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imatinib (CID 5291) - Compound BioActivity Data
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Filters: All Data » PKc like      
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BioActivity Outcomes:
Active(4)
 
 
Inactive(1)
 
 
Unspecified(14)
 
 
Top Targets:
PKc like(19)
 
 
 
 
BioAssay Types:
Literature(19)
 
 
 
 
BioActivity Types:
Kd(15)
 
 
 
 
Ki(2)
 
 
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Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 18    Data Row: 19   Total Pages: 1   
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID103245522]
Kd 0.96Binding constant for HIPK4 kinase domain [AID624720, Type: Literature]Homeodomain-interacting protein kinase 4 [gi:74762559]
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2
[SID46393540]
Ki 5Experimentally measured binding affinity data (Ki) for protein-ligand complexes derived from PDB [AID977610, Type: Literature]Chain A, Crystal Structure Of The Syk Tyrosine Kinase Domain With Gleevec [gi:56554455]
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3
[SID46393540]
Ki 5Experimentally measured binding affinity data (Ki) for protein-ligand complexes derived from PDB [AID977610, Type: Literature]Chain A, Crystal Structure Of The Syk Tyrosine Kinase Domain With Gleevec [gi:56554455]
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4
[SID46393540]
Experimentally measured binding affinity data derived from PDB [AID1811, Type: Literature]Chain A, Crystal Structure Of The Syk Tyrosine Kinase Domain With Gleevec [gi:56554455]
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5
[SID103245522]
Kd 10Binding constant for full-length p38-beta [AID435551, Type: Literature]Mitogen-activated protein kinase 11 [gi:134047835]
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6
[SID103245522]
Kd 10Binding constant for CDK4-cyclinD1 kinase domain [AID624780, Type: Literature]Cyclin-dependent kinase 4 [gi:1168867]
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7
[SID103245522]
Kd 10Binding constant for CDK4-cyclinD3 kinase domain [AID624781, Type: Literature]Cyclin-dependent kinase 4 [gi:1168867]
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8
[SID103245522]
Kd 10Binding constant for PIM3 kinase domain [AID435679, Type: Literature]Serine/threonine-protein kinase pim-3 [gi:215274221]
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9
[SID103245522]
Kd 10Binding constant for PIM3 kinase domain [AID624802, Type: Literature]Serine/threonine-protein kinase pim-3 [gi:215274221]
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10
[SID103245522]
Kd 10Binding constant for p38-beta kinase domain [AID624890, Type: Literature]Mitogen-activated protein kinase 11 [gi:134047835]
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11
[SID103245522]
Kd 10Binding constant for full-length PCTK3 [AID435826, Type: Literature]Cyclin-dependent kinase 18 [gi:116242704]
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12
[SID103245522]
Kd 10Binding constant for PCTK3 kinase domain [AID624874, Type: Literature]Cyclin-dependent kinase 18 [gi:116242704]
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13
[SID103245522]
Kd 10Binding constant for SgK110 kinase domain [AID624747, Type: Literature]Putative uncharacterized serine/threonine-protein kinase SgK110 [gi:161783904]
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14
[SID103245522]
Kd 10Binding constant for full-length SRPK2 [AID435196, Type: Literature]SRSF protein kinase 2 [gi:300669676]
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15
[SID103245522]
Kd 10Binding constant for SRPK2 kinase domain [AID624768, Type: Literature]SRSF protein kinase 2 [gi:300669676]
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16
[SID103245522]
Kd 10Binding constant for AURKB kinase domain [AID435519, Type: Literature]Aurora kinase B [gi:317373473]
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17
[SID103245522]
Kd 10Binding constant for AURKB kinase domain [AID624772, Type: Literature]Aurora kinase B [gi:317373473]
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18
[SID103245522]
Inhibition of human SAPK2b activity at 10 uM by radiometric assay [AID512375, Type: Literature]Mitogen-activated protein kinase 11 [gi:134047835]
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19
[SID103245522]
Kd Average Binding Constant for p38-beta; NA=Not Active at 10 uM [AID256658, Type: Literature]Mitogen-activated protein kinase 11 [gi:134047835]
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