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axitinib (CID 6450551) - Compound BioActivity Data
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Filters: All Data » PKc      
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BioActivity Outcomes:
Active(8)
 
 
Unspecified(40)
 
 
Top Targets:
PKc(48)
 
 
 
BioAssay Types:
Literature(48)
 
 
 
BioActivity Types:
Kd(48)
 
 
 
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Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 48    Data Row: 48   Total Pages: 1   
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID123098392]
Kd 0.37Binding constant for STK16 kinase domain [AID624775, Type: Literature]Serine/threonine-protein kinase 16 [gi:46577677]
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2
[SID123098392]
Kd 1.3Binding constant for MYLK2 kinase domain [AID624705, Type: Literature]Myosin light chain kinase 2, skeletal/cardiac muscle [gi:24211884]
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3
[SID123098392]
Kd 1.4Binding constant for RIPK4 kinase domain [AID624763, Type: Literature]Receptor-interacting serine/threonine-protein kinase 4 [gi:10719883]
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4
[SID123098392]
Kd 1.7Binding constant for MLCK kinase domain [AID624738, Type: Literature]Myosin light chain kinase 3 [gi:254763411]
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5
[SID123098392]
Kd 2.9Binding constant for BMPR1B kinase domain [AID624825, Type: Literature]Bone morphogenetic protein receptor type-1B [gi:6226778]
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6
[SID123098392]
Kd 3.6Binding constant for ANKK1 kinase domain [AID624735, Type: Literature]Ankyrin repeat and protein kinase domain-containing protein 1 [gi:74762569]
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7
[SID123098392]
Kd 4.3Binding constant for TESK1 kinase domain [AID625056, Type: Literature]Dual specificity testis-specific protein kinase 1 [gi:209572684]
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8
[SID123098392]
Kd 5.2Binding constant for ACVR2B kinase domain [AID624820, Type: Literature]Activin receptor type-2B [gi:97535735]
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9
[SID123098392]
Kd 10Binding constant for QSK kinase domain [AID624774, Type: Literature]Serine/threonine-protein kinase SIK3 [gi:115502238]
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10
[SID123098392]
Kd 10Binding constant for BRSK2 kinase domain [AID624929, Type: Literature]Serine/threonine-protein kinase BRSK2 [gi:116241272]
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11
[SID123098392]
Kd 10Binding constant for MYLK4 kinase domain [AID624809, Type: Literature]Myosin light chain kinase family member 4 [gi:118573873]
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12
[SID123098392]
Kd 10Binding constant for SgK110 kinase domain [AID624747, Type: Literature]Uncharacterized serine/threonine-protein kinase SBK3 [gi:161783904]
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13
[SID123098392]
Kd 10Binding constant for CSNK1G3 kinase domain [AID624949, Type: Literature]Casein kinase I isoform gamma-3 [gi:47117932]
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14
[SID123098392]
Kd 10Binding constant for MELK kinase domain [AID625087, Type: Literature]Maternal embryonic leucine zipper kinase [gi:50400857]
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15
[SID123098392]
Kd 10Binding constant for SIK2 kinase domain [AID625095, Type: Literature]Serine/threonine-protein kinase SIK2 [gi:59798973]
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16
[SID123098392]
Kd 10Binding constant for BMPR1A kinase domain [AID624945, Type: Literature]Bone morphogenetic protein receptor type-1A [gi:61252444]
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17
[SID123098392]
Kd 10Binding constant for TBK1 kinase domain [AID625072, Type: Literature]Serine/threonine-protein kinase TBK1 [gi:74761953]
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18
[SID123098392]
Kd 10Binding constant for SBK1 kinase domain [AID624812, Type: Literature]Serine/threonine-protein kinase SBK1 [gi:74762155]
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19
[SID123098392]
Kd 10Binding constant for CSNK1A1L kinase domain [AID624723, Type: Literature]Casein kinase I isoform alpha-like [gi:212286065]
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20
[SID123098392]
Kd 10Binding constant for PIM3 kinase domain [AID624802, Type: Literature]Serine/threonine-protein kinase pim-3 [gi:215274221]
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21
[SID123098392]
Kd 10Binding constant for PIM1 kinase domain [AID624878, Type: Literature]Serine/threonine-protein kinase pim-1 [gi:83305339]
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22
[SID123098392]
Kd 10Binding constant for VRK2 kinase domain [AID625058, Type: Literature]Serine/threonine-protein kinase VRK2 [gi:90116515]
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23
[SID123098392]
