Bookmark and Share
imatinib (CID 5291) - Compound BioActivity Data
.
Filters: All Data » Inactive      
Filter selected
BioActivity Outcomes:
Inactive(405)
 
 
Top Targets:
PKc like(13)
 
 
STKc AGC(11)
 
 
PKc(10)
 
 
PTKc Src like(6)
 
 
ANK(5)
 
 
BioAssay Types:
Literature(263)
 
 
Confirmatory(126)
 
 
Screening(10)
 
 
BioActivity Types:
Kd(96)
 
 
Potency(88)
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 194    Data Row: 405   Total Pages: 9   Display: Page     
Sort: [Click the result table header to sort]
#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID124892207]
Potency 0.3162qHTS for Inhibitors of TGF-b: Cytotox Counterscreen [AID588856, Type: confirmatory]
View
2
[SID50100104]
12Kinase Inhibitor Selectivity Profiling Assay [AID1433_73, Type: confirmatory]tyrosine-protein kinase ABL1 isoform a [Homo sapiens] [gi:62362414]
View
3
[SID50100104]
14Kinase Inhibitor Selectivity Profiling Assay [AID1433_56, Type: confirmatory]platelet-derived growth factor receptor beta precursor [Homo sapiens] [gi:4505683]
View
4
[SID50100104]
14Kinase Inhibitor Selectivity Profiling Assay [AID1433_36, Type: confirmatory]mast/stem cell growth factor receptor Kit isoform 1 precursor [Homo sapiens] [gi:4557695]
View
5
[SID50100104]
15Kinase Inhibitor Selectivity Profiling Assay [AID1433_40, Type: confirmatory]mast/stem cell growth factor receptor Kit isoform 1 precursor [Homo sapiens] [gi:4557695]
View
6
[SID50100104]
15Kinase Inhibitor Selectivity Profiling Assay [AID1433_18, Type: confirmatory]protein-tyrosine kinase [Homo sapiens] [gi:433338]
View
7
[SID50100104]
19Kinase Inhibitor Selectivity Profiling Assay [AID1433_16, Type: confirmatory]macrophage colony-stimulating factor 1 receptor precursor [Homo sapiens] [gi:27262659]
View
8
[SID50100104]
21Kinase Inhibitor Selectivity Profiling Assay [AID1433_98, Type: confirmatory]tyrosine-protein kinase ABL1 isoform a [Homo sapiens] [gi:62362414]
View
9
[SID124892208]
Potency 25.1189qHTS for Inhibitors of TGF-b: Cytotox Counterscreen [AID588856, Type: confirmatory]
View
10
[SID124892209]
Potency 29.5659Cell Proliferation Assay against a hMSC Cell Line [AID651696, Type: confirmatory]
View
11
[SID50100104]
31Kinase Inhibitor Selectivity Profiling Assay [AID1433_55, Type: confirmatory]platelet-derived growth factor receptor alpha precursor [Homo sapiens] [gi:5453870]
View
12
[SID50100104]
35Kinase Inhibitor Selectivity Profiling Assay [AID1433_96, Type: confirmatory]tyrosine-protein kinase ABL1 isoform a [Homo sapiens] [gi:62362414]
View
13
[SID124892209]
Potency 37.2212Cell Proliferation Assay against the TMD8 Cell Line [AID651645, Type: confirmatory]
View
14
[SID124892209]
Potency 37.2212Cell Proliferation Assay against the HBL1 Cell Line [AID651646, Type: confirmatory]
View
15
[SID50100104]
40Kinase Inhibitor Selectivity Profiling Assay [AID1433_89, Type: confirmatory]tyrosine-protein kinase Lck precursor [Homo sapiens] [gi:112789546]
View
16
[SID50100104]
