescence-based cell-based primary high throughput screening assay to identify activators of the DAF-12 from the parasite H. contortus (hcDAF-12)",71987181,"Protein DAF-12, isoform a [Caenorhabditis elegans]","screening","",""
652104,"",49718670,1001,"inactive","","Potency","qHTS of TDP-43 Inhibitors","","","confirmatory","",""
652105,"",49718670,1001,"inactive","","Potency","qHTS for Inhibitors of phosphatidylinositol 5-phosphate 4-kinase (PI5P4K)","","","confirmatory","",""
652106,"",49718670,1001,"inactive","","Potency","qHTS of alpha-syn Inhibitors","","","confirmatory","",""
652115,"",49718670,1001,"inactive","","","MLPCN SirT-5 Measured in Biochemical System Using Imaging - 7044-01_Inhibitor_SinglePoint_HTS_Activity_Set5","","","screening","",""
652126,"",49718670,1001,"inactive","","","Luminescence-based cell-based primary high throughput screening assay to identify activators of the DAF-12 from the parasite S. stercoralis (ssDAF-12)",71987181,"Protein DAF-12, isoform a [Caenorhabditis elegans]","screening","",""
652162,"",49718670,1001,"inactive","","","C. difficile toxins: HTS for inhibitors of TcdB glycohydrolase activity Measured in Biochemical System Using Plate Reader - 7074-01_Inhibitor_SinglePoint_HTS_Activity",126698238,"Toxin B [Clostridium difficile 630]","screening","",""
652163,"",49718670,1001,"inactive","","","S100A4: HTS Measured in Biochemical System Using Plate Reader - 7045-01_Inhibitor_SinglePoint_HTS_Activity","","","screening","",""
652197,"",49718670,1001,"inactive","","","MLPCN ERAP1 Measured in Biochemical System Using Plate Reader - 7016-01_Inhibitor_SinglePoint_HTS_Activity","","","screening","",""
652257,"",49718670,1001,"inactive","","","Primary biochemical fluorescence polarization-based high throughput screening assay to identify inhibitors of protein arginine methyltransferase 1 (PRMT1)",32425330,"PRMT1 protein [Homo sapiens]","screening","",""
681336,"",103185023,1001,"unspecified","","","TP_TRANSPORTER: cell accumulation of 0.05u daunomycin in MCF-7/ADR cells","","","","",""
686940,"",49718670,1001,"inactive","","","Luminescence-based cell-based primary high throughput screening assay to identify inhibitors of COUP-TFII (NR2F2)","","","screening","",""
686964,"",49718670,1001,"inactive","","","TRFRET-based biochemical primary high throughput screening assay to identify inhibitors of 5-meCpG-binding domain protein 2 (MBD2)-DBD binding to methylated oligonucleotide","","","screening","",""
686970,"",49718670,1001,"inactive","","Potency","qHTS for induction of synthetic lethality in tumor cells producing 2HG: qHTS for the HT-1080-NT fibrosarcoma cell line",49168486,"IDH1 [Homo sapiens]","confirmatory","",""
686971,"",49718670,1001,"inactive","","Potency","qHTS for induction of synthetic lethality in tumor cells producing 2HG: qHTS for the HT-1080-IDH1KD cell line","","","confirmatory","",""
686978,"",49718670,1001,"inactive","","Potency","qHTS for Inhibitors of human tyrosyl-DNA phosphodiesterase 1 (TDP1): qHTS in cells in absence of CPT","","","confirmatory","",""
686978,"",26756723,1001,"inactive","","Potency","qHTS for Inhibitors of human tyrosyl-DNA phosphodiesterase 1 (TDP1): qHTS in cells in absence of CPT","","","confirmatory","",""
686979,"",26756723,1001,"inactive","","Potency","qHTS for Inhibitors of human tyrosyl-DNA phosphodiesterase 1 (TDP1): qHTS in cells in presence of CPT","","","confirmatory","",""
686979,"",49718670,1001,"inactive","","Potency","qHTS for Inhibitors of human tyrosyl-DNA phosphodiesterase 1 (TDP1): qHTS in cells in presence of CPT","","","confirmatory","",""