Bookmark and Share
imatinib (CID 5291) - Compound BioActivity Data
.
Filters: All Data » confirmatory      
Filter selected
BioActivity Outcomes:
Active(11)
 
 
Inactive(126)
 
 
Inconclusive(12)
 
 
Unspecified(2)
 
 
Top Targets:
PTKc Abl(6)
 
 
 
ANK(5)
 
 
PLDc mTdp1 2(5)
 
 
 
 
PTKc Kit(5)
 
 
PKc like(4)
 
 
BioAssay Types:
Confirmatory(150)
 
 
 
 
 
Literature(1)
 
 
BioActivity Types:
Potency(110)
 
 
 
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 88    Data Row: 151   Total Pages: 4   Display: Page     
Sort: [Click the result table header to sort]
#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID50100104]
0.7Kinase Inhibitor Selectivity Profiling Assay [AID1433_17, Type: confirmatory]epithelial discoidin domain-containing receptor 1 isoform 1 precursor [Homo sapiens] [gi:38327632]
View
2
[SID29215405]
Potency 4.2562Primary qHTS for delayed death inhibitors of the malarial parasite plastid, 48 hour incubation [AID504832, Type: confirmatory]
View
3
[SID124892207]
Potency 7.5699qHTS for Inhibitors of the Phosphatase Activity of Eya2: Carboxyl-terminal binding protein (CtBP) Counterscreen for Cherry-picked Compounds [AID720541, Type: confirmatory]C-terminal-binding protein 1 [gi:6014741]
View
4
[SID50100104]
8.5Kinase Inhibitor Selectivity Profiling Assay [AID1433_97, Type: confirmatory]tyrosine-protein kinase ABL1 isoform a [Homo sapiens] [gi:62362414]
View
5
[SID124892207]
Potency 9.53qHTS for Inhibitors of the Phosphatase Activity of Eya2: Confirmatory Assay for Cherry-picked Compounds [AID720540, Type: confirmatory]eyes absent homolog 2 isoform a [Homo sapiens] [gi:26667227]
View
6
[SID50100104]
10Kinase Inhibitor Selectivity Profiling Assay [AID1433_100, Type: confirmatory]arg tyrosine kinase isoform a [Homo sapiens] [gi:153266757]
View
7
[SID124892207]
Potency 11.2202qHTS for Inhibitors of human tyrosyl-DNA phosphodiesterase 1 (TDP1): qHTS in cells in absence of CPT [AID686978, Type: confirmatory]TDP1 protein [Homo sapiens] [gi:79154014]
View
8
[SID124892208]
Potency 12.5893qHTS for Inhibitors of TGF-b [AID588855, Type: confirmatory]Smad3 [Homo sapiens] [gi:18418623]
View
9
[SID29215405]
Potency 12.8178Biochemical firefly luciferase enzyme assay for NPC [AID624030, Type: confirmatory]Luciferase [Photinus pyralis] [gi:160794]
View
10
[SID124892207]
Potency 17.7828qHTS for Inhibitors of human tyrosyl-DNA phosphodiesterase 1 (TDP1): qHTS in cells in presence of CPT [AID686979, Type: confirmatory]TDP1 protein [Homo sapiens] [gi:79154014]
View
11
[SID124892209]
Potency 27.4038qHTS for small molecule inhibitors of Yes1 kinase: Primary Screen [AID686947, Type: Literature]tyrosine-protein kinase Yes [Homo sapiens] [gi:4885661]
View
12
[SID124892207]
Potency qHTS for Inhibitors of Human Acid Sphingomyelinase Assay: Native Substrate [AID624178, Type: confirmatory]acid sphingomyelinase [Homo sapiens] [gi:179095]
View
13
[SID124892208]
Potency qHTS for Inhibitors of Human Acid Sphingomyelinase Assay: Native Substrate [AID624178, Type: confirmatory]acid sphingomyelinase [Homo sapiens] [gi:179095]
View
14