Kd 10Binding constant for STK35 kinase domain [AID624711, Type: Literature]Serine/threonine-protein kinase 35 [gi:292495039]
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24
[SID123098392]
Kd 10Binding constant for RIPK5 kinase domain [AID624758, Type: Literature]Dual serine/threonine and tyrosine protein kinase [gi:296434486]
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25
[SID123098392]
Kd 10Binding constant for IKK-alpha kinase domain [AID624832, Type: Literature]Inhibitor of nuclear factor kappa-B kinase subunit alpha [gi:317373368]
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26
[SID123098392]
Kd 10Binding constant for DAPK1 kinase domain [AID624971, Type: Literature]Death-associated protein kinase 1 [gi:317373595]
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27
[SID123098392]
Kd 10Binding constant for BRSK1 kinase domain [AID624702, Type: Literature]Serine/threonine-protein kinase BRSK1 [gi:347595639]
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28
[SID123098392]
Kd 10Binding constant for BMPR2 kinase domain [AID624826, Type: Literature]Bone morphogenetic protein receptor type-2 [gi:12643724]
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29
[SID123098392]
Kd 10Binding constant for IKK-beta kinase domain [AID624836, Type: Literature]Inhibitor of nuclear factor kappa-B kinase subunit beta [gi:14285497]
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30
[SID123098392]
Kd 10Binding constant for DRAK2 kinase domain [AID624942, Type: Literature]Serine/threonine-protein kinase 17B [gi:14423909]
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31
[SID123098392]
Kd 10Binding constant for IKK-epsilon kinase domain [AID625074, Type: Literature]Inhibitor of nuclear factor kappa-B kinase subunit epsilon [gi:14548079]
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32
[SID123098392]
Kd 10Binding constant for CSNK1G1 kinase domain [AID625128, Type: Literature]Casein kinase I isoform gamma-1 [gi:18202957]
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33
[SID123098392]
Kd 10Binding constant for PIM2 kinase domain [AID625064, Type: Literature]Serine/threonine-protein kinase pim-2 [gi:20139243]
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34
[SID123098392]
Kd 10Binding constant for CSNK1D kinase domain [AID624716, Type: Literature]Casein kinase I isoform delta [gi:27923980]
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35
[SID123098392]
Kd 10Binding constant for TSSK1B kinase domain [AID625142, Type: Literature]Testis-specific serine/threonine-protein kinase 1 [gi:30316282]
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36
[SID123098392]
Kd 10Binding constant for CSNK1A1 kinase domain [AID624846, Type: Literature]Casein kinase I isoform alpha [gi:31077177]
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37
[SID123098392]
Kd 10Binding constant for TLK2 kinase domain [AID624771, Type: Literature]Serine/threonine-protein kinase tousled-like 2 [gi:34222826]
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38
[SID123098392]
Kd 10Binding constant for TLK1 kinase domain [AID625069, Type: Literature]Serine/threonine-protein kinase tousled-like 1 [gi:34223086]
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39
[SID123098392]
Kd 10Binding constant for DAPK3 kinase domain [AID624834, Type: Literature]Death-associated protein kinase 3 [gi:38604691]
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40
[SID123098392]
Kd 10Binding constant for ACVR2A kinase domain [AID624838, Type: Literature]Activin receptor type-2A [gi:114722]
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41
[SID123098392]
Kd 10Binding constant for ACVR1 kinase domain [AID624819, Type: Literature]Activin receptor type-1 [gi:462447]
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42
[SID123098392]
Kd 10Binding constant for ACVR1B kinase domain [AID624943, Type: Literature]Activin receptor type-1B [gi:547775]
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43
[SID123098392]
Kd 10Binding constant for TGFBR1 kinase domain [AID624961, Type: Literature]TGF-beta receptor type-1 [gi:547777]
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44
[SID123098392]
Kd 10Binding constant for CSNK1E kinase domain [AID624847, Type: Literature]Casein kinase I isoform epsilon [gi:1346369]
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45
[SID123098392]
Kd 10Binding constant for WEE1 kinase domain [AID624914, Type: Literature]Wee1-like protein kinase [gi:1351419]
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46
[SID123098392]
Kd 10Binding constant for CSNK1G2 kinase domain [AID624833, Type: Literature]Casein kinase I isoform gamma-2 [gi:3024060]
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47
[SID123098392]
Kd 10Binding constant for LKB1 kinase domain [AID624798, Type: Literature]Serine/threonine-protein kinase STK11 [gi:3024670]
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48
[SID123098392]
Kd 10Binding constant for ACVRL1 kinase domain [AID624778, Type: Literature]Serine/threonine-protein kinase receptor R3 [gi:3915750]
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