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Estradiol (CID 5757) - Compound BioActivity Data
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Filters: All Data » Ki      
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BioActivity Outcomes:
Active(24)
 
 
Unspecified(1)
 
 
Top Targets:
NR LBD ER(15)
 
 
Sulfotransfer..(2)
 
 
KAZAL SLC21(1)
 
 
BioAssay Types:
Literature(25)
 
 
 
BioActivity Types:
Ki(25)
 
 
 
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Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 19    Data Row: 25   Total Pages: 2   Display: Page     
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID103189263]
Ki 0.000113Apparent inhibition constant for estrogen receptor in Human Breast cancer cytosol in 2.5%DMF [AID68905, Type: Literature]Estrogen receptor beta [gi:6166154]
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2
[SID103189263]
Ki 0.000113Apparent inhibition constant for estrogen receptor in Human Breast cancer cytosol in 2.5%DMF [AID68905, Type: Literature]Estrogen receptor [gi:544257]
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3
[SID103189263]
Ki 0.00012Apparent inhibition constant for estrogen receptor in Human uterine cytosol in 3.3%ethanol [AID68909, Type: Literature]Estrogen receptor [gi:544257]
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4
[SID103189263]
Ki 0.00012Apparent inhibition constant for estrogen receptor in Human uterine cytosol in 3.3%ethanol [AID68909, Type: Literature]Estrogen receptor beta [gi:6166154]
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5
[SID103189263]
Ki 0.000138Inhibition of estradiol binding to estrogen receptor in Human Breast cancer cytosol (3.3% ethanol) [AID68906, Type: Literature]Estrogen receptor [gi:544257]
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6
[SID103189263]
Ki 0.000138Inhibition of estradiol binding to estrogen receptor in Human Breast cancer cytosol (3.3% ethanol) [AID68906, Type: Literature]Estrogen receptor beta [gi:6166154]
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7
[SID103189263]
Ki 0.00016Displacement of [2,4,6,7-3H]estradiol from human ERalpha expressed in HeLa cells after 18 hrs by liquid scintillation counting [AID497602, Type: Literature]Estrogen receptor [gi:544257]
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8
[SID103189263]
Ki 0.000181Apparent inhibition constant for estrogen receptor in Human uterine cytosol in 2.5%DMF [AID68908, Type: Literature]Estrogen receptor [gi:544257]
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9
[SID103189263]
Ki 0.000181Apparent inhibition constant for estrogen receptor in Human uterine cytosol in 2.5%DMF [AID68908, Type: Literature]Estrogen receptor beta [gi:6166154]
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10
[SID103189263]
Ki 0.0003Displacement of E2-Alexa633 from GFP-tagged ERalpha expressed in COS7 cells by FACS [AID503066, Type: Literature]
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11
[SID103189263]
Ki 0.00038Displacement of E2-Alexa633 from GFP-tagged ERbeta expressed in COS7 cells by FACS [AID503067, Type: Literature]
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12
[SID103189263]
Ki 0.00038Binding affinity for human estrogen receptor [AID68900, Type: Literature]Estrogen receptor [gi:544257]
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13
[SID103189263]
Ki 0.00038Binding affinity for human estrogen receptor [AID68900, Type: Literature]Estrogen receptor beta [gi:6166154]
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14
[SID103189263]
Ki 0.002Displacement of [3H]estradiol from full length biotinylated human ERalpha by scintillation proximity assay [AID387083, Type: Literature]Estrogen receptor [gi:544257]
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15
[SID103189263]
Ki 0.002Displacement of [3H]estradiol from full length biotinylated human ERbeta by scintillation proximity assay [AID387084, Type: Literature]Estrogen receptor beta [gi:6166154]
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16
[SID103189263]
Ki 0.0022Ability to displace [3H]17-beta-estradiol from Estrogen receptor alpha by scintillation proximity assay. [AID70345, Type: Literature]
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17
[SID103189263]
Ki 0.0035Ability to displace [3H]17-beta-estradiol from Estrogen receptor beta by scintillation proximity assay. [AID70656, Type: Literature]
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18
[SID103189263]
Ki 0.0057Displacement of E2-Alexa633 from GFP-tagged GPR30 expressed in COS7 cells by FACS [AID503065, Type: Literature]
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19
[SID103189263]
Ki 0.0057Inhibition of estrogen binding to GPR30 (unknown origin) [AID769552, Type: Literature]G-protein coupled estrogen receptor 1 [gi:3023539]
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20
[SID103189263]
Ki 0.012Binding affinity to ERalpha [AID307129, Type: Literature]
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