44Kinase Inhibitor Selectivity Profiling Assay [AID1433_99, Type: confirmatory]tyrosine-protein kinase ABL1 isoform a [Homo sapiens] [gi:62362414]
View
17
[SID50100104]
71Kinase Inhibitor Selectivity Profiling Assay [AID1433_39, Type: confirmatory]mast/stem cell growth factor receptor Kit isoform 1 precursor [Homo sapiens] [gi:4557695]
View
18
[SID50100104]
77Kinase Inhibitor Selectivity Profiling Assay [AID1433_95, Type: confirmatory]tyrosine-protein kinase ABL1 isoform a [Homo sapiens] [gi:62362414]
View
19
[SID50100104]
520Kinase Inhibitor Selectivity Profiling Assay [AID1433_74, Type: confirmatory]tyrosine-protein kinase Blk [Homo sapiens] [gi:33469982]
View
20
[SID50100104]
820Kinase Inhibitor Selectivity Profiling Assay [AID1433_37, Type: confirmatory]mast/stem cell growth factor receptor Kit isoform 1 precursor [Homo sapiens] [gi:4557695]
View
21
[SID50100104]
890Kinase Inhibitor Selectivity Profiling Assay [AID1433_90, Type: confirmatory]tyrosine-protein kinase Lyn isoform A [Homo sapiens] [gi:4505055]
View
22
[SID50100104]
1000Kinase Inhibitor Selectivity Profiling Assay [AID1433_129, Type: confirmatory]cyclin-G-associated kinase isoform 1 [Homo sapiens] [gi:157384971]
View
23
[SID50100104]
1400Kinase Inhibitor Selectivity Profiling Assay [AID1433_123, Type: confirmatory]ephrin type-A receptor 8 isoform 1 precursor [Homo sapiens] [gi:10140845]
View
24
[SID50100104]
1500Kinase Inhibitor Selectivity Profiling Assay [AID1433_33, Type: confirmatory]tyrosine-protein kinase FRK [Homo sapiens] [gi:4503787]
View
25
[SID50100104]
1700Kinase Inhibitor Selectivity Profiling Assay [AID1433_92, Type: confirmatory]RAF proto-oncogene serine/threonine-protein kinase [Homo sapiens] [gi:4506401]
View
26
[SID50100104]
1900Kinase Inhibitor Selectivity Profiling Assay [AID1433_138, Type: confirmatory]maternal embryonic leucine zipper kinase isoform 1 [Homo sapiens] [gi:7661974]
View
27
[SID50100104]
2100Kinase Inhibitor Selectivity Profiling Assay [AID1433_15, Type: confirmatory]dual specificity protein kinase CLK4 [Homo sapiens] [gi:10190706]
View
28
[SID50100104]
2400Kinase Inhibitor Selectivity Profiling Assay [AID1433_86, Type: confirmatory]tyrosine-protein kinase Fgr [Homo sapiens] [gi:4885235]
View
29
[SID50100104]
2600Kinase Inhibitor Selectivity Profiling Assay [AID1433_94, Type: confirmatory]mitogen-activated protein kinase kinase kinase MLT isoform 2 [Homo sapiens] [gi:19526767]
View
30
[SID50100104]
2900Kinase Inhibitor Selectivity Profiling Assay [AID1433_38, Type: confirmatory]mast/stem cell growth factor receptor Kit isoform 1 precursor [Homo sapiens] [gi:4557695]
View
31
[SID50100104]
3100Kinase Inhibitor Selectivity Profiling Assay [AID1433_135, Type: confirmatory]mitogen-activated protein kinase 10 isoform 1 [Homo sapiens] [gi:4506081]
View
32
[SID50100104]
3100Kinase Inhibitor Selectivity Profiling Assay [AID1433_87, Type: confirmatory]tyrosine-protein kinase Fyn isoform b [Homo sapiens] [gi:23510362]
View
33
[SID50100104]
3300Kinase Inhibitor Selectivity Profiling Assay [AID1433_76, Type: confirmatory]serine/threonine-protein kinase B-raf [Homo sapiens] [gi:33188459]
