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Morphine (CID 5288826) - Compound BioActivity Data
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Filters: All Data » 7TM GPCR Srx      
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BioActivity Outcomes:
Active(99)
 
 
Inconclusive(3)
 
 
Unspecified(55)
 
 
Top Targets:
7TM GPCR Srx(157)
 
 
 
 
BioAssay Types:
Literature(153)
 
 
 
 
Confirmatory(4)
 
 
BioActivity Types:
Ki(47)
 
 
 
EC50(28)
 
 
 
IC50(24)
 
 
 
 
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Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 145    Data Row: 157   Total Pages: 8   Display: Page     
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID103169185]
Ki 0.00088Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cells [AID259394, Type: Literature]Mu-type opioid receptor [gi:2851402]
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2
[SID103169185]
Ki 0.00088Displacement of [3H]-DAMGO from human mu opioid receptor expressed in CHO cells after 60 mins by scintillation counting [AID670110, Type: Literature]Mu-type opioid receptor [gi:2851402]
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3
[SID103169185]
Ki 0.001Inhibition of [3H]DAMGO binding to mu opioid receptor of rat brain membranes [AID151606, Type: Literature]Mu-type opioid receptor [gi:464314]
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4
[SID103169185]
Ki 0.0011Displacement of [3H]DAMGO from human recombinant MOR expressed in CHO cells [AID269569, Type: Literature]Mu-type opioid receptor [gi:2851402]
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5
[SID103169185]
Ki 0.0011Displacement of [3H]DAMGO from human cloned mu opioid receptor [AID298631, Type: Literature]Mu-type opioid receptor [gi:2851402]
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6
[SID103169185]
IC50 0.00127Displacement of [3H]DAMGO from mu opioid receptor in ICR mouse whole brain [AID383161, Type: Literature]Mu-type opioid receptor [gi:1171911]
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7
[SID103169185]
IC50 0.00127Displacement of [3H]DAMGO from mu opioid receptor in mouse whole brain without cerebellum [AID411134, Type: Literature]Mu-type opioid receptor [gi:1171911]
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8
[SID103169185]
Ki 0.0018Displacement of [3H]DPDPE from delta opioid receptor in rat brain membranes [AID601797, Type: Literature]Delta-type opioid receptor [gi:464311]
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9
[SID103169185]
Ki 0.0018Binding affinity against mu opioid receptor in mouse hot plate test [AID238659, Type: Literature]Mu-type opioid receptor [gi:1171911]
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10
[SID103169185]
IC50 0.00194Inhibition of [3H]- DAMGO binding to Rat brain Opioid receptor mu 1 [AID151303, Type: Literature]Mu-type opioid receptor [gi:464314]
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11
[SID103169185]
Ki 0.0022Displacement of [3H]DAMGO from human mu opioid receptor expressed in HEK-293 cells by scintillation counting [AID669684, Type: confirmatory]Mu-type opioid receptor [gi:2851402]
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12
[SID103169185]
Ki 0.0025Binding affinity towards opioid receptor mu 2 [AID152210, Type: Literature]Mu-type opioid receptor [gi:6093615]
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13
[SID103169185]
Ki 0.00255Displacement of [125I]IOXY from human mu opioid receptor expressed in CHO cells coexpressing human recombinant MOR after 2 hrs by liquid scintillation counting [AID607794, Type: Literature]Mu-type opioid receptor [gi:2851402]
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14
[SID103169185]
Ki 0.00255Displacement of [3H]DAMGO from human recombinant mu opioid receptor expressed in CHO cells [AID440049, Type: Literature]Mu-type opioid receptor [gi:2851402]
View
15
[SID103169185]
Ki 0.0026Displacement of [3H]DAMGO from human recombinant mu opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation counting [AID612049, Type: Literature]Mu-type opioid receptor [gi:2851402]
View
16
[SID103169185]
Ki 0.0026Displacement of [3H]-DAMGO from human mu opioid receptor expressed in CHO cells membrane after 2 hrs by liquid scintillation counting [AID647794, Type: Literature]Mu-type opioid receptor [gi:2851402]
View
17
[SID103169185]
Ki 0.0026Displacement of [3H]DAMGO from human recombinant mu opioid receptor expressed in CHO cell membranes after 2 hrs by liquid scintillation counting analysis [AID749692, Type: Literature]Mu-type opioid receptor [gi:2851402]
View
18
[SID103169185]
Ki 0.0026Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation counting [AID765827, Type: Literature]Mu-type opioid receptor [gi:2851402]
View
19
[SID103169185]
Ki 0.0028Inhibition of [3H]DAMGO binding to rat brain homogenat Opioid receptor mu 1 [AID151750, Type: Literature]Mu-type opioid receptor [gi:464314]
View
20
[SID103169185]
Ki 0.003Inhibition of [3H]dihydromorphine (1 nM) binding to mu opioid receptor of rat brain homogenate [AID141761, Type: confirmatory]Mu-type opioid receptor [gi:464314]
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