Bookmark and Share
Estradiol (CID 5757) - Compound BioActivity Data
.
Filters: All Data » NR LBD AR      
Filter selected
BioActivity Outcomes:
Active(14)
 
 
Inactive(3)
 
 
Inconclusive(9)
 
 
Unspecified(1)
 
 
Top Targets:
NR LBD AR(27)
 
 
 
 
 
BioAssay Types:
Confirmatory(15)
 
 
 
 
Summary(9)
 
 
 
 
Literature(3)
 
 
 
 
BioActivity Types:
Potency(23)
 
 
 
 
IC50(2)
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 13    Data Row: 27   Total Pages: 2   Display: Page     
Sort: [Click the result table header to sort]
#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID103189263]
IC50 0.0191Inhibitory activity against AR [AID260157, Type: Literature]Androgen receptor [gi:113830]
View
2
[SID144204699]
Ratio Potency (uM) 0.0600704qHTS assay to identify small molecule antagonists of the androgen receptor (AR) signaling pathway: Summary [AID743063, Type: summary]AR protein [Homo sapiens] [gi:124375976]
View
3
[SID103189263]
IC50 0.353DRUGMATRIX: Androgen (Testosterone) AR radioligand binding (ligand: [3H] Mibolerone) [AID625228, Type: confirmatory]Androgen receptor [gi:113832]
View
4
[SID144210608]
Potency-Replicate_1 1.23qHTS assay to identify small molecule agonists of the androgen receptor (AR) signaling pathway [AID743036, Type: confirmatory]AR protein [Homo sapiens] [gi:124375976]
View
5
[SID144210608]
Potency-Replicate_1 1.3685qHTS assay to identify small molecule agonists of the androgen receptor (AR) signaling pathway using the MDA cell line [AID743040, Type: confirmatory]AR protein [Homo sapiens] [gi:124375976]
View
6
[SID144209255]
Potency-Replicate_1 1.5324qHTS assay to identify small molecule agonists of the androgen receptor (AR) signaling pathway using the MDA cell line [AID743040, Type: confirmatory]AR protein [Homo sapiens] [gi:124375976]
View
7
[SID144210608]
Ratio Potency (uM) 1.73739qHTS assay to identify small molecule agonists of the androgen receptor (AR) signaling pathway: Summary [AID743053, Type: summary]AR protein [Homo sapiens] [gi:124375976]
View
8
[SID144204699]
Potency-Replicate_1 2.1314qHTS assay to identify small molecule agonists of the androgen receptor (AR) signaling pathway [AID743036, Type: confirmatory]AR protein [Homo sapiens] [gi:124375976]
View
9
[SID144209255]
Potency-Replicate_1 2.449qHTS assay to identify small molecule agonists of the androgen receptor (AR) signaling pathway [AID743036, Type: confirmatory]AR protein [Homo sapiens] [gi:124375976]
View
10
[SID144209255]
Ratio Potency (uM) 2.77116qHTS assay to identify small molecule agonists of the androgen receptor (AR) signaling pathway: Summary [AID743053, Type: summary]AR protein [Homo sapiens] [gi:124375976]
View
11
[SID144204699]
Ratio Potency (uM) 2.8973qHTS assay to identify small molecule agonists of the androgen receptor (AR) signaling pathway: Summary [AID743053, Type: summary]AR protein [Homo sapiens] [gi:124375976]
View
12
[SID144204699]
Potency-Replicate_1 3.3491qHTS assay to identify small molecule agonists of the androgen receptor (AR) signaling pathway using the MDA cell line [AID743040, Type: confirmatory]AR protein [Homo sapiens] [gi:124375976]
View
13
[SID144210608]
Ratio Potency (uM) 51.8676qHTS assay to identify small molecule antagonists of the androgen receptor (AR) signaling pathway: Summary [AID743063, Type: summary]AR protein [Homo sapiens] [gi:124375976]
View
14
[SID144209255]
AR Potency (uM) qHTS assay to identify small molecule antagonists of the androgen receptor (AR) signaling pathway using the MDA cell line: Summary [AID743054, Type: summary]AR protein [Homo sapiens] [gi:124375976]
View
15
[SID103189263]
Binding affinity to rat ventral prostate androgen receptor at 0.01 uM [AID417711, Type: Literature]Androgen receptor [gi:113832]
View
16
[SID144204699]
Potency-Replicate_1 qHTS assay to identify small molecule antagonists of the androgen receptor (AR) signaling pathway using the MDA cell line [AID743042, Type: confirmatory]AR protein [Homo sapiens] [gi:124375976]
View
17
[SID144204699]
AR Potency (uM) qHTS assay to identify small molecule antagonists of the androgen receptor (AR) signaling pathway using the MDA cell line: Summary [AID743054, Type: summary]AR protein [Homo sapiens] [gi:124375976]
View
18
[SID144210608]
Potency-Replicate_1 qHTS assay to identify small molecule antagonists of the androgen receptor (AR) signaling pathway using the MDA cell line [AID743042, Type: confirmatory]AR protein [Homo sapiens] [gi:124375976]
View
19
[SID144204699]
Potency-Replicate_1 0.0674qHTS assay to identify small molecule antagonists of the androgen receptor (AR) signaling pathway [AID743035, Type: confirmatory]AR protein [Homo sapiens] [gi:124375976]
View
20
[SID17389898]
Potency 0.631qHTS assay for small molecule agonists of androgen receptor signaling [AID588515, Type: confirmatory]AR protein [Homo sapiens] [gi:124375976]
View