[SID124892207]
Potency 0.3162qHTS for Inhibitors of TGF-b: Cytotox Counterscreen [AID588856, Type: confirmatory]
View
15
[SID50100104]
12Kinase Inhibitor Selectivity Profiling Assay [AID1433_73, Type: confirmatory]tyrosine-protein kinase ABL1 isoform a [Homo sapiens] [gi:62362414]
View
16
[SID50100104]
14Kinase Inhibitor Selectivity Profiling Assay [AID1433_56, Type: confirmatory]platelet-derived growth factor receptor beta precursor [Homo sapiens] [gi:4505683]
View
17
[SID50100104]
14Kinase Inhibitor Selectivity Profiling Assay [AID1433_36, Type: confirmatory]mast/stem cell growth factor receptor Kit isoform 1 precursor [Homo sapiens] [gi:4557695]
View
18
[SID50100104]
15Kinase Inhibitor Selectivity Profiling Assay [AID1433_40, Type: confirmatory]mast/stem cell growth factor receptor Kit isoform 1 precursor [Homo sapiens] [gi:4557695]
View
19
[SID50100104]
15Kinase Inhibitor Selectivity Profiling Assay [AID1433_18, Type: confirmatory]protein-tyrosine kinase [Homo sapiens] [gi:433338]
View
20
[SID50100104]
19Kinase Inhibitor Selectivity Profiling Assay [AID1433_16, Type: confirmatory]macrophage colony-stimulating factor 1 receptor precursor [Homo sapiens] [gi:27262659]
View
21
[SID50100104]
21Kinase Inhibitor Selectivity Profiling Assay [AID1433_98, Type: confirmatory]tyrosine-protein kinase ABL1 isoform a [Homo sapiens] [gi:62362414]
View
22
[SID124892208]
Potency 25.1189qHTS for Inhibitors of TGF-b: Cytotox Counterscreen [AID588856, Type: confirmatory]
View
23
[SID124892209]
Potency 29.5659Cell Proliferation Assay against a hMSC Cell Line [AID651696, Type: confirmatory]
View
24
[SID50100104]
31Kinase Inhibitor Selectivity Profiling Assay [AID1433_55, Type: confirmatory]platelet-derived growth factor receptor alpha precursor [Homo sapiens] [gi:5453870]
View
25
[SID50100104]
35Kinase Inhibitor Selectivity Profiling Assay [AID1433_96, Type: confirmatory]tyrosine-protein kinase ABL1 isoform a [Homo sapiens] [gi:62362414]
View
26
[SID124892209]
Potency 37.2212Cell Proliferation Assay against the TMD8 Cell Line [AID651645, Type: confirmatory]
View
27
[SID124892209]
Potency 37.2212Cell Proliferation Assay against the HBL1 Cell Line [AID651646, Type: confirmatory]
View
28
[SID50100104]
40Kinase Inhibitor Selectivity Profiling Assay [AID1433_89, Type: confirmatory]tyrosine-protein kinase Lck precursor [Homo sapiens] [gi:112789546]
View
29
[SID50100104]
44Kinase Inhibitor Selectivity Profiling Assay [AID1433_99, Type: confirmatory]tyrosine-protein kinase ABL1 isoform a [Homo sapiens] [gi:62362414]
View
30
[SID50100104]
71Kinase Inhibitor Selectivity Profiling Assay [AID1433_39, Type: confirmatory]mast/stem cell growth factor receptor Kit isoform 1 precursor [Homo sapiens] [gi:4557695]
View
31
[SID50100104]
77Kinase Inhibitor Selectivity Profiling Assay [AID1433_95, Type: confirmatory]tyrosine-protein kinase ABL1 isoform a [Homo sapiens] [gi:62362414]
View
32
[SID50100104]
520Kinase Inhibitor Selectivity Profiling Assay [AID1433_74, Type: confirmatory]tyrosine-protein kinase Blk [Homo sapiens] [gi:33469982]
View
33
[SID50100104]
