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imatinib (CID 5291) - Compound BioActivity Data
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Filters: All Data » STKc AGC      
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BioActivity Outcomes:
Active(3)
 
 
Inactive(11)
 
 
Unspecified(34)
 
 
Top Targets:
STKc AGC(48)
 
 
 
 
BioAssay Types:
Literature(47)
 
 
 
 
Confirmatory(1)
 
 
BioActivity Types:
Kd(43)
 
 
 
 
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Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 48    Data Row: 48   Total Pages: 1   
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID103245522]
Kd 7.8Binding constant for PLK4 kinase domain [AID436044, Type: Literature]Serine/threonine-protein kinase PLK4 [gi:160113150]
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2
[SID103245522]
Kd 7.8Binding constant for PLK4 kinase domain [AID625076, Type: Literature]Serine/threonine-protein kinase PLK4 [gi:160113150]
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3
[SID103245522]
Kd 9Average Binding Constant for STK18 ; NA=Not Active at 10 uM [AID256607, Type: Literature]Serine/threonine-protein kinase PLK4 [gi:160113150]
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4
[SID103245522]
Kd 10Binding constant for DCAMKL3 kinase domain [AID435399, Type: Literature]Serine/threonine-protein kinase DCLK3 [gi:115502142]
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5
[SID103245522]
Kd 10Binding constant for DCAMKL3 kinase domain [AID624707, Type: Literature]Serine/threonine-protein kinase DCLK3 [gi:115502142]
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6
[SID103245522]
Kd 10Binding constant for AMPK-alpha1 kinase domain [AID435148, Type: Literature]5'-AMP-activated protein kinase catalytic subunit alpha-1 [gi:254763436]
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7
[SID103245522]
Kd 10Binding constant for AMPK-alpha1 kinase domain [AID624773, Type: Literature]5'-AMP-activated protein kinase catalytic subunit alpha-1 [gi:254763436]
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8
[SID103245522]
Kd 10Binding constant for ULK3 kinase domain [AID624818, Type: Literature]Serine/threonine-protein kinase ULK3 [gi:259016166]
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9
[SID103245522]
Kd 10Binding constant for CAMK1D kinase domain [AID435393, Type: Literature]Calcium/calmodulin-dependent protein kinase type 1D [gi:56404610]
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10
[SID103245522]
Kd 10Binding constant for CAMK1D kinase domain [AID625118, Type: Literature]Calcium/calmodulin-dependent protein kinase type 1D [gi:56404610]
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11
[SID103245522]
Kd 10Binding constant for CAMK2G kinase domain [AID435784, Type: Literature]Calcium/calmodulin-dependent protein kinase type II subunit gamma [gi:62512173]
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12
[SID103245522]
Kd 10Binding constant for CAMK2G kinase domain [AID624731, Type: Literature]Calcium/calmodulin-dependent protein kinase type II subunit gamma [gi:62512173]
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13
[SID103245522]
Kd 10Binding constant for CAMK1G kinase domain [AID435151, Type: Literature]Calcium/calmodulin-dependent protein kinase type 1G [gi:73620970]
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14
[SID103245522]
Kd 10Binding constant for CAMK1G kinase domain [AID625119, Type: Literature]Calcium/calmodulin-dependent protein kinase type 1G [gi:73620970]
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15
[SID103245522]
Kd 10Binding constant for full-length STK33 [AID436053, Type: Literature]Serine/threonine-protein kinase 33 [gi:74761329]
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16
[SID103245522]
Kd 10Binding constant for STK33 kinase domain [AID625138, Type: Literature]Serine/threonine-protein kinase 33 [gi:74761329]
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17
[SID103245522]
Kd 10Binding constant for SNRK kinase domain [AID624752, Type: Literature]SNF-related serine/threonine-protein kinase [gi:90185235]
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18
[SID103245522]
Kd 10Binding constant for PHKG2 kinase domain [AID435930, Type: Literature]Phosphorylase b kinase gamma catalytic chain, liver/testis isoform [gi:125536]
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19
[SID103245522]
Kd 10Binding constant for PHKG2 kinase domain [AID624797, Type: Literature]Phosphorylase b kinase gamma catalytic chain, liver/testis isoform [gi:125536]
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20
[SID103245522]
Kd 10Binding constant for CAMK4 kinase domain [AID435152, Type: Literature]Calcium/calmodulin-dependent protein kinase type IV [gi:2499586]
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21
[SID103245522]
Kd 10Binding constant for CAMK4 kinase domain [AID624843, Type: Literature]Calcium/calmodulin-dependent protein kinase type IV [gi:2499586]
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22
[SID103245522]
Kd 10Binding constant for full-length CAMK1 [AID436009, Type: Literature]Calcium/calmodulin-dependent protein kinase type 1 [gi:3122301]
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23
[SID103245522]
Kd 10Binding constant for CAMK1 kinase domain [AID624922, Type: Literature]Calcium/calmodulin-dependent protein kinase type 1 [gi:3122301]
