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imatinib (CID 5291) - Compound BioActivity Data
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Filters: All Data » PKc      
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BioActivity Outcomes:
Active(2)
 
 
Inactive(10)
 
 
Unspecified(85)
 
 
Top Targets:
PKc(97)
 
 
 
 
BioAssay Types:
Literature(96)
 
 
 
 
Confirmatory(1)
 
 
BioActivity Types:
Kd(94)
 
 
 
 
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Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 97    Data Row: 97   Total Pages: 2   Display: Page     
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID103245522]
Kd 1.9Binding constant for full-length MELK [AID435660, Type: Literature]Maternal embryonic leucine zipper kinase [gi:50400857]
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2
[SID103245522]
Kd 1.9Binding constant for MELK kinase domain [AID625087, Type: Literature]Maternal embryonic leucine zipper kinase [gi:50400857]
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3
[SID103245522]
Kd 10Binding constant for full-length SNF1LK2 [AID436052, Type: Literature]Serine/threonine-protein kinase SIK2 [gi:59798973]
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4
[SID103245522]
Kd 10Binding constant for SIK2 kinase domain [AID625095, Type: Literature]Serine/threonine-protein kinase SIK2 [gi:59798973]
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5
[SID103245522]
Kd 10Binding constant for BMPR1A kinase domain [AID435276, Type: Literature]Bone morphogenetic protein receptor type-1A [gi:61252444]
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6
[SID103245522]
Kd 10Binding constant for BMPR1A kinase domain [AID624945, Type: Literature]Bone morphogenetic protein receptor type-1A [gi:61252444]
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7
[SID103245522]
Kd 10Binding constant for TBK1 kinase domain [AID625072, Type: Literature]Serine/threonine-protein kinase TBK1 [gi:74761953]
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8
[SID103245522]
Kd 10Binding constant for SBK1 kinase domain [AID624812, Type: Literature]Serine/threonine-protein kinase SBK1 [gi:74762155]
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9
[SID103245522]
Kd 10Binding constant for ANKK1 kinase domain [AID436005, Type: Literature]Ankyrin repeat and protein kinase domain-containing protein 1 [gi:74762569]
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10
[SID103245522]
Kd 10Binding constant for ANKK1 kinase domain [AID624735, Type: Literature]Ankyrin repeat and protein kinase domain-containing protein 1 [gi:74762569]
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11
[SID103245522]
Kd 10Binding constant for IKK-alpha kinase domain [AID624832, Type: Literature]Inhibitor of nuclear factor kappa-B kinase subunit alpha [gi:317373368]
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12
[SID103245522]
Kd 10Binding constant for DAPK1 kinase domain [AID435283, Type: Literature]Death-associated protein kinase 1 [gi:317373595]
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13
[SID103245522]
Kd 10Binding constant for DAPK1 kinase domain [AID624971, Type: Literature]Death-associated protein kinase 1 [gi:317373595]
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14
[SID103245522]
Kd 10Binding constant for BRSK1 kinase domain [AID435782, Type: Literature]Serine/threonine-protein kinase BRSK1 [gi:347595639]
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15
[SID103245522]
Kd 10Binding constant for BRSK1 kinase domain [AID624702, Type: Literature]Serine/threonine-protein kinase BRSK1 [gi:347595639]
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16
[SID103245522]
Kd 10Binding constant for PIM2 kinase domain [AID435440, Type: Literature]Serine/threonine-protein kinase pim-2 [gi:20139243]
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17
[SID103245522]
Kd 10Binding constant for PIM2 kinase domain [AID625064, Type: Literature]Serine/threonine-protein kinase pim-2 [gi:20139243]
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18
[SID103245522]
Kd 10Binding constant for ACVR2A kinase domain [AID436004, Type: Literature]Activin receptor type-2A [gi:114722]
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19
[SID103245522]
Kd 10Binding constant for ACVR2A kinase domain [AID624838, Type: Literature]Activin receptor type-2A [gi:114722]
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20
[SID103245522]
Kd 10Binding constant for ACVR1 kinase domain [AID435274, Type: Literature]Activin receptor type-1 [gi:462447]
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21
[SID103245522]
Kd 10Binding constant for ACVR1 kinase domain [AID624819, Type: Literature]Activin receptor type-1 [gi:462447]
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22
[SID103245522]
Kd 10Binding constant for ACVR1B kinase domain [AID435898, Type: Literature]Activin receptor type-1B [gi:547775]
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23
[SID103245522]
Kd 10Binding constant for ACVR1B kinase domain [AID624943, Type: Literature]Activin receptor type-1B [gi:547775]
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24
[SID103245522]
Kd 10Binding constant for TGFBR1 kinase domain [AID435938, Type: Literature]TGF-beta receptor type-1 [gi:547777]
