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imatinib (CID 5291) - Compound BioActivity Data
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Filters: All Data » PKc like      
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BioActivity Outcomes:
Active(10)
 
 
Inactive(13)
 
 
Unspecified(62)
 
 
Top Targets:
PKc like(85)
 
 
 
 
BioAssay Types:
Literature(81)
 
 
 
 
Confirmatory(4)
 
 
BioActivity Types:
Kd(76)
 
 
 
 
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Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 82    Data Row: 85   Total Pages: 2   Display: Page     
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID103245522]
Kd 0.96Binding constant for HIPK4 kinase domain [AID624720, Type: Literature]Homeodomain-interacting protein kinase 4 [gi:74762559]
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2
[SID103245522]
Kd 2.1Binding constant for CLK4 kinase domain [AID435788, Type: Literature]Dual specificity protein kinase CLK4 [gi:34922132]
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3
[SID103245522]
Kd 2.1Binding constant for CLK4 kinase domain [AID625125, Type: Literature]Dual specificity protein kinase CLK4 [gi:34922132]
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4
[SID103245522]
Kd 2.8Average Binding Constant for STK17A ; NA=Not Active at 10 uM [AID256568, Type: Literature]Serine/threonine-protein kinase 17A [gi:317373279]
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5
[SID103245522]
Kd 4.2Average Binding Constant for CLK4 ; NA=Not Active at 10 uM [AID256577, Type: Literature]Dual specificity protein kinase CLK4 [gi:34922132]
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6
[SID103245522]
Kd 4.5Average Binding Constant for CLK1 ; NA=Not Active at 10 uM [AID256597, Type: Literature]Dual specificity protein kinase CLK1 [gi:206729857]
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7
[SID103245522]
Kd 4.5Binding constant for full-length CLK1 [AID435786, Type: Literature]Dual specificity protein kinase CLK1 [gi:206729857]
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8
[SID103245522]
Kd 4.5Binding constant for CLK1 kinase domain [AID624764, Type: Literature]Dual specificity protein kinase CLK1 [gi:206729857]
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9
[SID103245522]
Kd 5.3Binding constant for DRAK1 kinase domain [AID624968, Type: Literature]Serine/threonine-protein kinase 17A [gi:317373279]
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10
[SID103245522]
Kd 5.3Binding constant for DRAK1 kinase domain [AID435790, Type: Literature]Serine/threonine-protein kinase 17A [gi:317373279]
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11
[SID103245522]
Kd 10Binding constant for full-length CLK3 [AID436011, Type: Literature]Dual specificity protein kinase CLK3 [gi:148887358]
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12
[SID103245522]
Kd 10Binding constant for CLK3 kinase domain [AID624931, Type: Literature]Dual specificity protein kinase CLK3 [gi:148887358]
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13
[SID103245522]
Kd 10Binding constant for DYRK2 kinase domain [AID624918, Type: Literature]Dual specificity tyrosine-phosphorylation-regulated kinase 2 [gi:148887370]
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14
[SID103245522]
Kd 10Binding constant for PRP4 kinase domain [AID624750, Type: Literature]Serine/threonine-protein kinase PRP4 homolog [gi:317373526]
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15
[SID103245522]
Kd 10Binding constant for SRPK3 kinase domain [AID625078, Type: Literature]SRSF protein kinase 3 [gi:332278151]
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16
[SID103245522]
Kd 10Binding constant for full-length SRPK1 [AID435936, Type: Literature]SRSF protein kinase 1 [gi:209572680]
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17
[SID103245522]
Kd 10Binding constant for SRPK1 kinase domain [AID624903, Type: Literature]SRSF protein kinase 1 [gi:209572680]
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18
[SID103245522]
Kd 10Binding constant for WEE2 kinase domain [AID624746, Type: Literature]Wee1-like protein kinase 2 [gi:254763343]
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19
[SID103245522]
Kd 10Binding constant for AAK1 kinase domain [AID435896, Type: Literature]AP2-associated protein kinase 1 [gi:300669613]
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20
[SID103245522]
Kd 10Binding constant for AAK1 kinase domain [AID625089, Type: Literature]AP2-associated protein kinase 1 [gi:300669613]
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21
[SID103245522]
Kd 10Binding constant for full-length SRPK2 [AID435196, Type: Literature]SRSF protein kinase 2 [gi:300669676]
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22
[SID103245522]
Kd 10Binding constant for SRPK2 kinase domain [AID624768, Type: Literature]SRSF protein kinase 2 [gi:300669676]
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23
[SID103245522]
Kd 10Binding constant for TAOK3 kinase domain [AID625101, Type: Literature]Serine/threonine-protein kinase TAO3 [gi:78099183]
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24
[SID103245522]
Kd 10Binding constant for CAMKK1 kinase domain [AID435521, Type: Literature]Calcium/calmodulin-dependent protein kinase kinase 1 [gi:56404620]
