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Dopamine (CID 681) - Compound BioActivity Data
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Filters: All Data » Ki      
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BioActivity Outcomes:
Active(84)
 
 
Inconclusive(4)
 
 
Unspecified(14)
 
 
Top Targets:
7TM GPCR Srsx(27)
 
 
7TM GPCR Srx(10)
 
 
 
 
FAM101(2)
 
 
MFS(2)
 
 
SLC6sbd DAT1(1)
 
 
BioAssay Types:
Literature(98)
 
 
 
 
BioActivity Types:
Ki(102)
 
 
 
 
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Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 102    Data Row: 102   Total Pages: 3   Display: Page     
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID103167911]
Ki 0.0012Binding Affinity was tested on the high affinity site of Dopamine receptor D4.4 [AID64028, Type: Literature]D(4) dopamine receptor [gi:1345939]
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2
[SID103167911]
Ki 0.0018Binding Affinity on high Affinity Site of Bovine dopamine receptor D2. Tested for ability to displace the radioligand [3H]pramipexole was tested [AID62319, Type: Literature]
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3
[SID103167911]
Ki 0.00189Displacement of [3H]quinpirole from human dopamine D2A receptors expressed in LtK cells [AID61612, Type: Literature]D(2) dopamine receptor [gi:118206]
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4
[SID103167911]
Ki 0.00189Displacement of [3H]quinpirole from Dopamine receptor D2 [AID63075, Type: Literature]
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5
[SID103167911]
Ki 0.0029Displacement of [3H]spiperone from human dopamine D2 receptor at high affinity state expressed in HEK293 cells [AID458633, Type: Literature]D(2) dopamine receptor [gi:118206]
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6
[SID103167911]
Ki 0.0062Displacement of [3H]spiperone from human D4 receptor expressed in CHO cells [AID388670, Type: Literature]D(4) dopamine receptor [gi:1345939]
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7
[SID103167911]
Ki 0.007Binding Affinity was tested on High Affinity Site of Bovine Dopamine receptor D1. Tested for ability to displace the radioligand [3H]-SCH- 23390 [AID63176, Type: Literature]
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8
[SID103167911]
Ki 0.0089Displacement of [3H]spiperone from human dopamine D4.4 receptor expressed in CHO cells [AID733805, Type: Literature]
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9
[SID103167911]
Ki 0.011Binding Affinity was tested on high Affinity Site of Bovine Dopamine D2 Receptor. Tested for ability to displace the radioligand [3H]spiperone was tested [AID42820, Type: Literature]
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10
[SID103167911]
Ki 0.011Binding affinity which represents concentration giving half-maximal inhibition of [3H]7-OH-DPAT binding to Dopamine receptor D3 in rat tissue homogenate [AID65613, Type: Literature]
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11
[SID103167911]
Ki 0.0132Displacement of [3H]raclopride from Dopamine receptor D3 [AID65128, Type: Literature]D(3) dopamine receptor [gi:1169206]
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12
[SID103167911]
Ki 0.0149Inhibition of [3H]YM-09151-2 binding to bovine retina membrane Dopamine receptor D2, high affinity site [AID64172, Type: Literature]D(2) dopamine receptor [gi:118205]
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13
[SID103167911]
Ki 0.015In vitro affinity against Dopamine receptor D2 using [3H]DP-5,6-ADTN radioligand in rat striatal homogenate. [AID65716, Type: Literature]
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14
[SID103167911]
Ki 0.015Binding affinity for dopamine D4-like receptor labelled with [3H]YM-09151-2 in retina [AID63853, Type: Literature]
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15
[SID103167911]
Ki 0.015Displacement of [3H]raclopride from human D3 receptor expressed in HEK293 cells [AID675148, Type: Literature]D(3) dopamine receptor [gi:1169206]
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16
[SID103167911]
Ki 0.017Binding Affinity on High Affinity Site of Dopamine receptor D2S [AID64658, Type: Literature]D(2) dopamine receptor [gi:118206]
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17
[SID103167911]
Ki 0.02Binding affinity on High Affinity Site of Dopamine receptor D2L [AID64329, Type: Literature]D(2) dopamine receptor [gi:118206]
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18
[SID103167911]
Ki 0.02Displacement of [3H]YM-09151-2 from human dopamine D3 receptor expressed in CHOp cells [AID709660, Type: Literature]D(3) dopamine receptor [gi:1169206]
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19
[SID103167911]
Ki 0.021Displacement of [3H]spiperone from human dopamine D3 receptor expressed in CHO cells [AID733801, Type: Literature]D(3) dopamine receptor [gi:1169206]
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20
[SID103167911]
Ki 0.034Binding Affinity was tested on relative proportion of High Affinity Site of Dopamine receptor D2S [AID64659, Type: Literature]
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21
[SID103167911]
Ki 0.034High binding affinity for dopamine D-2 receptor from bovine anterior pitutary membrane, using radioligand [3H]spiroperidol [AID62339, Type: Literature]
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22
[SID103167911]
Ki 0.036Binding Affinity was tested on relative proportion of High Affinity Site of Bovine dopamine receptor D1. Tested for ability to displace the radioligand [3H]-SCH- 23390 at the binding site. [AID63178, Type: Literature]
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23
[SID103167911]
Ki 0.042Binding Affinity was tested on relative proportion of High Affinity Site of Dopamine receptor D2L [AID64319, Type: Literature]
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24
[SID103167911]