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25
[SID103245522]
Kd 10Binding constant for TGFBR1 kinase domain [AID624961, Type: Literature]TGF-beta receptor type-1 [gi:547777]
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26
[SID103245522]
Kd 10Binding constant for full-length CSNK1G2 [AID435282, Type: Literature]Casein kinase I isoform gamma-2 [gi:3024060]
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27
[SID103245522]
Kd 10Binding constant for CSNK1G2 kinase domain [AID624833, Type: Literature]Casein kinase I isoform gamma-2 [gi:3024060]
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28
[SID103245522]
Kd 10Binding constant for full-length LKB1 [AID435909, Type: Literature]Serine/threonine-protein kinase STK11 [gi:3024670]
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29
[SID103245522]
Kd 10Binding constant for LKB1 kinase domain [AID624798, Type: Literature]Serine/threonine-protein kinase STK11 [gi:3024670]
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30
[SID103245522]
Kd 10Binding constant for ACVRL1 kinase domain [AID435645, Type: Literature]Serine/threonine-protein kinase receptor R3 [gi:3915750]
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31
[SID103245522]
Kd 10Binding constant for ACVRL1 kinase domain [AID624778, Type: Literature]Serine/threonine-protein kinase receptor R3 [gi:3915750]
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32
[SID103245522]
Kd 10Binding constant for BMPR1B kinase domain [AID624825, Type: Literature]Bone morphogenetic protein receptor type-1B [gi:6226778]
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33
[SID103245522]
Kd 10Binding constant for full-length CSNK1E [AID435650, Type: Literature]Casein kinase I isoform epsilon [gi:1346369]
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34
[SID103245522]
Kd 10Binding constant for CSNK1E kinase domain [AID624847, Type: Literature]Casein kinase I isoform epsilon [gi:1346369]
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35
[SID103245522]
Kd 10Binding constant for WEE1 kinase domain [AID435204, Type: Literature]Wee1-like protein kinase [gi:1351419]
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36
[SID103245522]
Kd 10Binding constant for WEE1 kinase domain [AID624914, Type: Literature]Wee1-like protein kinase [gi:1351419]
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37
[SID103245522]
Kd 10Binding constant for MLCK kinase domain [AID435413, Type: Literature]Myosin light chain kinase, smooth muscle [gi:2851396]
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38
[SID103245522]
Kd 10Binding constant for RIPK4 kinase domain [AID624763, Type: Literature]Receptor-interacting serine/threonine-protein kinase 4 [gi:10719883]
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39
[SID103245522]
Kd 10Binding constant for BMPR2 kinase domain [AID435780, Type: Literature]Bone morphogenetic protein receptor type-2 [gi:12643724]
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40
[SID103245522]
Kd 10Binding constant for BMPR2 kinase domain [AID624826, Type: Literature]Bone morphogenetic protein receptor type-2 [gi:12643724]
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41
[SID103245522]
Kd 10Binding constant for full-length DRAK2 [AID435401, Type: Literature]Serine/threonine-protein kinase 17B [gi:14423909]
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42
[SID103245522]
Kd 10Binding constant for DRAK2 kinase domain [AID624942, Type: Literature]Serine/threonine-protein kinase 17B [gi:14423909]
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43
[SID103245522]
Kd 10Binding constant for full-length IKK-epsilon [AID435657, Type: Literature]Inhibitor of nuclear factor kappa-B kinase subunit epsilon [gi:14548079]
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44
[SID103245522]
Kd 10Binding constant for IKK-epsilon kinase domain [AID625074, Type: Literature]Inhibitor of nuclear factor kappa-B kinase subunit epsilon [gi:14548079]
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45
[SID103245522]
Kd 10Binding constant for IKK-beta kinase domain [AID624836, Type: Literature]Inhibitor of nuclear factor kappa-B kinase subunit beta [gi:14285497]
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46
[SID103245522]
Kd 10Binding constant for CSNK1G1 kinase domain [AID435397, Type: Literature]Casein kinase I isoform gamma-1 [gi:18202957]
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47
[SID103245522]
Kd 10Binding constant for CSNK1G1 kinase domain [AID625128, Type: Literature]Casein kinase I isoform gamma-1 [gi:18202957]
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48
[SID103245522]
Kd 10Binding constant for MYLK2 kinase domain [AID435415, Type: Literature]Myosin light chain kinase 2, skeletal/cardiac muscle [gi:24211884]
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49
[SID103245522]
Kd 10Binding constant for MYLK2 kinase domain [AID624705, Type: Literature]Myosin light chain kinase 2, skeletal/cardiac muscle [gi:24211884]
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50
[SID103245522]
Kd 10Binding constant for full-length CSNK1D [AID435524, Type: Literature]Casein kinase I isoform delta [gi:27923980]
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