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25
[SID103245522]
Kd 10Binding constant for CAMKK1 kinase domain [AID625143, Type: Literature]Calcium/calmodulin-dependent protein kinase kinase 1 [gi:56404620]
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26
[SID103245522]
Kd 10Binding constant for SNF1LK kinase domain [AID435560, Type: Literature]Serine/threonine-protein kinase SIK1 [gi:59803093]
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27
[SID103245522]
Kd 10Binding constant for SIK kinase domain [AID624733, Type: Literature]Serine/threonine-protein kinase SIK1 [gi:59803093]
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28
[SID103245522]
Kd 10Binding constant for HIPK3 kinase domain [AID625023, Type: Literature]Homeodomain-interacting protein kinase 3 [gi:61213741]
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29
[SID103245522]
Kd 10Binding constant for NIM1 kinase domain [AID624728, Type: Literature]Serine/threonine-protein kinase NIM1 [gi:74759697]
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30
[SID103245522]
Kd 10Binding constant for SNARK kinase domain [AID435559, Type: Literature]NUAK family SNF1-like kinase 2 [gi:74761376]
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31
[SID103245522]
Kd 10Binding constant for SNARK kinase domain [AID625139, Type: Literature]NUAK family SNF1-like kinase 2 [gi:74761376]
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32
[SID103245522]
Kd 10Binding constant for MKNK2 kinase domain [AID435531, Type: Literature]MAP kinase-interacting serine/threonine-protein kinase 2 [gi:90102033]
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33
[SID103245522]
Kd 10Binding constant for MKNK2 kinase domain [AID625108, Type: Literature]MAP kinase-interacting serine/threonine-protein kinase 2 [gi:90102033]
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34
[SID103245522]
Kd 10Binding constant for DLK kinase domain [AID624762, Type: Literature]Mitogen-activated protein kinase kinase kinase 12 [gi:116242624]
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35
[SID103245522]
Kd 10Binding constant for full-length p38-beta [AID435551, Type: Literature]Mitogen-activated protein kinase 11 [gi:134047835]
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36
[SID103245522]
Kd 10Binding constant for p38-beta kinase domain [AID624890, Type: Literature]Mitogen-activated protein kinase 11 [gi:134047835]
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37
[SID103245522]
Kd 10Binding constant for PKMYT1 kinase domain [AID436043, Type: Literature]Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase [gi:55976573]
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38
[SID103245522]
Kd 10Binding constant for PKMYT1 kinase domain [AID624757, Type: Literature]Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase [gi:55976573]
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39
[SID103245522]
Kd 10Binding constant for full-length DAPK2 [AID435153, Type: Literature]Death-associated protein kinase 2 [gi:38605084]
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40
[SID103245522]
Kd 10Binding constant for DAPK2 kinase domain [AID625077, Type: Literature]Death-associated protein kinase 2 [gi:38605084]
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41
[SID103245522]
Kd 10Binding constant for MAPKAPK5 kinase domain [AID435806, Type: Literature]MAP kinase-activated protein kinase 5 [gi:52000829]
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42
[SID103245522]
Kd 10Binding constant for MAPKAPK5 kinase domain [AID624923, Type: Literature]MAP kinase-activated protein kinase 5 [gi:52000829]
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43
[SID103245522]
Kd 10Binding constant for CLK2 kinase domain [AID435787, Type: Literature]Dual specificity protein kinase CLK2 [gi:1705919]
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44
[SID103245522]
Kd 10Binding constant for CLK2 kinase domain [AID624932, Type: Literature]Dual specificity protein kinase CLK2 [gi:1705919]
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45
[SID103245522]
Kd 10Binding constant for full-length GSK3B [AID435163, Type: Literature]Glycogen synthase kinase-3 beta [gi:20455502]
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46
[SID103245522]
Kd 10Binding constant for GSK3B kinase domain [AID624856, Type: Literature]Glycogen synthase kinase-3 beta [gi:20455502]
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47
[SID103245522]
Kd 10Binding constant for HIPK2 kinase domain [AID625129, Type: Literature]Homeodomain-interacting protein kinase 2 [gi:21431782]
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48
[SID103245522]
Kd 10Binding constant for full-length MKNK1 [AID435661, Type: Literature]MAP kinase-interacting serine/threonine-protein kinase 1 [gi:30316115]
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49
[SID103245522]
Kd 10Binding constant for MKNK1 kinase domain [AID624823, Type: Literature]MAP kinase-interacting serine/threonine-protein kinase 1 [gi:30316115]
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50
[SID103245522]
Kd 10Binding constant for EIF2AK1 kinase domain [AID625080, Type: Literature]Eukaryotic translation initiation factor 2-alpha kinase 1 [gi:32172458]
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