View
34
[SID50100104]
4300Kinase Inhibitor Selectivity Profiling Assay [AID1433_93, Type: confirmatory]serine/threonine-protein kinase TNNI3K [Homo sapiens] [gi:7705748]
View
35
[SID50100104]
4500Kinase Inhibitor Selectivity Profiling Assay [AID1433_14, Type: confirmatory]clk1 [gi:632964]
View
36
[SID50100104]
5000Kinase Inhibitor Selectivity Profiling Assay [AID1433_134, Type: confirmatory]mitogen-activated protein kinase 8 isoform alpha1 [Homo sapiens] [gi:4506095]
View
37
[SID50100104]
5300Kinase Inhibitor Selectivity Profiling Assay [AID1433_188, Type: confirmatory]serine/threonine-protein kinase 17A [Homo sapiens] [gi:109255245]
View
38
[SID50100104]
5500Kinase Inhibitor Selectivity Profiling Assay [AID1433_10, Type: confirmatory]cyclin-dependent kinase 19 [Homo sapiens] [gi:30387611]
View
39
[SID50100104]
7600Kinase Inhibitor Selectivity Profiling Assay [AID1433_80, Type: confirmatory]epidermal growth factor receptor isoform a precursor [Homo sapiens] [gi:29725609]
View
40
[SID50100104]
7800Kinase Inhibitor Selectivity Profiling Assay [AID1433_179, Type: confirmatory]Sak [Homo sapiens] [gi:16215696]
View
41
[SID103245522]
Kd Average Binding Constant for CSNK1G1 ; NA=Not Active at 10 uM [AID256655, Type: Literature]Casein kinase I isoform gamma-1 [gi:18202957]
View
42
[SID29215405]
Potency qHTS Assay for Inhibitors Targeting the Menin-MLL Interaction in MLL Related Leukemias: Competition With Texas Red Labeled MLL-derived Mutant Peptide [AID1768, Type: confirmatory]menin isoform 1 [Homo sapiens] [gi:18860839]
View
43
[SID29215405]
Potency qHTS Assay for Inhibitors Targeting the Menin-MLL Interaction in MLL Related Leukemias: Competition With Fluorescein Labeled MLL-derived Peptide [AID1766, Type: confirmatory]menin isoform 1 [Homo sapiens] [gi:18860839]
View
44
[SID103245522]
Kd Average Binding Constant for MYLK2 ; NA=Not Active at 10 uM [AID256623, Type: Literature]Myosin light chain kinase 2, skeletal/cardiac muscle [gi:24211884]
View
45
[SID103245522]
Kd Average Binding Constant for Aurora3 ; NA=Not Active at 10 uM [AID256610, Type: Literature]Aurora kinase C [gi:27805738]
View
46
[SID103245522]
Kd Average Binding Constant for Aurora2 ; NA=Not Active at 10 uM [AID256613, Type: Literature]Aurora kinase A [gi:27923855]
View
47
[SID103245522]
Kd Average Binding Constant for EPHB4 ; NA=Not Active at 10 uM [AID256559, Type: Literature]Ephrin type-B receptor 4 [gi:19860819]
View
48
[SID103245522]
Kd Average Binding Constant for PIM2 ; NA=Not Active at 10 uM [AID256570, Type: Literature]Serine/threonine-protein kinase pim-2 [gi:20139243]
View
49
[SID103245522]
Kd Average Binding Constant for HCK ; NA=Not Active at 10 uM [AID256629, Type: Literature]Tyrosine-protein kinase HCK [gi:20141296]
View
50
[SID29215405]
Potency qHTS Assay for Inhibitors of Tyrosyl-DNA Phosphodiesterase (TDP1) [AID485290, Type: confirmatory]Chain A, Crystal Structure Of Human Tyrosyl-Dna Phosphodiesterase (Tdp1) [gi:20150581]
View