Ki 0.0493Tested for binding affinity against dopamine receptor D3 expressed in Sf9 cells. [AID65625, Type: Literature]
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25
[SID103167911]
Ki 0.05Binding Affinity was tested on the high affinity site of Dopamine receptor D3 [AID64971, Type: Literature]D(3) dopamine receptor [gi:1169206]
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26
[SID103167911]
Ki 0.051Binding Affinity was tested on relative proportion of high Affinity Site of Bovine dopamine receptor D2. Tested for ability to displace the radioligand [3H]spiperone at the binding site. [AID62326, Type: Literature]
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27
[SID103167911]
Ki 0.052Binding Affinity was tested on relative proportion of High Affinity Site of Dopamine receptor D3 [AID64973, Type: Literature]
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28
[SID103167911]
Ki 0.057Binding Affinity was tested on relative proportion of High Affinity Site of Dopamine receptor D4.4 [AID64030, Type: Literature]
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29
[SID103167911]
Ki 0.058Binding of [3H]clonidine to alpha-2-adrenergic receptor of rat cerebral cortical membranes [AID219797, Type: Literature]
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30
[SID103167911]
Ki 0.062Binding Affinity was tested on low Affinity Site of Dopamine receptor D4.4 [AID64029, Type: Literature]
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31
[SID103167911]
Ki 0.072Displacement of [3H]spiperone from human wild type D3 receptor expressed in human HEK293 cells [AID388686, Type: Literature]D(3) dopamine receptor [gi:1169206]
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32
[SID103167911]
Ki 0.097Binding Affinity was determined in the presence of 100 micro M Gpp(NH)p for decoupling of the ternary complex of Compound to Dopamine receptor D4.4 [AID64027, Type: Literature]
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33
[SID103167911]
Ki 0.11Displacement of [3H]spiperone from human dopamine D2short receptor expressed in CHO cells [AID733804, Type: Literature]D(2) dopamine receptor [gi:118206]
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34
[SID103167911]
Ki 0.124Displacement of [3H]SCH23390 from dopamine D1 receptor expressed in Ltk deficient fibroblast cells by liquid scintillation counting [AID427225, Type: Literature]
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35
[SID103167911]
Ki 0.13Binding affinity against cloned human Dopamine receptor D1 using [125I]-SCH 23982 as radioligand transfected in HEK cells [AID63344, Type: Literature]
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36
[SID103167911]
Ki 0.13Binding affinity for dopamine D2-D3 like receptor labelled with [3H]YM-09151-2 in striatum [AID64302, Type: Literature]
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37
[SID103167911]
Ki 0.15Displacement of [3H]fenoldopam from Dopamine receptor D1 of rat striatum membranes [AID61510, Type: Literature]D(1A) dopamine receptor [gi:118229]
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38
[SID103167911]
Ki 0.19Displacement of [3H]spiperone from human dopamine D2long receptor expressed in CHO cells [AID733806, Type: Literature]D(2) dopamine receptor [gi:118206]
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39
[SID103167911]
Ki 0.192Binding affinity to displace [3H]- SCH 23390 against Dopamine receptor D1 [AID61822, Type: Literature]
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40
[SID103167911]
Ki 0.197Displacement of [3H]raclopride from rat dopamine D2short receptor expressed in CHO-K1 cells by liquid scintillation counting [AID427139, Type: Literature]D(2) dopamine receptor [gi:47117674]
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41
[SID103167911]
Ki 0.24Displacement of [3H]spiperone from human D3 receptor expressed in CHO cells [AID388669, Type: Literature]D(3) dopamine receptor [gi:1169206]
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42
[SID103167911]
Ki 0.26Binding affinity against cloned human Dopamine receptor D2 using [3H]spiperone as radioligand transfected in HEK cells [AID62918, Type: Literature]
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43
[SID103167911]
Ki 0.29Binding Affinity was determined in the presence of 100 micro M Gpp(NH)p for decoupling of the ternary complex of Compound to Dopamine receptor D3 [AID64970, Type: Literature]
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44
[SID103167911]
Ki 0.296Inhibitory constant against binding of [125I]- IBZM to rat striatal membrane [AID65881, Type: Literature]
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45
[SID103167911]
Ki 0.36Displacement of [3H]spiperone from human D2short receptor expressed in CHO cells [AID388668, Type: Literature]D(2) dopamine receptor [gi:118206]
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46
[SID103167911]
Ki 0.422Displacement of [3H]YM-09151-2 from human dopamine D2 receptor expressed in CHOp cells [AID709659, Type: Literature]D(2) dopamine receptor [gi:118206]
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47
[SID103167911]
Ki 0.44Displacement of [3H]SCH23390 from dopamine D1 receptor in bovine striatum [AID733807, Type: Literature]D(1A) dopamine receptor [gi:110832828]
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48
[SID103167911]
Ki 0.45Displacement of [3H]spiperone from human D2long receptor expressed in CHO cells [AID388667, Type: Literature]D(2) dopamine receptor [gi:118206]
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49
[SID103167911]
Ki 0.572Inhibition of [3H]raclopride binding to Dopamine receptor D2 [AID63076, Type: Literature]D(2) dopamine receptor [gi:118206]
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50
[SID103167911]
Ki 0.617Tested for binding affinity against Dopamine receptor D2 like from bovine striatum membranes by using [3H]YM-09151-2 radioligand [AID64170, Type: Literature]D(2) dopamine receptor [gi:118205]
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