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24
[SID103245522]
Kd 10Binding constant for AMPK-alpha2 kinase domain [AID435149, Type: Literature]5'-AMP-activated protein kinase catalytic subunit alpha-2 [gi:20178276]
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25
[SID103245522]
Kd 10Binding constant for AMPK-alpha2 kinase domain [AID625047, Type: Literature]5'-AMP-activated protein kinase catalytic subunit alpha-2 [gi:20178276]
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26
[SID103245522]
Kd 10Binding constant for full-length AURKC [AID436006, Type: Literature]Aurora kinase C [gi:27805738]
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27
[SID103245522]
Kd 10Binding constant for AURKC kinase domain [AID624769, Type: Literature]Aurora kinase C [gi:27805738]
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28
[SID103245522]
Kd 10Binding constant for AURKA kinase domain [AID435518, Type: Literature]Aurora kinase A [gi:27923855]
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29
[SID103245522]
Kd 10Binding constant for AURKA kinase domain [AID624919, Type: Literature]Aurora kinase A [gi:27923855]
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30
[SID103245522]
Kd 10Binding constant for CAMKK2 kinase domain [AID435648, Type: Literature]Calcium/calmodulin-dependent protein kinase kinase 2 [gi:317373374]
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31
[SID103245522]
Kd 10Binding constant for CAMKK2 kinase domain [AID625060, Type: Literature]Calcium/calmodulin-dependent protein kinase kinase 2 [gi:317373374]
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32
[SID103245522]
Kd 10Binding constant for AURKB kinase domain [AID435519, Type: Literature]Aurora kinase B [gi:317373473]
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33
[SID103245522]
Kd 10Binding constant for AURKB kinase domain [AID624772, Type: Literature]Aurora kinase B [gi:317373473]
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34
[SID103245522]
Binding affinity to human CAMKK2 isoleucine residue assessed as residual binding at 10 uM by site dependent competitive binding assay [AID592103, Type: Literature]Calcium/calmodulin-dependent protein kinase kinase 2 [gi:317373374]
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35
[SID103245522]
Inhibition of human aurora-A activity at 10 uM by radiometric assay [AID512379, Type: Literature]Aurora kinase A [gi:27923855]
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36
[SID103245522]
Inhibition of human CaMK4 activity at 10 uM by radiometric assay [AID512377, Type: Literature]Calcium/calmodulin-dependent protein kinase type IV [gi:2499586]
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37
[SID103245522]
Inhibition of rat AMPK activity at 10 uM by radiometric assay [AID512378, Type: Literature]5'-AMP-activated protein kinase catalytic subunit alpha-2 [gi:728758]
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38
[SID50100104]
7800Kinase Inhibitor Selectivity Profiling Assay [AID1433_179, Type: confirmatory]Sak [Homo sapiens] [gi:16215696]
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39
[SID103245522]
Kd Average Binding Constant for CAMK1 ; NA=Not Active at 10 uM [AID256643, Type: Literature]Calcium/calmodulin-dependent protein kinase type 1 [gi:3122301]
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40
[SID103245522]
Kd Average Binding Constant for CAMK1D ; NA=Not Active at 10 uM [AID256584, Type: Literature]Calcium/calmodulin-dependent protein kinase type 1D [gi:56404610]
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41
[SID103245522]
Kd Average Binding Constant for Aurora2 ; NA=Not Active at 10 uM [AID256613, Type: Literature]Aurora kinase A [gi:27923855]
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42
[SID103245522]
Kd Average Binding Constant for Aurora3 ; NA=Not Active at 10 uM [AID256610, Type: Literature]Aurora kinase C [gi:27805738]
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43
[SID103245522]
Kd Average Binding Constant for ULK3 m ; NA=Not Active at 10 uM [AID256563, Type: Literature]Serine/threonine-protein kinase ULK3 [gi:115311890]
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44
[SID103245522]
Kd Average Binding Constant for CAMK1G ; NA=Not Active at 10 uM [AID256581, Type: Literature]Calcium/calmodulin-dependent protein kinase type 1G [gi:73620970]
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45
[SID103245522]
Kd Average Binding Constant for CAMK2G ; NA=Not Active at 10 uM [AID256672, Type: Literature]Calcium/calmodulin-dependent protein kinase type II subunit gamma [gi:62512173]
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46
[SID103245522]
Kd Average Binding Constant for CAMKK2 ; NA=Not Active at 10 uM [AID256580, Type: Literature]Calcium/calmodulin-dependent protein kinase kinase 2 [gi:317373374]
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47
[SID103245522]
Kd Average Binding Constant for PHkg2 ; NA=Not Active at 10 uM [AID256618, Type: Literature]Phosphorylase b kinase gamma catalytic chain, liver/testis isoform [gi:125536]
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48
[SID103245522]
Kd Average Binding Constant for PRKAA1 ; NA=Not Active at 10 uM [AID256638, Type: Literature]5'-AMP-activated protein kinase catalytic subunit alpha-1 [gi:254763436]
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