820Kinase Inhibitor Selectivity Profiling Assay [AID1433_37, Type: confirmatory]mast/stem cell growth factor receptor Kit isoform 1 precursor [Homo sapiens] [gi:4557695]
View
34
[SID50100104]
890Kinase Inhibitor Selectivity Profiling Assay [AID1433_90, Type: confirmatory]tyrosine-protein kinase Lyn isoform A [Homo sapiens] [gi:4505055]
View
35
[SID50100104]
1000Kinase Inhibitor Selectivity Profiling Assay [AID1433_129, Type: confirmatory]cyclin-G-associated kinase isoform 1 [Homo sapiens] [gi:157384971]
View
36
[SID50100104]
1400Kinase Inhibitor Selectivity Profiling Assay [AID1433_123, Type: confirmatory]ephrin type-A receptor 8 isoform 1 precursor [Homo sapiens] [gi:10140845]
View
37
[SID50100104]
1500Kinase Inhibitor Selectivity Profiling Assay [AID1433_33, Type: confirmatory]tyrosine-protein kinase FRK [Homo sapiens] [gi:4503787]
View
38
[SID50100104]
1700Kinase Inhibitor Selectivity Profiling Assay [AID1433_92, Type: confirmatory]RAF proto-oncogene serine/threonine-protein kinase [Homo sapiens] [gi:4506401]
View
39
[SID50100104]
1900Kinase Inhibitor Selectivity Profiling Assay [AID1433_138, Type: confirmatory]maternal embryonic leucine zipper kinase isoform 1 [Homo sapiens] [gi:7661974]
View
40
[SID50100104]
2100Kinase Inhibitor Selectivity Profiling Assay [AID1433_15, Type: confirmatory]dual specificity protein kinase CLK4 [Homo sapiens] [gi:10190706]
View
41
[SID50100104]
2400Kinase Inhibitor Selectivity Profiling Assay [AID1433_86, Type: confirmatory]tyrosine-protein kinase Fgr [Homo sapiens] [gi:4885235]
View
42
[SID50100104]
2600Kinase Inhibitor Selectivity Profiling Assay [AID1433_94, Type: confirmatory]mitogen-activated protein kinase kinase kinase MLT isoform 2 [Homo sapiens] [gi:19526767]
View
43
[SID50100104]
2900Kinase Inhibitor Selectivity Profiling Assay [AID1433_38, Type: confirmatory]mast/stem cell growth factor receptor Kit isoform 1 precursor [Homo sapiens] [gi:4557695]
View
44
[SID50100104]
3100Kinase Inhibitor Selectivity Profiling Assay [AID1433_135, Type: confirmatory]mitogen-activated protein kinase 10 isoform 1 [Homo sapiens] [gi:4506081]
View
45
[SID50100104]
3100Kinase Inhibitor Selectivity Profiling Assay [AID1433_87, Type: confirmatory]tyrosine-protein kinase Fyn isoform b [Homo sapiens] [gi:23510362]
View
46
[SID50100104]
3300Kinase Inhibitor Selectivity Profiling Assay [AID1433_76, Type: confirmatory]serine/threonine-protein kinase B-raf [Homo sapiens] [gi:33188459]
View
47
[SID50100104]
4300Kinase Inhibitor Selectivity Profiling Assay [AID1433_93, Type: confirmatory]serine/threonine-protein kinase TNNI3K [Homo sapiens] [gi:7705748]
View
48
[SID50100104]
4500Kinase Inhibitor Selectivity Profiling Assay [AID1433_14, Type: confirmatory]clk1 [gi:632964]
View
49
[SID50100104]
5000Kinase Inhibitor Selectivity Profiling Assay [AID1433_134, Type: confirmatory]mitogen-activated protein kinase 8 isoform alpha1 [Homo sapiens] [gi:4506095]
View
50
[SID50100104]
5300Kinase Inhibitor Selectivity Profiling Assay [AID1433_188, Type: confirmatory]serine/threonine-protein kinase 17A [Homo sapiens] [gi:109255245]
View