Bookmark and Share
imatinib (CID 5291) - Compound BioActivity Data
.
Filters: All Data » Ki      
Filter selected
BioActivity Outcomes:
Active(13)
 
 
Inconclusive(1)
 
 
Top Targets:
PTKc Abl(3)
 
 
PTKc Src(3)
 
 
PKc like(2)
 
 
Flavodoxin 2(1)
 
 
BioAssay Types:
Literature(14)
 
 
 
BioActivity Types:
Ki(14)
 
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 13    Data Row: 14   Total Pages: 1   
Sort: [Click the result table header to sort]
#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID103245522]
Ki 3.08e-08Inhibition of PTK [AID442505, Type: Literature]
View
2
[SID103245522]
Ki 0.013Inhibition of human recombinant Abl [AID317426, Type: Literature]Tyrosine-protein kinase ABL1 [gi:85681908]
View
3
[SID103245522]
Ki 0.013Inhibition of human recombinant Abl by filter-binding assay [AID370599, Type: Literature]Tyrosine-protein kinase ABL1 [gi:85681908]
View
4
[SID103245522]
Ki 0.013Inhibition of human recombinant c-Abl by filter-binding assay [AID595769, Type: Literature]Tyrosine-protein kinase ABL1 [gi:85681908]
View
5
[SID103245522]
Ki 0.014Inhibition of Bcr-Abl [AID512579, Type: Literature]
View
6
[SID103245522]
Ki 0.037Inhibition of unphosphorylated Abl [AID513122, Type: Literature]
View
7
[SID46393540]
Ki 5Experimentally measured binding affinity data (Ki) for protein-ligand complexes derived from PDB [AID977610, Type: Literature]Chain A, Crystal Structure Of The Syk Tyrosine Kinase Domain With Gleevec [gi:56554455]
View
8
[SID46393540]
Ki 5Experimentally measured binding affinity data (Ki) for protein-ligand complexes derived from PDB [AID977610, Type: Literature]Chain A, Crystal Structure Of The Syk Tyrosine Kinase Domain With Gleevec [gi:56554455]
View
9
[SID103245522]
Ki 7Inhibition of phosphorylated Abl [AID513123, Type: Literature]
View
10
[SID103245522]
Ki 14.3Inhibition of CYP3A4-mediated midazolam 1'-hydroxylation [AID705603, Type: Literature]
View
11
[SID103245522]
Ki 31Inhibition of human recombinant c-Src by filter-binding assay [AID595768, Type: Literature]Proto-oncogene tyrosine-protein kinase Src [gi:125711]
View
12
[SID103245522]
Ki 31Inhibition of recombinant human c-Src [AID317425, Type: Literature]Proto-oncogene tyrosine-protein kinase Src [gi:125711]
View
13
[SID103245522]
Ki 31Inhibition of human recombinant c-Src by filter-binding assay [AID370598, Type: Literature]Proto-oncogene tyrosine-protein kinase Src [gi:125711]
View
14
[SID103245522]
Ki Inhibition of human recombinant NQO2-mediated mitomycin C metabolism using NADH as cosubstrate incubated for 5 mins prior to NADH addition measured after 30 mins by spectrophotometric analysis [AID719846, Type: Literature]Ribosyldihydronicotinamide dehydrogenase [quinone] [gi:317373581]
View